NO20055230L - HIV-integraseinhibitorer - Google Patents
HIV-integraseinhibitorerInfo
- Publication number
- NO20055230L NO20055230L NO20055230A NO20055230A NO20055230L NO 20055230 L NO20055230 L NO 20055230L NO 20055230 A NO20055230 A NO 20055230A NO 20055230 A NO20055230 A NO 20055230A NO 20055230 L NO20055230 L NO 20055230L
- Authority
- NO
- Norway
- Prior art keywords
- optionally
- substituted
- multisubstituted
- het2
- nr8r9
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Tropical Medicine & Parasitology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- AIDS & HIV (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
A, sammen med de to karbonatomer av fenylringen som den er bundet til, danner monocyklisk aryl eller monocyklisk Het2; R1 er hydrogen, halo, nitro, cyano, sultam, sultim, C3.7-cykloalkyl, C(=O)-R5, S(=O)y-R6, OR7, NR8R9, C(=NR8)-R5, valgfritt flersubstituert C^-alkyl, valgfritt flersubsti-tuert C2.6-alkenyl eller valgfritt flersubstituert C2.6-alkynyl; R2 er hydrogen, C3.7-cykloalkyl, aryl, Het1, Het2, C(=O)-R5, S(=O)y-R6, OR7, NR8R9, C (=NR8) -R5 eller valgfritt flersubstituert C^g-alkyl, valgfritt flersubstituert C2.6-alkenyl eller valgfritt flersubstituert C2.6-alkynyl. Anvendelse derav som HIV-integraseinhibitorer, fremgangs-mater for deres fremstilling samt farmasoytiske sammenset-ninger og diagnostiske sett som inneholder dem. Dessuten kombinasjoner derav med andre anti-retrovirale midler og deres anvendelse i assayer som referanseforbindelser eller som reagensmidler.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US46598703P | 2003-04-28 | 2003-04-28 | |
EP03101164 | 2003-04-28 | ||
PCT/EP2004/050621 WO2004096807A2 (en) | 2003-04-28 | 2004-04-27 | Hiv integrase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20055230L true NO20055230L (no) | 2005-11-07 |
Family
ID=33420586
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20055230A NO20055230L (no) | 2003-04-28 | 2005-11-07 | HIV-integraseinhibitorer |
Country Status (13)
Country | Link |
---|---|
US (1) | US20060211724A1 (no) |
EP (1) | EP1625130A2 (no) |
KR (1) | KR20060006047A (no) |
CN (1) | CN1812992A (no) |
AP (1) | AP2005003451A0 (no) |
AR (1) | AR044518A1 (no) |
AU (1) | AU2004234087A1 (no) |
BR (1) | BRPI0409873A (no) |
CA (1) | CA2522990A1 (no) |
MX (1) | MXPA05011726A (no) |
NO (1) | NO20055230L (no) |
TW (1) | TW200507848A (no) |
WO (1) | WO2004096807A2 (no) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200716632A (en) * | 2005-05-16 | 2007-05-01 | Gilead Sciences Inc | Integrase inhibitor compounds |
EP1885722B1 (en) | 2005-05-19 | 2011-11-16 | Merck Canada Inc. | Quinoline derivatives as ep4 antagonists |
AR057455A1 (es) * | 2005-07-22 | 2007-12-05 | Merck & Co Inc | Inhibidores de la transcriptasa reversa de vih y composicion farmaceutica |
WO2007014352A2 (en) * | 2005-07-27 | 2007-02-01 | Gilead Sciences, Inc. | Antiviral phosphonate conjugates for inhibition of hiv |
WO2007076005A2 (en) * | 2005-12-21 | 2007-07-05 | Gilead Sciences, Inc. | Processes and intermediates useful for preparing integrase inhibitor compounds |
CA2651579A1 (en) * | 2006-05-16 | 2007-11-29 | Gilead Sciences, Inc. | Integrase inhibitors |
EP1916249A1 (en) * | 2006-10-10 | 2008-04-30 | LEK Pharmaceuticals D.D. | 3-(benzo[d][1,3]dioxol-5-ylmethyl)-4-(thio)oxo-2-(thio)oxo-azolidin-5-ylidene derivatives as antibacterial agents |
DK2124562T3 (en) | 2007-03-09 | 2016-08-01 | Second Genome Inc | BICYCLOHETEROARYLFORBINDELSER AS P2X7 modulators and uses thereof |
WO2009067541A2 (en) * | 2007-11-20 | 2009-05-28 | Gilead Sciences, Inc. | Integrase inhibitors |
US8993542B2 (en) | 2008-01-25 | 2015-03-31 | Chimerix Inc. | Methods of treating viral infections |
US8815906B2 (en) | 2008-03-19 | 2014-08-26 | Chembridge Corporation | Tyrosine kinase inhibitors |
US9249147B2 (en) | 2008-03-19 | 2016-02-02 | Chembridge Corporation | Tyrosine kinase inhibitors |
MX2011010582A (es) * | 2009-04-09 | 2011-10-19 | Boehringer Ingelheim Int | Inhibidores de la replicacion del vih. |
US8283366B2 (en) | 2010-01-22 | 2012-10-09 | Ambrilia Biopharma, Inc. | Derivatives of pyridoxine for inhibiting HIV integrase |
AU2011216243B2 (en) | 2010-02-12 | 2015-07-09 | Chimerix, Inc. | Nucleoside phosphonate salts |
WO2012037155A2 (en) | 2010-09-13 | 2012-03-22 | Gtx, Inc. | Tyrosine kinase inhibitors |
US10513515B2 (en) | 2017-08-25 | 2019-12-24 | Biotheryx, Inc. | Ether compounds and uses thereof |
CA3106239A1 (en) | 2018-07-27 | 2020-01-30 | Biotheryx, Inc. | Bifunctional compounds as cdk modulators |
EP4143329A2 (en) | 2020-04-28 | 2023-03-08 | Anwita Biosciences, Inc. | Interleukin-2 polypeptides and fusion proteins thereof, and their pharmaceutical compositions and therapeutic applications |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6544732B1 (en) * | 1999-05-20 | 2003-04-08 | Illumina, Inc. | Encoding and decoding of array sensors utilizing nanocrystals |
DE60124577T2 (de) * | 2000-10-12 | 2007-09-27 | Merck & Co., Inc. | Aza- und polyaza-naphthalenylcarbonsäureamide als hiv-integrase-hemmer |
AU2003301439A1 (en) * | 2002-10-16 | 2004-05-04 | Gilead Sciences, Inc. | Pre-organized tricyclic integrase inhibitor compounds |
US7442773B2 (en) * | 2004-01-23 | 2008-10-28 | The Board Of Trustees Of The University Of Illinois | Universal peptide-binding scaffolds and protein chips |
-
2004
- 2004-04-27 EP EP04741485A patent/EP1625130A2/en not_active Withdrawn
- 2004-04-27 CN CNA2004800180526A patent/CN1812992A/zh active Pending
- 2004-04-27 US US10/554,712 patent/US20060211724A1/en not_active Abandoned
- 2004-04-27 BR BRPI0409873-0A patent/BRPI0409873A/pt not_active IP Right Cessation
- 2004-04-27 AP AP2005003451A patent/AP2005003451A0/xx unknown
- 2004-04-27 MX MXPA05011726A patent/MXPA05011726A/es unknown
- 2004-04-27 WO PCT/EP2004/050621 patent/WO2004096807A2/en active Application Filing
- 2004-04-27 AU AU2004234087A patent/AU2004234087A1/en not_active Abandoned
- 2004-04-27 KR KR1020057020004A patent/KR20060006047A/ko not_active Application Discontinuation
- 2004-04-27 CA CA002522990A patent/CA2522990A1/en not_active Abandoned
- 2004-04-28 AR ARP040101446A patent/AR044518A1/es not_active Application Discontinuation
- 2004-04-28 TW TW093111823A patent/TW200507848A/zh unknown
-
2005
- 2005-11-07 NO NO20055230A patent/NO20055230L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
US20060211724A1 (en) | 2006-09-21 |
MXPA05011726A (es) | 2006-01-23 |
CN1812992A (zh) | 2006-08-02 |
KR20060006047A (ko) | 2006-01-18 |
AR044518A1 (es) | 2005-09-14 |
CA2522990A1 (en) | 2004-11-11 |
BRPI0409873A (pt) | 2006-05-16 |
AU2004234087A1 (en) | 2004-11-11 |
TW200507848A (en) | 2005-03-01 |
EP1625130A2 (en) | 2006-02-15 |
WO2004096807A2 (en) | 2004-11-11 |
WO2004096807A3 (en) | 2005-01-06 |
WO2004096807A8 (en) | 2005-09-22 |
AP2005003451A0 (en) | 2005-12-31 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |