NO20051641L - Improved imaging agents comprising barbituric acid derivatives - Google Patents
Improved imaging agents comprising barbituric acid derivativesInfo
- Publication number
- NO20051641L NO20051641L NO20051641A NO20051641A NO20051641L NO 20051641 L NO20051641 L NO 20051641L NO 20051641 A NO20051641 A NO 20051641A NO 20051641 A NO20051641 A NO 20051641A NO 20051641 L NO20051641 L NO 20051641L
- Authority
- NO
- Norway
- Prior art keywords
- imaging
- imaging agents
- barbituric acid
- acid derivatives
- improved imaging
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0497—Organic compounds conjugates with a carrier being an organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/04—X-ray contrast preparations
- A61K49/0433—X-ray contrast preparations containing an organic halogenated X-ray contrast-enhancing agent
- A61K49/0438—Organic X-ray contrast-enhancing agent comprising an iodinated group or an iodine atom, e.g. iopamidol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/041—Heterocyclic compounds
- A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
- A61K51/0459—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Physics & Mathematics (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Optics & Photonics (AREA)
- Pharmacology & Pharmacy (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
Foreliggende oppfinnelsen angår diagnostiske avbildingsmidler for in vivo avbilding. Avbildingsmidlene omfatter et syntetisk barbitursyrederivat merket i 5-posisjon med en avbildingsdel som egner seg for diagnostisk avbilding in vivo. Oppfinnelsen tilveiebringer også fannasøytiske og radiofarmasøytiske sammensetninger som omfatter avbildingsmidlene, sammen med utstyrene for fremstilling av radiofarmasøytika. Videre er det beskrevet chelator -konjugater av barbitursyrederivatet, som egner seg for fremstilling av avbildingsmidler som omfatter et radioaktivt eller paramagnetisk metallion. Avbildingsmidlene er nyttige for diagnostisk avbilding in vivo av forskjellige sykdomstilstander, inkludert aterosklerose.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0223249.4A GB0223249D0 (en) | 2002-10-08 | 2002-10-08 | Improved imaging agents |
PCT/GB2003/004351 WO2004032936A1 (en) | 2002-10-08 | 2003-10-08 | Improved imaging agents comprising barbituric acid derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20051641L true NO20051641L (no) | 2005-06-02 |
Family
ID=9945439
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20051641A NO20051641L (no) | 2002-10-08 | 2005-04-04 | Improved imaging agents comprising barbituric acid derivatives |
Country Status (10)
Country | Link |
---|---|
US (1) | US20060120956A1 (no) |
EP (1) | EP1549317A1 (no) |
JP (1) | JP2006505550A (no) |
CN (1) | CN1720050A (no) |
AU (1) | AU2003273505B2 (no) |
CA (1) | CA2501136A1 (no) |
GB (1) | GB0223249D0 (no) |
NO (1) | NO20051641L (no) |
RU (1) | RU2005109272A (no) |
WO (1) | WO2004032936A1 (no) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102006021495A1 (de) * | 2006-05-09 | 2007-11-15 | Bayer Schering Pharma Ag | Verwendung von perfluoralkylhaltigen Metallkomplexen als Kontrastmittel zur Diagnose der Alzheimer Krankheit |
GB0612333D0 (en) * | 2006-06-21 | 2006-08-02 | Ge Healthcare Ltd | Radiopharmaceutical products |
US10328164B2 (en) | 2006-06-21 | 2019-06-25 | Ge Healthcare Limited | Radiopharmaceutical products |
US8529874B2 (en) * | 2007-05-16 | 2013-09-10 | Ge Healthcare As | Peptide imaging agents |
GB0718386D0 (en) * | 2007-09-21 | 2007-10-31 | Ge Healthcare As | Improved radiopharmaceutical formulation |
GB201115937D0 (en) | 2011-09-14 | 2011-10-26 | Univ Aberdeen | 18F-labelled compounds for use as positron emission imaging agents |
CA3109419A1 (en) * | 2018-08-24 | 2020-02-27 | Xeniopro GmbH | Novel compounds |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3952971A (en) * | 1971-11-09 | 1976-04-27 | The United States Of America As Represented By The Administrator Of The National Aeronautics And Space Administration | Airfoil shape for flight at subsonic speeds |
US3952091A (en) * | 1974-10-23 | 1976-04-20 | Hoffmann-La Roche Inc. | Simultaneous multiple radioimmunoassay |
GB1527416A (en) * | 1976-07-20 | 1978-10-04 | Ciba Geigy Ag | Photopolymerisible diepoxides |
US6472227B1 (en) * | 1986-06-04 | 2002-10-29 | Abbott Laboratories | Barbiturate assay, tracers, immunogens, antibodies and kit |
US5102786A (en) * | 1987-05-21 | 1992-04-07 | Pb Diagnostic Systems, Inc. | Biological diagnostic assay system |
KR100660509B1 (ko) * | 1998-05-15 | 2006-12-22 | 지이 헬쓰케어 리미티드 | 표지된 글루타민 및 라이신 유사체 |
US6656448B1 (en) * | 2000-02-15 | 2003-12-02 | Bristol-Myers Squibb Pharma Company | Matrix metalloproteinase inhibitors |
EP1309579B1 (en) * | 2000-05-30 | 2005-10-12 | Board Of Governors Of Wayne State University | Inhibitors of matrix metalloproteinases |
KR20030061825A (ko) * | 2000-10-26 | 2003-07-22 | 화이자 프로덕츠 인크. | 피리미딘-2,4,6-트리온 메탈로프로테이나제 억제제 |
WO2002034753A2 (en) * | 2000-10-26 | 2002-05-02 | Pfizer Products Inc. | Spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors |
WO2002047701A1 (en) * | 2000-12-12 | 2002-06-20 | Angiolab, Inc. | Composition comprising melissa leaf extract for anti-angiogenic and matrix metalloproteinase inhibitory activity |
GB0115929D0 (en) * | 2001-06-29 | 2001-08-22 | Nycomed Amersham Plc | Solid-phase electrophilic fluorination |
-
2002
- 2002-10-08 GB GBGB0223249.4A patent/GB0223249D0/en not_active Ceased
-
2003
- 2003-10-08 JP JP2004542629A patent/JP2006505550A/ja active Pending
- 2003-10-08 AU AU2003273505A patent/AU2003273505B2/en not_active Expired - Fee Related
- 2003-10-08 EP EP03755663A patent/EP1549317A1/en not_active Withdrawn
- 2003-10-08 CN CN200380105207.5A patent/CN1720050A/zh active Pending
- 2003-10-08 CA CA002501136A patent/CA2501136A1/en not_active Abandoned
- 2003-10-08 WO PCT/GB2003/004351 patent/WO2004032936A1/en active Application Filing
- 2003-10-08 RU RU2005109272/15A patent/RU2005109272A/ru not_active Application Discontinuation
- 2003-10-08 US US10/530,836 patent/US20060120956A1/en not_active Abandoned
-
2005
- 2005-04-04 NO NO20051641A patent/NO20051641L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
RU2005109272A (ru) | 2006-01-27 |
AU2003273505B2 (en) | 2007-04-19 |
GB0223249D0 (en) | 2002-11-13 |
WO2004032936A1 (en) | 2004-04-22 |
US20060120956A1 (en) | 2006-06-08 |
AU2003273505A1 (en) | 2004-05-04 |
EP1549317A1 (en) | 2005-07-06 |
CN1720050A (zh) | 2006-01-11 |
CA2501136A1 (en) | 2004-04-22 |
JP2006505550A (ja) | 2006-02-16 |
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Legal Events
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FC2A | Withdrawal, rejection or dismissal of laid open patent application |