NO20052727L - Tetrahydrokinolinderivater - Google Patents
TetrahydrokinolinderivaterInfo
- Publication number
- NO20052727L NO20052727L NO20052727A NO20052727A NO20052727L NO 20052727 L NO20052727 L NO 20052727L NO 20052727 A NO20052727 A NO 20052727A NO 20052727 A NO20052727 A NO 20052727A NO 20052727 L NO20052727 L NO 20052727L
- Authority
- NO
- Norway
- Prior art keywords
- alkoxy
- alkylamino
- heterocycloalkyl
- derivatives
- heteroaryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Foreliggende oppfinnelse omhandler telrahydrokinolinderivater sonn har generell R3 fornnel (I) Formel I eller et farmasøytisk akseptabelt salt derav, hvor R^ og R^ er H eller Me; R' er H, hydroksy, (1-4C)alkoksy, (di)(1-4C)alkylamino(2-4C)alkoksy eller (2- 6)heterocykloalkyl(2-4C)alkoksy; R'' er H, OH, (1-4C)alkoksy eller R^; R^ er H, OH, (1 -4C)alkoksy eller R^med det forbehold at hvis R" er H, er R^ ikke H, OH eller (1- 4C)alkoksy og at hvis R^ er H, er R"* ikke H, OH eller (1-4C)alkoksy; R^ er (2- 5C)heteroaryl, (6C)aryl, (3-8C)cykloalkyl, (2-6C)heterocykloalkyl eller (1-6C)alkyl; r'^ er amino, (di)(1-4C)alkylamino, (6C)arylkarbonylamino, (6C)arylkarbonyloksy, (2-5C)heteroarylkarbonylamino, (2-5C)heteroarylkarbonyloksy, R^-(2- 4C)alkylamino, R°-(2-4C)alkoksy, R^-metylamino eller R^-metoksy; R^ er hydroksy, amino, (1-4C)alkoksy, (di)(1-4C)alkylamino, (2-6C)heterocykloalkyl, (2- 6C)heterocykloalkylkarbonylamino, (di)(1-4C)alkylaminokarbonylannino, (1- 4C)alkoksykarbonylamino og R^ er aminokarbonyl, (di)(1-4C)alkylaminokarbonyl, (2-5C)heteroaryl eller (6C)aryl. Foreliggende oppfinnelse omhandler også famna- søytiske preparater som omfatter nevnte derivater og anvendelsen av disse deri- vatene for å regulere fertilitet.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US43504002P | 2002-12-20 | 2002-12-20 | |
EP02102866 | 2002-12-20 | ||
PCT/EP2003/051025 WO2004056780A2 (en) | 2002-12-20 | 2003-12-16 | Tetrahydroquinoline derivatives |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20052727D0 NO20052727D0 (no) | 2005-06-07 |
NO20052727L true NO20052727L (no) | 2005-07-13 |
NO330612B1 NO330612B1 (no) | 2011-05-30 |
Family
ID=32683821
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20052727A NO330612B1 (no) | 2002-12-20 | 2005-06-07 | Tetrahydrokinolinderivater, farmasoytisk preparat omfattende slike, slike forbindelser for anvendelse i terapi samt anvendelse av slike for fremstilling av medikament for fruktbarhetsregulering |
Country Status (10)
Country | Link |
---|---|
KR (1) | KR20050084341A (no) |
CO (1) | CO5590903A2 (no) |
DE (1) | DE60326390D1 (no) |
EC (1) | ECSP055871A (no) |
EG (1) | EG24958A (no) |
HK (1) | HK1077577A1 (no) |
HR (1) | HRP20050576A2 (no) |
IS (1) | IS2647B (no) |
MX (1) | MXPA05006767A (no) |
NO (1) | NO330612B1 (no) |
-
2003
- 2003-12-16 KR KR1020057011089A patent/KR20050084341A/ko active IP Right Grant
- 2003-12-16 MX MXPA05006767A patent/MXPA05006767A/es active IP Right Grant
- 2003-12-16 DE DE60326390T patent/DE60326390D1/de not_active Expired - Lifetime
-
2005
- 2005-05-26 IS IS7871A patent/IS2647B/is unknown
- 2005-06-07 NO NO20052727A patent/NO330612B1/no not_active IP Right Cessation
- 2005-06-18 EG EGNA2005000309 patent/EG24958A/xx active
- 2005-06-20 HR HR20050576A patent/HRP20050576A2/hr not_active Application Discontinuation
- 2005-06-20 EC EC2005005871A patent/ECSP055871A/es unknown
- 2005-07-19 CO CO05071364A patent/CO5590903A2/es not_active Application Discontinuation
- 2005-12-28 HK HK05112055.2A patent/HK1077577A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
NO330612B1 (no) | 2011-05-30 |
CO5590903A2 (es) | 2005-12-30 |
IS2647B (is) | 2010-08-15 |
KR20050084341A (ko) | 2005-08-26 |
HRP20050576A2 (en) | 2005-10-31 |
DE60326390D1 (en) | 2009-04-09 |
NO20052727D0 (no) | 2005-06-07 |
IS7871A (is) | 2005-05-26 |
EG24958A (en) | 2011-02-28 |
HK1077577A1 (en) | 2006-02-17 |
ECSP055871A (es) | 2005-09-20 |
MXPA05006767A (es) | 2005-09-08 |
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Legal Events
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MM1K | Lapsed by not paying the annual fees |