NO20005303L - Fastfase syntese av sulfonerte 2-oksopiperaziner - Google Patents

Fastfase syntese av sulfonerte 2-oksopiperaziner

Info

Publication number
NO20005303L
NO20005303L NO20005303A NO20005303A NO20005303L NO 20005303 L NO20005303 L NO 20005303L NO 20005303 A NO20005303 A NO 20005303A NO 20005303 A NO20005303 A NO 20005303A NO 20005303 L NO20005303 L NO 20005303L
Authority
NO
Norway
Prior art keywords
oxopiperazines
sulfonated
solid phase
resin
phase synthesis
Prior art date
Application number
NO20005303A
Other languages
English (en)
Norwegian (no)
Other versions
NO20005303D0 (no
Inventor
Adam Golebiowski
Sean Rees Klopfenstein
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of NO20005303D0 publication Critical patent/NO20005303D0/no
Publication of NO20005303L publication Critical patent/NO20005303L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D241/00Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/08Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Indole Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20005303A 1998-04-29 2000-10-20 Fastfase syntese av sulfonerte 2-oksopiperaziner NO20005303L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8346898P 1998-04-29 1998-04-29
PCT/US1999/009091 WO1999055684A1 (en) 1998-04-29 1999-04-27 Solid supported synthesis of sulfonated 2-oxopiperazines

Publications (2)

Publication Number Publication Date
NO20005303D0 NO20005303D0 (no) 2000-10-20
NO20005303L true NO20005303L (no) 2000-12-20

Family

ID=22178551

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20005303A NO20005303L (no) 1998-04-29 2000-10-20 Fastfase syntese av sulfonerte 2-oksopiperaziner

Country Status (7)

Country Link
EP (1) EP1073644A1 (ja)
JP (1) JP2002513010A (ja)
AU (1) AU3764399A (ja)
CA (1) CA2328934A1 (ja)
IL (1) IL139121A0 (ja)
NO (1) NO20005303L (ja)
WO (1) WO1999055684A1 (ja)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8114844B2 (en) 2006-03-30 2012-02-14 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptidomimetics
US7964181B2 (en) 2006-03-30 2011-06-21 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5811241A (en) * 1995-09-13 1998-09-22 Cortech, Inc. Method for preparing and identifying N-substitued 1,4-piperazines and N-substituted 1,4-piperazinediones

Also Published As

Publication number Publication date
NO20005303D0 (no) 2000-10-20
EP1073644A1 (en) 2001-02-07
IL139121A0 (en) 2001-11-25
WO1999055684A1 (en) 1999-11-04
CA2328934A1 (en) 1999-11-04
JP2002513010A (ja) 2002-05-08
AU3764399A (en) 1999-11-16

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