NO20061395L - Nye pyridinderivater - Google Patents
Nye pyridinderivaterInfo
- Publication number
- NO20061395L NO20061395L NO20061395A NO20061395A NO20061395L NO 20061395 L NO20061395 L NO 20061395L NO 20061395 A NO20061395 A NO 20061395A NO 20061395 A NO20061395 A NO 20061395A NO 20061395 L NO20061395 L NO 20061395L
- Authority
- NO
- Norway
- Prior art keywords
- pyridine derivatives
- compounds
- new pyridine
- preparation
- relates
- Prior art date
Links
- 150000003222 pyridines Chemical class 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 3
- 238000002360 preparation method Methods 0.000 abstract 2
- 102000050488 Urotensin II Human genes 0.000 abstract 1
- 108010018369 Urotensin II Proteins 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000002644 neurohormonal effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- HFNHAPQMXICKCF-USJMABIRSA-N urotensin-ii Chemical compound N([C@@H](CC(O)=O)C(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](CC=2C=CC(O)=CC=2)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CC=2C3=CC=CC=C3NC=2)NC(=O)[C@H](CC=2C=CC=CC=2)NC1=O)C(=O)N[C@@H](C(C)C)C(O)=O)C(=O)[C@@H]1CCCN1C(=O)[C@@H](NC(=O)[C@@H](N)CCC(O)=O)[C@@H](C)O HFNHAPQMXICKCF-USJMABIRSA-N 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Ophthalmology & Optometry (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Physical Education & Sports Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Addiction (AREA)
- Reproductive Health (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Obesity (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Gastroenterology & Hepatology (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP0310746 | 2003-09-26 | ||
PCT/EP2004/010559 WO2005030209A1 (fr) | 2003-09-26 | 2004-09-21 | Derives de pyridine et leur utilisation comme antagonistes de l'urotensine ii |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20061395L true NO20061395L (no) | 2006-06-22 |
Family
ID=34384524
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20061395A NO20061395L (no) | 2003-09-26 | 2006-03-27 | Nye pyridinderivater |
Country Status (18)
Country | Link |
---|---|
US (1) | US7750161B2 (fr) |
EP (1) | EP1670470B1 (fr) |
JP (1) | JP4851328B2 (fr) |
KR (1) | KR20070014108A (fr) |
CN (1) | CN1856305B (fr) |
AR (1) | AR045949A1 (fr) |
AT (1) | ATE427748T1 (fr) |
AU (1) | AU2004275488A1 (fr) |
BR (1) | BRPI0414777A (fr) |
CA (1) | CA2540196C (fr) |
DE (1) | DE602004020486D1 (fr) |
IL (1) | IL174497A0 (fr) |
MX (1) | MXPA06003264A (fr) |
NO (1) | NO20061395L (fr) |
RU (1) | RU2006113948A (fr) |
TW (1) | TW200526630A (fr) |
WO (1) | WO2005030209A1 (fr) |
ZA (1) | ZA200602442B (fr) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20050026844A1 (en) | 2003-04-03 | 2005-02-03 | Regents Of The University Of California | Inhibitors for the soluble epoxide hydrolase |
DE10358539A1 (de) * | 2003-12-15 | 2005-07-07 | Merck Patent Gmbh | Carbonsäureamidderivate |
CA2559665A1 (fr) | 2004-03-16 | 2005-09-29 | The Regents Of The University Of California | Reduction de la nephropathie au moyen d'inhibiteurs d'hydrolase d'epoxyde soluble et d'epoxyeicosanoides |
RU2397978C2 (ru) * | 2004-10-12 | 2010-08-27 | Актелион Фармасьютиклз Лтд | 1-[2-(4-бензил-4-гидроксипиперидин-1-ил)-этил]-3-(2-метилхинолин-4-ил)-мочевина в виде кристаллического сульфата |
TW200630337A (en) * | 2004-10-14 | 2006-09-01 | Euro Celtique Sa | Piperidinyl compounds and the use thereof |
CA2584342C (fr) | 2004-10-20 | 2013-04-30 | The Regents Of The University Of California | Inhibiteurs ameliores de l'epoxyde hydrolase soluble |
SE0403084D0 (sv) | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Chemical process |
WO2006135694A2 (fr) * | 2005-06-10 | 2006-12-21 | Acadia Pharmaceuticals Inc. | Composes modulateurs d'uii et utilisation |
TW200808723A (en) | 2006-03-13 | 2008-02-16 | Univ California | Conformationally restricted urea inhibitors of soluble epoxide hydrolase |
WO2007110449A1 (fr) | 2006-03-29 | 2007-10-04 | Euro-Celtique S.A. | Composés de benzènesulfonamide et utilisation de ceux-ci |
TW200812963A (en) * | 2006-04-13 | 2008-03-16 | Euro Celtique Sa | Benzenesulfonamide compounds and the use thereof |
US8791264B2 (en) * | 2006-04-13 | 2014-07-29 | Purdue Pharma L.P. | Benzenesulfonamide compounds and their use as blockers of calcium channels |
AU2007337659A1 (en) * | 2006-12-22 | 2008-07-03 | Actelion Pharmaceuticals Ltd. | 5,6,7,8-tetrahydro-imidazo[1,5-a]pyrazine derivatives |
WO2008124118A1 (fr) | 2007-04-09 | 2008-10-16 | Purdue Pharma L.P. | Composés benzènesulfonylés et leur utilisation |
WO2009040659A2 (fr) * | 2007-09-28 | 2009-04-02 | Purdue Pharma L.P. | Composés benzènesulfonamides et leurs utilisations |
JP2011506466A (ja) | 2007-12-11 | 2011-03-03 | 株式会社サイトパスファインダー | カルボキサミド化合物ならびにケモカイン受容体アゴニストとしてのそれらの使用 |
US9296693B2 (en) | 2010-01-29 | 2016-03-29 | The Regents Of The University Of California | Acyl piperidine inhibitors of soluble epoxide hydrolase |
Family Cites Families (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IE903957A1 (en) | 1989-11-06 | 1991-05-08 | Sanofi Sa | Aromatic amine compounds, their method of preparation and¹pharmaceutical compositions in which they are present |
US6159700A (en) | 1997-01-27 | 2000-12-12 | Smithkline Beecham Corporation | Method of finding agonist and antagonist to human and rat GPR14 |
AUPP003197A0 (en) | 1997-09-03 | 1997-11-20 | Fujisawa Pharmaceutical Co., Ltd. | New heterocyclic compounds |
US6331541B1 (en) * | 1998-12-18 | 2001-12-18 | Soo S. Ko | N-ureidoalkyl-piperidines as modulators of chemokine receptor activity |
KR20010101287A (ko) * | 1998-12-18 | 2001-11-14 | 블레어 큐. 퍼거슨 | 케모킨 수용체 활성의 조절자로서 n-우레이도알킬-피페리딘 |
ATE321751T1 (de) | 1999-07-28 | 2006-04-15 | Kirin Brewery | Harnstoffderivate als ccr-3 rezeptor-inhibitoren |
CA2394603A1 (fr) | 1999-12-21 | 2001-06-28 | Dashyant Dhanak | Antagonistes des recepteurs de l'urotensine ii |
ES2207566T3 (es) | 1999-12-21 | 2004-06-01 | Smithkline Beecham Corporation | Derivados carboxamida de pirrolidina y piperidina como antagonistas del receptor de urotensina-ii. |
ES2225297T3 (es) | 1999-12-21 | 2005-03-16 | Smithkline Beecham Corporation | Antagonistas del receptor de urotensina ii. |
EP1262195A4 (fr) | 2000-03-07 | 2003-05-21 | Takeda Chemical Industries Ltd | Agents vasoactifs |
WO2001098269A2 (fr) * | 2000-06-21 | 2001-12-27 | Bristol-Myers Squibb Pharma Company | N-ureidoalkyl-piperidines utiles comme modulateurs de l'activite du recepteur de chimiokine |
WO2002000606A1 (fr) | 2000-06-28 | 2002-01-03 | Takeda Chemical Industries, Ltd. | Compose biphenyle |
WO2002002530A1 (fr) | 2000-07-04 | 2002-01-10 | Takeda Chemical Industries, Ltd. | Antagoniste de gpr14 |
US20040053963A1 (en) | 2000-12-11 | 2004-03-18 | Dashyant Dhanak | Urotensin-II receptor antagonists |
US20040039017A1 (en) | 2000-12-11 | 2004-02-26 | Dashyant Dhanak | Urotensin-II receptor antagonists |
EP1359915A4 (fr) | 2001-01-26 | 2004-07-21 | Smithkline Beecham | Antagonistes des recepteurs de l'urotensine-ii |
EP1379523B1 (fr) * | 2001-03-27 | 2005-07-27 | Actelion Pharmaceuticals Ltd. | Derives de 1,2,3,4-tetrahydro-isoquinoline en tant qu'antagonistes du recepteur de l'urotensine ii |
JP2004529134A (ja) | 2001-03-29 | 2004-09-24 | スミスクライン・ビーチャム・コーポレイション | ピロリジンスルホンアミド |
JP2004525156A (ja) | 2001-03-29 | 2004-08-19 | スミスクライン・ビーチャム・コーポレイション | ピロリジンスルホンアミド |
JP2004524355A (ja) | 2001-03-29 | 2004-08-12 | スミスクライン・ビーチャム・コーポレイション | ピロリジンスルホンアミド |
US20040152692A1 (en) | 2001-03-29 | 2004-08-05 | Dashyant Dhanak | Pyrrolidine sulfonamides |
EP1385495A4 (fr) | 2001-05-07 | 2005-12-21 | Smithkline Beecham Corp | Sulfonamides |
EP1385830A4 (fr) | 2001-05-07 | 2005-08-17 | Smithkline Beecham Corp | Sulfonamides |
WO2002089793A1 (fr) | 2001-05-07 | 2002-11-14 | Smithkline Beecham Corporation | Sulfonamides |
JP2004535390A (ja) | 2001-05-07 | 2004-11-25 | スミスクライン・ビーチャム・コーポレイション | スルホンアミド |
JP2004529170A (ja) | 2001-05-07 | 2004-09-24 | スミスクライン・ビーチャム・コーポレイション | スルホンアミド |
AR033879A1 (es) | 2001-05-07 | 2004-01-07 | Smithkline Beecham Corp | Compuesto sulfonamida, composicion farmaceutica que lo comprende, su uso para preparar dicha composicion y procedimiento para la obtencion de dicho compuesto |
ES2254772T3 (es) | 2001-12-04 | 2006-06-16 | Actelion Pharmaceuticals Ltd. | 4-(piperidil-y pirrolidil-alquil-ureido)-quinoleinas como receptores antagonistas de urotensina ii. |
WO2004026836A2 (fr) * | 2002-09-17 | 2004-04-01 | Actelion Pharmaceuticals Ltd | Derives de 1-pyridin-4-yl-uree |
AU2003291303A1 (en) | 2002-11-06 | 2004-06-03 | Smithkline Beecham Corporation | Sulfonamides |
AR041885A1 (es) | 2002-11-06 | 2005-06-01 | Smithkline Beecham Corp | Compuesto de sulfonamida, composicion farmaceutica que lo comprende y su uso para preparar dicha composicion |
WO2004043917A1 (fr) | 2002-11-06 | 2004-05-27 | Smithkline Beecham Corporation | Sulfonamides |
WO2004043369A2 (fr) | 2002-11-06 | 2004-05-27 | Smithkline Beecham Corporation | Sulfonamides |
AU2003295408A1 (en) | 2002-11-06 | 2004-06-03 | Smithkline Beecham Corporation | Sulfonamides |
WO2004073634A2 (fr) | 2003-02-20 | 2004-09-02 | Encysive Pharmaceuticals Inc. | Antagonistes du recepteur de l'urotensine-ii de la phenylenediamine et antagonistes du ccr-9 |
US20060211707A1 (en) | 2003-05-07 | 2006-09-21 | Hamed Aissaoui | Piperazine-alkyl-ureido derivatives |
-
2004
- 2004-09-21 EP EP04765436A patent/EP1670470B1/fr active Active
- 2004-09-21 US US10/573,516 patent/US7750161B2/en not_active Expired - Fee Related
- 2004-09-21 BR BRPI0414777-4A patent/BRPI0414777A/pt not_active Application Discontinuation
- 2004-09-21 CN CN2004800277254A patent/CN1856305B/zh not_active Expired - Fee Related
- 2004-09-21 AU AU2004275488A patent/AU2004275488A1/en not_active Abandoned
- 2004-09-21 AT AT04765436T patent/ATE427748T1/de not_active IP Right Cessation
- 2004-09-21 MX MXPA06003264A patent/MXPA06003264A/es unknown
- 2004-09-21 JP JP2006527332A patent/JP4851328B2/ja not_active Expired - Fee Related
- 2004-09-21 KR KR1020067005848A patent/KR20070014108A/ko not_active Application Discontinuation
- 2004-09-21 CA CA2540196A patent/CA2540196C/fr not_active Expired - Fee Related
- 2004-09-21 RU RU2006113948/04A patent/RU2006113948A/ru unknown
- 2004-09-21 DE DE602004020486T patent/DE602004020486D1/de active Active
- 2004-09-21 WO PCT/EP2004/010559 patent/WO2005030209A1/fr active Application Filing
- 2004-09-24 AR ARP040103475A patent/AR045949A1/es unknown
- 2004-09-24 TW TW093129149A patent/TW200526630A/zh unknown
-
2006
- 2006-03-22 IL IL174497A patent/IL174497A0/en unknown
- 2006-03-24 ZA ZA200602442A patent/ZA200602442B/en unknown
- 2006-03-27 NO NO20061395A patent/NO20061395L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
MXPA06003264A (es) | 2006-06-08 |
US20070043081A1 (en) | 2007-02-22 |
CA2540196C (fr) | 2012-03-20 |
CA2540196A1 (fr) | 2005-04-07 |
AU2004275488A1 (en) | 2005-04-07 |
CN1856305A (zh) | 2006-11-01 |
EP1670470B1 (fr) | 2009-04-08 |
JP4851328B2 (ja) | 2012-01-11 |
WO2005030209A8 (fr) | 2006-05-11 |
ZA200602442B (en) | 2007-09-26 |
JP2007506692A (ja) | 2007-03-22 |
EP1670470A1 (fr) | 2006-06-21 |
US7750161B2 (en) | 2010-07-06 |
WO2005030209A1 (fr) | 2005-04-07 |
DE602004020486D1 (de) | 2009-05-20 |
AR045949A1 (es) | 2005-11-16 |
ATE427748T1 (de) | 2009-04-15 |
RU2006113948A (ru) | 2007-11-10 |
IL174497A0 (en) | 2006-08-01 |
CN1856305B (zh) | 2010-04-28 |
KR20070014108A (ko) | 2007-01-31 |
TW200526630A (en) | 2005-08-16 |
BRPI0414777A (pt) | 2006-11-21 |
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