NO20062618L - Bicykliske pyrazolyl og imidazolylforbindelser og andvendelse derav - Google Patents

Bicykliske pyrazolyl og imidazolylforbindelser og andvendelse derav

Info

Publication number
NO20062618L
NO20062618L NO20062618A NO20062618A NO20062618L NO 20062618 L NO20062618 L NO 20062618L NO 20062618 A NO20062618 A NO 20062618A NO 20062618 A NO20062618 A NO 20062618A NO 20062618 L NO20062618 L NO 20062618L
Authority
NO
Norway
Prior art keywords
imidazolyl compounds
bicyclic pyrazolyl
compounds
pyrazolyl
bicyclic
Prior art date
Application number
NO20062618A
Other languages
English (en)
Inventor
Philip Albert Carpino
Robert Lee Dow
David Andrew Griffith
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO20062618L publication Critical patent/NO20062618L/no

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P25/36—Opioid-abuse
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Psychology (AREA)
  • Obesity (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Nutrition Science (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

Forbindelse med formel (I) er beskrevet heri. Forbindelsene har vist seg å virke som cannabinoid reseptorligander og er derfor anvendelige ved behandling av sykdommer knyttet til mediering av cannabinoidreseptorer hos dyr.
NO20062618A 2003-11-07 2006-06-07 Bicykliske pyrazolyl og imidazolylforbindelser og andvendelse derav NO20062618L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51828003P 2003-11-07 2003-11-07
PCT/IB2004/003522 WO2005044822A1 (en) 2003-11-07 2004-10-25 Bicyclic pyrazolyl and imidazolyl compounds and uses thereof

Publications (1)

Publication Number Publication Date
NO20062618L true NO20062618L (no) 2006-08-07

Family

ID=34572986

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20062618A NO20062618L (no) 2003-11-07 2006-06-07 Bicykliske pyrazolyl og imidazolylforbindelser og andvendelse derav

Country Status (29)

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US (2) US7151097B2 (no)
EP (1) EP1682554A1 (no)
JP (2) JP4056549B2 (no)
KR (1) KR20060086396A (no)
CN (1) CN1886407A (no)
AP (1) AP2006003601A0 (no)
AR (1) AR046831A1 (no)
AU (1) AU2004286909A1 (no)
BR (1) BRPI0416299A (no)
CA (1) CA2544752A1 (no)
CR (1) CR8387A (no)
DO (1) DOP2004001024A (no)
EA (1) EA009742B1 (no)
EC (1) ECSP066549A (no)
GT (1) GT200400226A (no)
HR (1) HRP20060166A2 (no)
IL (1) IL175283A0 (no)
IS (1) IS8426A (no)
MA (1) MA28151A1 (no)
MX (1) MXPA06005023A (no)
NL (1) NL1027434C2 (no)
NO (1) NO20062618L (no)
OA (1) OA13280A (no)
PA (1) PA8616801A1 (no)
PE (1) PE20050576A1 (no)
TN (1) TNSN06129A1 (no)
TW (2) TW200716135A (no)
WO (1) WO2005044822A1 (no)
ZA (1) ZA200603594B (no)

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US20050288340A1 (en) * 2004-06-29 2005-12-29 Pfizer Inc Substituted heteroaryl- and phenylsulfamoyl compounds
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TNSN06129A1 (fr) 2007-11-15
GT200400226A (es) 2005-09-06
IS8426A (is) 2006-04-21
NL1027434C2 (nl) 2007-11-27
AP2006003601A0 (en) 2006-04-30
DOP2004001024A (es) 2005-05-14
MA28151A1 (fr) 2006-09-01
JP4056549B2 (ja) 2008-03-05
PE20050576A1 (es) 2005-09-14
CN1886407A (zh) 2006-12-27
NL1027434A1 (nl) 2005-05-10
TWI280245B (en) 2007-05-01
EP1682554A1 (en) 2006-07-26
JP2007302685A (ja) 2007-11-22
TW200716135A (en) 2007-05-01
AR046831A1 (es) 2005-12-28
HRP20060166A2 (en) 2006-10-31
EA009742B1 (ru) 2008-04-28
CR8387A (es) 2007-05-30
US7151097B2 (en) 2006-12-19
IL175283A0 (en) 2006-09-05
CA2544752A1 (en) 2005-05-19
EA200600647A1 (ru) 2006-10-27
TW200526669A (en) 2005-08-16
US20070027133A1 (en) 2007-02-01
AU2004286909A1 (en) 2005-05-19
MXPA06005023A (es) 2006-07-06
JP2007510707A (ja) 2007-04-26
KR20060086396A (ko) 2006-07-31
OA13280A (en) 2007-01-31
ZA200603594B (en) 2007-09-26
ECSP066549A (es) 2006-10-17
WO2005044822A1 (en) 2005-05-19
BRPI0416299A (pt) 2007-01-23
US20050101592A1 (en) 2005-05-12
PA8616801A1 (es) 2006-05-16

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