NO20054199L - 6-substituerte imidazopyraziner - Google Patents

6-substituerte imidazopyraziner

Info

Publication number
NO20054199L
NO20054199L NO20054199A NO20054199A NO20054199L NO 20054199 L NO20054199 L NO 20054199L NO 20054199 A NO20054199 A NO 20054199A NO 20054199 A NO20054199 A NO 20054199A NO 20054199 L NO20054199 L NO 20054199L
Authority
NO
Norway
Prior art keywords
substituted imidazopyrazines
imidazopyrazines
substituted
gastric
substituents
Prior art date
Application number
NO20054199A
Other languages
English (en)
Other versions
NO20054199D0 (no
Inventor
Gerhard Grundler
Jorg Senn-Bilfinger
Stefan Postius
Wolfgang-Alexander Simon
Wolfgang Kromer
Wilm Buhr
Peter Jan Zimmermann
M Vittoria Chiesa
Andreas Palmer
Christof Brehm
Original Assignee
Altana Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Altana Pharma Ag filed Critical Altana Pharma Ag
Publication of NO20054199D0 publication Critical patent/NO20054199D0/no
Publication of NO20054199L publication Critical patent/NO20054199L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nutrition Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Oppfinnelsen vedrører 6-substituerte imidazopyraziner med formel 1, hvor substituentene og symbolene har betydningene indikert i beskrivelsen. Forbindelsene har gastrisk sekresjonshemming og utmerkede gastriske og intestinale beskyttende virkningsegenskaper.
NO20054199A 2003-02-18 2005-09-09 6-substituerte imidazopyraziner NO20054199L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03003652 2003-02-18
PCT/EP2004/050135 WO2004074289A1 (en) 2003-02-18 2004-02-16 6-substituted imidazopyrazines

Publications (2)

Publication Number Publication Date
NO20054199D0 NO20054199D0 (no) 2005-09-09
NO20054199L true NO20054199L (no) 2005-11-17

Family

ID=32892854

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20054199A NO20054199L (no) 2003-02-18 2005-09-09 6-substituerte imidazopyraziner

Country Status (19)

Country Link
US (1) US20060148796A1 (no)
EP (1) EP1599481A1 (no)
JP (1) JP2006517951A (no)
KR (1) KR20050100396A (no)
CN (1) CN1747956A (no)
AR (1) AR043002A1 (no)
AU (1) AU2004213177A1 (no)
BR (1) BRPI0407390A (no)
CA (1) CA2516021A1 (no)
EA (1) EA200501229A1 (no)
HR (1) HRP20050794A2 (no)
IS (1) IS8015A (no)
MX (1) MXPA05008582A (no)
NO (1) NO20054199L (no)
PL (1) PL376466A1 (no)
RS (1) RS20050619A (no)
TW (1) TW200504068A (no)
WO (1) WO2004074289A1 (no)
ZA (1) ZA200505670B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009507032A (ja) 2005-09-02 2009-02-19 アボット・ラボラトリーズ 新規なイミダゾ系複素環
US20090175852A1 (en) 2006-06-06 2009-07-09 Schering Corporation Imidazopyrazines as protein kinase inhibitors
AR061229A1 (es) * 2006-06-06 2008-08-13 Schering Corp Imidazopirazinas como inhibidores de la proteina quinasa
WO2008059373A1 (en) * 2006-11-17 2008-05-22 Raqualia Pharma Inc. Imidazo [1, 2-a] pyrazine derivatives and their use as acid pump antagonists
GB0716292D0 (en) 2007-08-21 2007-09-26 Biofocus Dpi Ltd Imidazopyrazine compounds
ES2744541T3 (es) 2008-12-08 2020-02-25 Gilead Connecticut Inc Inhibidores de imidazopirazina Syk
HUE030427T2 (en) * 2008-12-08 2017-05-29 Gilead Connecticut Inc Imidazopyrazine Syk inhibitors
EP2545052B1 (en) 2010-03-11 2014-11-12 Gilead Connecticut, Inc. Imidazopyridines syk inhibitors
CN116178295A (zh) * 2023-01-28 2023-05-30 山东亿盛实业股份有限公司 一种苯唑草酮代谢物t283的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4725601A (en) * 1985-06-04 1988-02-16 Fujisawa Pharmaceutical Co., Ltd. Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers
JPH07242666A (ja) * 1994-03-08 1995-09-19 Fujisawa Pharmaceut Co Ltd 複素環化合物
SE9704404D0 (sv) * 1997-11-28 1997-11-28 Astra Ab New compounds
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
CA2436487A1 (en) * 2001-01-30 2002-08-08 Cytopia Pty Ltd. Methods of inhibiting kinases

Also Published As

Publication number Publication date
BRPI0407390A (pt) 2006-02-07
ZA200505670B (en) 2006-04-26
US20060148796A1 (en) 2006-07-06
JP2006517951A (ja) 2006-08-03
IS8015A (is) 2005-09-08
AR043002A1 (es) 2005-07-13
CA2516021A1 (en) 2004-09-02
RS20050619A (en) 2007-09-21
WO2004074289A1 (en) 2004-09-02
EP1599481A1 (en) 2005-11-30
TW200504068A (en) 2005-02-01
EA200501229A1 (ru) 2006-04-28
HRP20050794A2 (en) 2006-12-31
MXPA05008582A (es) 2005-11-04
CN1747956A (zh) 2006-03-15
KR20050100396A (ko) 2005-10-18
AU2004213177A1 (en) 2004-09-02
PL376466A1 (en) 2005-12-27
NO20054199D0 (no) 2005-09-09

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Legal Events

Date Code Title Description
CREP Change of representative

Representative=s name: PLOUGMANN & VINGTOFT, POSTBOKS 1003 SENTRUM, 0104

FC2A Withdrawal, rejection or dismissal of laid open patent application