NO20025141L - 13-substituerte milbemycinderivater, fremstilling av slike, og anvendelse av dem mot insekter og andre skadedyr - Google Patents

13-substituerte milbemycinderivater, fremstilling av slike, og anvendelse av dem mot insekter og andre skadedyr

Info

Publication number
NO20025141L
NO20025141L NO20025141A NO20025141A NO20025141L NO 20025141 L NO20025141 L NO 20025141L NO 20025141 A NO20025141 A NO 20025141A NO 20025141 A NO20025141 A NO 20025141A NO 20025141 L NO20025141 L NO 20025141L
Authority
NO
Norway
Prior art keywords
optionally substituted
pests
preparation
against insects
use against
Prior art date
Application number
NO20025141A
Other languages
English (en)
Other versions
NO323751B1 (no
NO20025141D0 (no
Inventor
Akio Saito
Yoko Sugiyama
Toshimitsu Toyama
Toshihiko Nanba
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of NO20025141D0 publication Critical patent/NO20025141D0/no
Publication of NO20025141L publication Critical patent/NO20025141L/no
Publication of NO323751B1 publication Critical patent/NO323751B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Forbindelser med formel (I) og salter derav:. hvor: Rrepresenterer metyl, etyl, isopropyl eller s-butyl; Rrepresenterer hydrogen eller alkyl; R3 representerer hydrogen, eventuelt substituert alkanoyl, eventuelt substituert alkenoyl, eventuelt substituert alkynoyl, alkylsulfonyl eller alkoksy- karbonyl; eller R"og Rsammen med nitrogenatomet som de er bundet til, danner en mettet, eventuelt substituert, 4-til 6-leddet, heterosyklisk ringgruppe; og delen -a-, sammen med karbonatomet som den er bundet til, danner en 3- til 6-leddet sykloalkylgruppe. Disse forbindelser har anthelmintisk, akaricidal og insektdrepende aktivitet.
NO20025141A 2000-04-27 2002-10-25 13-substituerte milbemycinderivater, preparater omfattende disse og anvendelse av dem mot insekter og andre skadedyr NO323751B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000127209 2000-04-27
PCT/JP2001/003656 WO2001083500A1 (en) 2000-04-27 2001-04-26 13-substituted milbemycin derivatives, their preparation and their use against insects and other pests

Publications (3)

Publication Number Publication Date
NO20025141D0 NO20025141D0 (no) 2002-10-25
NO20025141L true NO20025141L (no) 2002-12-16
NO323751B1 NO323751B1 (no) 2007-07-02

Family

ID=18636847

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20025141A NO323751B1 (no) 2000-04-27 2002-10-25 13-substituerte milbemycinderivater, preparater omfattende disse og anvendelse av dem mot insekter og andre skadedyr

Country Status (24)

Country Link
US (1) US6653342B2 (no)
EP (1) EP1276748B1 (no)
KR (1) KR100711931B1 (no)
CN (1) CN1247607C (no)
AR (1) AR029250A1 (no)
AT (1) ATE315573T1 (no)
AU (2) AU5261301A (no)
BR (1) BR0110385A (no)
CA (1) CA2407611A1 (no)
CZ (1) CZ20023565A3 (no)
DE (1) DE60116615T2 (no)
DK (1) DK1276748T3 (no)
ES (1) ES2254400T3 (no)
HK (1) HK1057757A1 (no)
HU (1) HUP0301040A3 (no)
IL (1) IL152449A0 (no)
MX (1) MXPA02010587A (no)
NO (1) NO323751B1 (no)
NZ (1) NZ522247A (no)
PL (1) PL357598A1 (no)
RU (1) RU2226531C1 (no)
TW (1) TWI285206B (no)
WO (1) WO2001083500A1 (no)
ZA (1) ZA200208630B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2464403A1 (en) 2001-10-25 2003-05-01 Sankyo Lifetech Company, Limited Anthelmintic composition
TWI366442B (en) * 2003-07-30 2012-06-21 Novartis Ag Palatable ductile chewable veterinary composition
US20090281175A1 (en) * 2006-09-28 2009-11-12 Galderma S.A. Avermectin compounds and treatment of dermatological disorders in humans therewith
TWI457347B (zh) 2008-12-04 2014-10-21 Merial Ltd 二聚合的阿佛菌素（ａｖｅｒｍｅｃｔｉｎ）及密倍脈心（ｍｉｌｂｅｍｙｃｉｎ）衍生物
EP2512467A1 (en) 2009-12-17 2012-10-24 Merial Limited Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles
BR112014013371B1 (pt) 2011-12-02 2020-04-07 Merial Ltd formulações de moxidectina injetável de ação prolongada e novas formas de cristal de moxidectina
BR112015025875B1 (pt) 2013-04-12 2021-06-29 Zoetis Services Llc Composição injetável estável para o tratamento de uma infecção endoparasitária por helmintos em animais não humanos, composição para o tratamento de uma infecção ou infestação endoparasitária por helmintos em um animal não humano, e uso de doramectina e levamisol, ou um sal farmaceuticamente aceitável do mesmo
US20220142972A1 (en) * 2018-12-21 2022-05-12 ELANCO US, Inc. Parasiticidal formulations and use thereof

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ188459A (en) 1977-10-03 1982-09-07 Merck & Co Inc Derivatives of c-076 compounds and pesticidal compositions
US4201861A (en) 1977-10-03 1980-05-06 Merck & Co., Inc. Acyl derivatives of C-076 compounds
US4206205A (en) 1977-10-03 1980-06-03 Merck & Co., Inc. Monosaccharide and aglycone derivatives of C-076
US4173571A (en) 1977-12-19 1979-11-06 Merck & Co., Inc. 13-Halo and 13-deoxy derivatives of C-076 compounds
US4171314A (en) 1977-12-19 1979-10-16 Merck & Co., Inc. 13-Halo and 13-deoxy C-076 compounds
US4203976A (en) 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4200581A (en) 1978-08-04 1980-04-29 Merck & Co., Inc. Alkyl derivatives of C-076 compounds
US4289760A (en) 1980-05-02 1981-09-15 Merck & Co., Inc. 23-Keto derivatives of C-076 compounds
JPS57120589A (en) 1981-01-20 1982-07-27 Sankyo Co Ltd 5-methoxy and 5-lower alkanoyloxy derivative, its preparation and acaricide and parasiticide
IT1144368B (it) 1981-05-20 1986-10-29 Gaudino Di P Gaudino & C Sas O Perfezionamenti nei laminatoi con almeno un campo di stiro per la filatura diretta di pettinato e semipettinato
US4457920A (en) 1981-09-03 1984-07-03 Merck & Co., Inc. 4a-Substituted avermectin compounds
US4423209A (en) 1982-02-26 1983-12-27 Merck & Co., Inc. Processes for the interconversion of avermectin compounds
JPS5916894A (ja) 1982-07-21 1984-01-28 Sankyo Co Ltd ミルベマイシンｄの５−アシルオキシ誘導体
JPS5920285A (ja) 1982-07-23 1984-02-01 Sankyo Co Ltd ミルベマイシンｄの５−二塩基酸エステル誘導体及びその塩
JPS59108785A (ja) 1982-11-25 1984-06-23 Sankyo Co Ltd ミルベマイシン類の５−オキシム誘導体
US4469682A (en) 1983-01-28 1984-09-04 Merck & Co., Inc. Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US4579864A (en) 1984-06-11 1986-04-01 Merck & Co., Inc. Avermectin and milbemycin 13-keto, 13-imino and 13-amino derivatives
US4547491A (en) 1984-07-18 1985-10-15 Merck & Co., Inc. C-8A-Oxo-avermectin and milbemycin derivatives, pharmaceutical compositions and method of use
EP0180539A1 (de) 1984-09-18 1986-05-07 Ciba-Geigy Ag 13-Halo- und 13-Hydroximilbemycine
US4696922A (en) 1984-11-26 1987-09-29 Ciba-Geigy Corporation 5-azolylacetoxymilbemycins as ecto- and endoparasites
JPS6289685A (ja) 1985-05-31 1987-04-24 Sankyo Co Ltd １３−ハロゲンミルベマイシン誘導体
AR243191A1 (es) 1986-03-25 1993-07-30 Sankyo Co Procedimiento para preparar compuestos de macrolida
US5614470A (en) * 1994-04-01 1997-03-25 Sankyo Company, Limited 13-substituted milbemycin derivatives, their preparation and their use
ZA968183B (en) 1995-09-29 1997-04-25 Sankyo Co 13-Substituted milbemycin 5-oxime derivatives their preparation and their use against insects and other pests

Also Published As

Publication number Publication date
HUP0301040A3 (en) 2005-11-28
CZ20023565A3 (cs) 2003-04-16
NO323751B1 (no) 2007-07-02
HUP0301040A2 (hu) 2003-08-28
DK1276748T3 (da) 2006-03-20
CN1247607C (zh) 2006-03-29
TWI285206B (en) 2007-08-11
WO2001083500A8 (en) 2003-05-08
KR100711931B1 (ko) 2007-05-02
AR029250A1 (es) 2003-06-18
NO20025141D0 (no) 2002-10-25
PL357598A1 (en) 2004-07-26
CN1439016A (zh) 2003-08-27
AU2001252613B2 (en) 2004-05-13
EP1276748A1 (en) 2003-01-22
HK1057757A1 (en) 2004-04-16
US20030139601A1 (en) 2003-07-24
WO2001083500A1 (en) 2001-11-08
CA2407611A1 (en) 2001-11-08
ZA200208630B (en) 2004-02-12
NZ522247A (en) 2004-07-30
BR0110385A (pt) 2003-02-04
DE60116615T2 (de) 2006-09-07
AU5261301A (en) 2001-11-12
MXPA02010587A (es) 2003-03-10
KR20020087987A (ko) 2002-11-23
US6653342B2 (en) 2003-11-25
DE60116615D1 (de) 2006-04-06
ATE315573T1 (de) 2006-02-15
IL152449A0 (en) 2003-05-29
EP1276748B1 (en) 2006-01-11
RU2002131794A (ru) 2004-02-27
ES2254400T3 (es) 2006-06-16
RU2226531C1 (ru) 2004-04-10

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