NO178188C - Analogifremgangsmåte for fremstilling av terapeutisk aktive 4,5,6,7-tetrahydro-benzimidazolderivater - Google Patents

Analogifremgangsmåte for fremstilling av terapeutisk aktive 4,5,6,7-tetrahydro-benzimidazolderivater

Info

Publication number
NO178188C
NO178188C NO895198A NO895198A NO178188C NO 178188 C NO178188 C NO 178188C NO 895198 A NO895198 A NO 895198A NO 895198 A NO895198 A NO 895198A NO 178188 C NO178188 C NO 178188C
Authority
NO
Norway
Prior art keywords
group
tetrahydro
preparation
atom
therapeutically active
Prior art date
Application number
NO895198A
Other languages
English (en)
Norwegian (no)
Other versions
NO895198D0 (no
NO895198L (no
NO178188B (no
Inventor
Mitsuaki Ohta
Tokuo Koide
Takeshi Suzuki
Akira Matsuhisa
Isao Yanagisawa
Keiji Miyata
Original Assignee
Yamanouchi Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26389240&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO178188(C) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd
Publication of NO895198D0 publication Critical patent/NO895198D0/no
Publication of NO895198L publication Critical patent/NO895198L/no
Publication of NO178188B publication Critical patent/NO178188B/no
Publication of NO178188C publication Critical patent/NO178188C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08Radicals containing only hydrogen and carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Reinforced Plastic Materials (AREA)
  • Adhesive Tapes (AREA)
  • Analysing Materials By The Use Of Radiation (AREA)
NO895198A 1988-12-22 1989-12-21 Analogifremgangsmåte for fremstilling av terapeutisk aktive 4,5,6,7-tetrahydro-benzimidazolderivater NO178188C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP32532788 1988-12-22
JP4889689 1989-02-28

Publications (4)

Publication Number Publication Date
NO895198D0 NO895198D0 (no) 1989-12-21
NO895198L NO895198L (no) 1990-06-25
NO178188B NO178188B (no) 1995-10-30
NO178188C true NO178188C (no) 1996-02-07

Family

ID=26389240

Family Applications (1)

Application Number Title Priority Date Filing Date
NO895198A NO178188C (no) 1988-12-22 1989-12-21 Analogifremgangsmåte for fremstilling av terapeutisk aktive 4,5,6,7-tetrahydro-benzimidazolderivater

Country Status (15)

Country Link
US (1) US4977175A (de)
EP (1) EP0376624B1 (de)
KR (1) KR900009608A (de)
CN (1) CN1027536C (de)
AT (1) ATE111454T1 (de)
AU (1) AU630397B2 (de)
CA (1) CA2004911A1 (de)
DE (1) DE68918257T2 (de)
DK (1) DK653089A (de)
ES (1) ES2063831T3 (de)
FI (1) FI896075A7 (de)
IE (1) IE65639B1 (de)
NO (1) NO178188C (de)
PT (1) PT92609B (de)
YU (1) YU47216B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69028934T2 (de) * 1989-02-02 1997-03-20 Yamanouchi Pharma Co Ltd Tetrahydrobenzimidazol-Derivate
GB8928837D0 (en) * 1989-12-21 1990-02-28 Beecham Group Plc Pharmaceuticals
GB9214184D0 (en) * 1992-07-03 1992-08-12 Smithkline Beecham Plc Pharmaceuticals
GB9225141D0 (en) * 1992-12-01 1993-01-20 Smithkline Beecham Corp Chemical compounds
US5262537A (en) * 1993-03-19 1993-11-16 Anaquest, Inc. Derivatives of 4,5,6,7-tetrahydroimidazo-[4,5-c]pyridinyl-6-carboxylic acid
AU722514B2 (en) * 1995-12-28 2000-08-03 Fujisawa Pharmaceutical Co., Ltd. Benzimidazole derivatives
TW453999B (en) 1997-06-27 2001-09-11 Fujisawa Pharmaceutical Co Benzimidazole derivatives
EP1268484A1 (de) * 2000-03-17 2003-01-02 Novo Nordisk A/S Kondensierte imidazole als histamin h3-rezeptor liganden
US6437147B1 (en) 2000-03-17 2002-08-20 Novo Nordisk Imidazole compounds
DE60306918T2 (de) * 2002-05-17 2007-03-01 Neurogen Corp., Branford Substituierte, ringkondensierte imidazolderivate: gabaa-rezeptorliganden
MX2019001917A (es) * 2016-08-16 2019-07-15 Bayer Cropscience Ag Metodo para producir derivados de piridina 2-(3,6-dihalopyridin-2- yl)-3h-imidazol[4,5-c] y compuestos relacionados por reaccion del derivado de piridina 3h-imidazol[4,5-c] con una base organometalica de zinc-amina.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1260294A (en) * 1968-03-15 1972-01-12 Rhein Chemie Holding G M B H 4,5,6,7-tetrahydrobenzimidazoles, process for their production and their use as corrosion inhibitors and antioxidants
DE1948795A1 (de) * 1969-09-26 1971-04-08 Rhein Chemie Rheinau Gmbh 4,5,6,7-Tetrahydrobenzimidazole,Verfahren zu ihrer Herstellung und ihre Verwendung als Korrosionsinhibitoren und Alterungsschutzmittel
US3987054A (en) * 1970-09-23 1976-10-19 Pliva Pharmaceutical And Chemical Works 4,5,6,7-tetrahydrobenzimidazoles
FI74707C (fi) * 1982-06-29 1988-03-10 Sandoz Ag Foerfarande foer framstaellning av terapeutiskt anvaendbara alkylenoeverbryggade piperidylestrar eller -amider av bicykliska karboxylsyror.
LU88268I2 (de) * 1984-01-25 1994-02-03
DE3687080T2 (de) * 1985-04-27 1993-03-25 Beecham Group Plc Azabicyclononyl-indazol-carboxamid mit 5-ht-antagonistischer wirkung.
US4826990A (en) * 1987-09-30 1989-05-02 American Home Products Corporation 2-aryl substituted heterocyclic compounds as antiallergic and antiinflammatory agents

Also Published As

Publication number Publication date
EP0376624A1 (de) 1990-07-04
DE68918257T2 (de) 1995-02-02
ATE111454T1 (de) 1994-09-15
KR900009608A (ko) 1990-07-05
PT92609A (pt) 1990-06-29
ES2063831T3 (es) 1995-01-16
CN1027536C (zh) 1995-02-01
IE65639B1 (en) 1995-11-15
CN1043706A (zh) 1990-07-11
DK653089D0 (da) 1989-12-21
DK653089A (da) 1990-06-23
FI896075A0 (fi) 1989-12-19
IE894185L (en) 1990-06-22
NO895198D0 (no) 1989-12-21
US4977175A (en) 1990-12-11
NO895198L (no) 1990-06-25
EP0376624B1 (de) 1994-09-14
NO178188B (no) 1995-10-30
CA2004911A1 (en) 1990-06-22
YU243989A (en) 1991-02-28
DE68918257D1 (de) 1994-10-20
FI896075A7 (fi) 1990-06-23
AU4714589A (en) 1990-06-28
AU630397B2 (en) 1992-10-29
PT92609B (pt) 1995-09-12
YU47216B (sh) 1995-01-31

Similar Documents

Publication Publication Date Title
NO177638C (no) Analogifremgangsmåte for fremstilling av en terapeutisk aktiv spiroforbindelse
NO178188C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive 4,5,6,7-tetrahydro-benzimidazolderivater
NO174257C (no) Analogifremgangsmåte for fremstilling av terapeutisk aktive imidazopyridaziner
IS3828A (is) Hliðstæð aðferð til tilreiðslu á nýjum afleiðum thiazolidinone og oxazolidinone sem gagnlegar eru til æðaútvíkkunar
EP0417790A3 (en) S-triazolo(3,4-i)purine derivatives
IE893211L (en) Benzoxazepinone Process
AU8003594A (en) Quinolinecarboxylic acid derivative and salt thereof
NO931225L (no) Benzoksazinon- og benzotiazinon-derivater med kardiovaskulaer akrivitet
GR851843B (de)
AU1586588A (en) Fungicidal derivatives of propenoic acid and processes for their preparation
ES2017537B3 (es) Acidos 1,3,4,9-tetrahidropizano [3,4-b] indol-1-aceticos sustituidos.
AU7748487A (en) 2-amino-3-aroyl-omega-oxobenzenebutanoic acids and esters
ES2039270T3 (es) Derivados de gamma-l-glutamil-4-nitroanilida y procedimiento para determinar actividad de gamma-gtp utilizandolos.