NO20065339L - Cholinesteraseinhibitorer i liposomer og deres fremstilling og anvendelse - Google Patents

Cholinesteraseinhibitorer i liposomer og deres fremstilling og anvendelse

Info

Publication number
NO20065339L
NO20065339L NO20065339A NO20065339A NO20065339L NO 20065339 L NO20065339 L NO 20065339L NO 20065339 A NO20065339 A NO 20065339A NO 20065339 A NO20065339 A NO 20065339A NO 20065339 L NO20065339 L NO 20065339L
Authority
NO
Norway
Prior art keywords
liposomes
topical
active ingredient
cutaneous
relates
Prior art date
Application number
NO20065339A
Other languages
English (en)
Inventor
Eberhard Pirich
Werner Frantsits
Angelika Bodenteich
Josef Bockmann
Andreas Wagner
Karola Vorauer-Uhl
Original Assignee
Sanochemia Pharmazeutika Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanochemia Pharmazeutika Ag filed Critical Sanochemia Pharmazeutika Ag
Publication of NO20065339L publication Critical patent/NO20065339L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/127—Liposomes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Abstract

Oppfinnelsen vedrører en farmasøytisk sammensetning basert på en aktiv ingrediens som er innelukket i liposomer for topikal, transdermal påføring. Det indre av nevnte liposomer omfatter et surt, vandig medium som inneholder minst en kolinesterasehemmer, helst fra gruppen som inneholder donepezil, rivastigmin, galantamin, fysostigmin, heptylfysostigmin, fenserin, tolserin, cymserin, tiatolserin, tiacymserin, neostigmin, huperzin, takrin, metrifonat og diklorvos eller en enantiomer eller derivat av minst en av nevnte forbindelser. I tillegg vedrører oppfinnelsen en fremgangsmåte for å produsere nevnte sammensetning, valgfritt i en steril form og også anvendelsen av liposomene som er ladet med den aktive ingrediensen i forskjellige galeniske formuleringer for topikal, transdermal bruk med en depoteffekt i epidermisen, for profylaksen og/eller behandling av kutan neuropatisk smerte eller tapet av kutanøs sensorisk funksjon som et resultat av neuropati.
NO20065339A 2004-04-22 2006-11-21 Cholinesteraseinhibitorer i liposomer og deres fremstilling og anvendelse NO20065339L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT0069604A AT500143A1 (de) 2004-04-22 2004-04-22 Cholinesterase-inhibitoren in liposomen sowie deren herstellung und verwendung
PCT/AT2005/000138 WO2005102268A2 (de) 2004-04-22 2005-04-21 Cholinesterase-inhibitoren in liposomen sowie deren herstellung und verwendung

Publications (1)

Publication Number Publication Date
NO20065339L true NO20065339L (no) 2007-01-09

Family

ID=35197479

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20065339A NO20065339L (no) 2004-04-22 2006-11-21 Cholinesteraseinhibitorer i liposomer og deres fremstilling og anvendelse

Country Status (10)

Country Link
US (1) US20080031935A1 (no)
EP (1) EP1737426A2 (no)
JP (1) JP2007533666A (no)
CN (1) CN1946377A (no)
AT (1) AT500143A1 (no)
AU (1) AU2005235430A1 (no)
CA (1) CA2563861A1 (no)
NO (1) NO20065339L (no)
RU (1) RU2006141254A (no)
WO (1) WO2005102268A2 (no)

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US20060264455A1 (en) 2005-05-23 2006-11-23 Schachter Steven C Use of huperzine for disorders
DE102006056783A1 (de) * 2006-12-01 2008-06-05 Lts Lohmann Therapie-Systeme Ag Zubereitung zur transdermalen Verabreichung von Galanthamin
TWI428135B (zh) * 2007-03-26 2014-03-01 Hirofumi Takeuchi And a carrier composition for quick-acting nucleic acid delivery
CN103370055B (zh) * 2011-03-25 2015-06-24 泰尔茂株式会社 缓释性脂质体组合物及其制造方法
JP5848511B2 (ja) * 2011-03-29 2016-01-27 株式会社コーセー リポソーム組成物、並びにそれを用いた化粧料、皮膚外用剤及びその製造方法
CN102178680B (zh) * 2011-04-24 2012-09-05 浙江现代中药与天然药物研究院有限公司 一种长效高含量的石杉碱甲贴片及其制备方法
US9685730B2 (en) 2014-09-12 2017-06-20 Steelcase Inc. Floor power distribution system
GB2561157A (en) * 2017-03-27 2018-10-10 Univ Oxford Innovation Ltd Compartmentalised gel matrix and method of production
KR102046355B1 (ko) * 2018-02-08 2019-11-19 국방과학연구소 피하주사용 피소스티그민의 서방출성 리포좀 제제 및 이의 제조 방법
EP3826615A4 (en) * 2018-07-24 2022-05-04 Taiwan Liposome Company, Ltd. DELAYED RELEASE PHARMACEUTICAL COMPOSITIONS WITH A THERAPEUTIC AGENT FOR THE TREATMENT OF DEMENTIA AND USES THEREOF
TWI767133B (zh) * 2018-08-02 2022-06-11 台灣微脂體股份有限公司 含有治療憂鬱症或焦慮症之治療劑的緩釋組合物及其用途
WO2020033195A1 (en) * 2018-08-08 2020-02-13 Taiwan Liposome Co., Ltd. Sustained-release pharmaceutical compositions comprising an antipsychotic drug and uses thereof

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EP0152379A3 (de) * 1984-02-15 1986-10-29 Ciba-Geigy Ag Verfahren zur Herstellung von pharmazeutischen Zusammensetzungen enthaltend unilamellare Liposomen
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Also Published As

Publication number Publication date
EP1737426A2 (de) 2007-01-03
US20080031935A1 (en) 2008-02-07
WO2005102268A2 (de) 2005-11-03
AU2005235430A1 (en) 2005-11-03
JP2007533666A (ja) 2007-11-22
CN1946377A (zh) 2007-04-11
RU2006141254A (ru) 2008-05-27
AT500143A1 (de) 2005-11-15
CA2563861A1 (en) 2005-11-03
WO2005102268A3 (de) 2006-04-06

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