NO20002469L - Aromatisk sulfonhydroksamsyre-metalloproteaseinhibitor - Google Patents
Aromatisk sulfonhydroksamsyre-metalloproteaseinhibitorInfo
- Publication number
- NO20002469L NO20002469L NO20002469A NO20002469A NO20002469L NO 20002469 L NO20002469 L NO 20002469L NO 20002469 A NO20002469 A NO 20002469A NO 20002469 A NO20002469 A NO 20002469A NO 20002469 L NO20002469 L NO 20002469L
- Authority
- NO
- Norway
- Prior art keywords
- hydroxamic acid
- aromatic sulfonic
- metalloprotease inhibitor
- acid metalloprotease
- sulfonic hydroxamic
- Prior art date
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- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4166—1,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
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- C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
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Applications Claiming Priority (2)
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US6600797P | 1997-11-14 | 1997-11-14 | |
PCT/US1998/023242 WO1999025687A1 (en) | 1997-11-14 | 1998-11-12 | Aromatic sulfone hydroxamic acid metalloprotease inhibitor |
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NO20002469D0 NO20002469D0 (no) | 2000-05-12 |
NO20002469L true NO20002469L (no) | 2000-07-12 |
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NO20002469A NO20002469L (no) | 1997-11-14 | 2000-05-12 | Aromatisk sulfonhydroksamsyre-metalloproteaseinhibitor |
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US (3) | US6541489B1 (no) |
EP (1) | EP1042290A1 (no) |
JP (1) | JP2001523662A (no) |
CN (1) | CN1279669A (no) |
AR (1) | AR016010A1 (no) |
AU (1) | AU756150C (no) |
BR (1) | BR9814643A (no) |
CA (1) | CA2306460A1 (no) |
IL (1) | IL135106A0 (no) |
NO (1) | NO20002469L (no) |
NZ (1) | NZ503485A (no) |
PL (1) | PL341379A1 (no) |
RU (1) | RU2250105C2 (no) |
WO (1) | WO1999025687A1 (no) |
ZA (1) | ZA9810412B (no) |
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-
1998
- 1998-11-12 NZ NZ503485A patent/NZ503485A/en unknown
- 1998-11-12 IL IL13510698A patent/IL135106A0/xx unknown
- 1998-11-12 EP EP98957485A patent/EP1042290A1/en not_active Withdrawn
- 1998-11-12 RU RU2000115948/15A patent/RU2250105C2/ru not_active IP Right Cessation
- 1998-11-12 JP JP2000521071A patent/JP2001523662A/ja not_active Withdrawn
- 1998-11-12 AU AU13732/99A patent/AU756150C/en not_active Ceased
- 1998-11-12 CA CA002306460A patent/CA2306460A1/en not_active Abandoned
- 1998-11-12 US US09/554,082 patent/US6541489B1/en not_active Expired - Fee Related
- 1998-11-12 BR BR9814643-2A patent/BR9814643A/pt not_active Application Discontinuation
- 1998-11-12 CN CN98811130A patent/CN1279669A/zh active Pending
- 1998-11-12 PL PL98341379A patent/PL341379A1/xx unknown
- 1998-11-12 WO PCT/US1998/023242 patent/WO1999025687A1/en not_active Application Discontinuation
- 1998-11-13 AR ARP980105784A patent/AR016010A1/es unknown
- 1998-11-13 ZA ZA9810412A patent/ZA9810412B/xx unknown
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2000
- 2000-05-12 NO NO20002469A patent/NO20002469L/no not_active Application Discontinuation
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2003
- 2003-01-07 US US10/337,942 patent/US6890937B2/en not_active Expired - Fee Related
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2005
- 2005-01-28 US US11/046,645 patent/US20060084688A1/en not_active Abandoned
Also Published As
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CA2306460A1 (en) | 1999-05-27 |
AR016010A1 (es) | 2001-05-30 |
US20060084688A1 (en) | 2006-04-20 |
WO1999025687A1 (en) | 1999-05-27 |
PL341379A1 (en) | 2001-04-09 |
JP2001523662A (ja) | 2001-11-27 |
ZA9810412B (en) | 1999-12-09 |
EP1042290A1 (en) | 2000-10-11 |
BR9814643A (pt) | 2000-10-03 |
NZ503485A (en) | 2002-10-25 |
AU756150B2 (en) | 2003-01-02 |
RU2250105C2 (ru) | 2005-04-20 |
NO20002469D0 (no) | 2000-05-12 |
AU756150C (en) | 2004-03-04 |
US20040048852A1 (en) | 2004-03-11 |
US6890937B2 (en) | 2005-05-10 |
CN1279669A (zh) | 2001-01-10 |
AU1373299A (en) | 1999-06-07 |
US6541489B1 (en) | 2003-04-01 |
IL135106A0 (en) | 2001-05-20 |
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