NO156011C - Analogifremgangsmaate for fremstilling av nye terapeutisk aktive 3, 6, 7, 8-substituerte-s-triazolo (4,3-b) pyridaziner. - Google Patents

Analogifremgangsmaate for fremstilling av nye terapeutisk aktive 3, 6, 7, 8-substituerte-s-triazolo (4,3-b) pyridaziner.

Info

Publication number
NO156011C
NO156011C NO803218A NO803218A NO156011C NO 156011 C NO156011 C NO 156011C NO 803218 A NO803218 A NO 803218A NO 803218 A NO803218 A NO 803218A NO 156011 C NO156011 C NO 156011C
Authority
NO
Norway
Prior art keywords
pyridazines
triazolo
substituted
preparation
new therapeutic
Prior art date
Application number
NO803218A
Other languages
English (en)
Norwegian (no)
Other versions
NO803218L (no
NO156011B (no
Inventor
Norton Paul Peet
Shyam Sunder
Original Assignee
Dow Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Chemical Co filed Critical Dow Chemical Co
Publication of NO803218L publication Critical patent/NO803218L/no
Publication of NO156011B publication Critical patent/NO156011B/no
Publication of NO156011C publication Critical patent/NO156011C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO803218A 1979-10-29 1980-10-28 Analogifremgangsmaate for fremstilling av nye terapeutisk aktive 3, 6, 7, 8-substituerte-s-triazolo (4,3-b) pyridaziner. NO156011C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8907179A 1979-10-29 1979-10-29

Publications (3)

Publication Number Publication Date
NO803218L NO803218L (no) 1981-04-30
NO156011B NO156011B (no) 1987-03-30
NO156011C true NO156011C (no) 1987-07-08

Family

ID=22215530

Family Applications (1)

Application Number Title Priority Date Filing Date
NO803218A NO156011C (no) 1979-10-29 1980-10-28 Analogifremgangsmaate for fremstilling av nye terapeutisk aktive 3, 6, 7, 8-substituerte-s-triazolo (4,3-b) pyridaziner.

Country Status (18)

Country Link
EP (1) EP0029130B1 (fi)
JP (1) JPS5679690A (fi)
KR (1) KR850001701B1 (fi)
AR (2) AR227651A1 (fi)
AT (1) ATE16808T1 (fi)
AU (1) AU536351B2 (fi)
CA (1) CA1144544A (fi)
DE (1) DE3071278D1 (fi)
DK (1) DK158353C (fi)
ES (2) ES496354A0 (fi)
FI (1) FI70413C (fi)
GB (1) GB2061275B (fi)
GR (1) GR70309B (fi)
IL (1) IL61316A (fi)
NO (1) NO156011C (fi)
NZ (1) NZ195355A (fi)
PT (1) PT71952B (fi)
ZA (1) ZA806523B (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH21834A (en) * 1982-01-18 1988-03-17 Lepetit Spa New 6-substituted-s-triazolo(3,4-a)phthalazine derivatives
US4485106A (en) * 1982-07-12 1984-11-27 The Dow Chemical Company Substituted tetrahydrotetrazolo[5,1-a]phthalazines
US4487930A (en) * 1982-09-07 1984-12-11 The Dow Chemical Company 6-[(Cyclic amino)alkylamino]-tetrahydrotriazolo[3,4-a]phthalazines
IT1194310B (it) * 1983-07-12 1988-09-14 Lepetit Spa Derivati triazolo (3,4-a) ftalazinici 3,6-disostituiti
US4578464A (en) * 1983-11-22 1986-03-25 Merrell Dow Pharmaceuticals Inc. 6-Hydroxyalkylamino-8-methyl-1,2,4-triazolo-[4,3-b]pyridazine and related compounds
US5011835A (en) * 1990-02-07 1991-04-30 Merrell Dow Pharmaceuticals Inc. Substituted triazolopyridazines, pharmaceutical compositions and use
KR20120111739A (ko) 2009-12-31 2012-10-10 센트로 내셔널 드 인베스티가시오네스 온콜로지카스 (씨엔아이오) 키나제 억제제로서의 사용을 위한 삼환식 화합물
WO2012098387A1 (en) 2011-01-18 2012-07-26 Centro Nacional De Investigaciones Oncológicas (Cnio) 6, 7-ring-fused triazolo [4, 3 - b] pyridazine derivatives as pim inhibitors
WO2013005041A1 (en) 2011-07-07 2013-01-10 Centro Nacional De Investigaciones Oncológicas (Cnio) Tricyclic heterocyclic compounds as kinase inhibitors
WO2013004984A1 (en) 2011-07-07 2013-01-10 Centro Nacional De Investigaciones Oncologicas (Cnio) Tricyclic compounds for use as kinase inhibitors
WO2013005057A1 (en) 2011-07-07 2013-01-10 Centro Nacional De Investigaciones Oncológicas (Cnio) New compounds
CN103694244B (zh) * 2014-01-09 2016-03-30 郑州大学 3,6位取代-1,2,4-三氮唑并[3,4-a]酞嗪类化合物及其制备和用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3708484A (en) * 1970-10-16 1973-01-02 Sandoz Ag Amino and substituted amino-s-triazolo-(4,3-b)-pyridazines
US3915968A (en) * 1973-09-21 1975-10-28 Lepetit Spa Triazolopyridazines
DE2418435A1 (de) * 1974-04-17 1975-10-30 Boehringer Mannheim Gmbh Nitroimidazolyl-triazolo-pyridazine und verfahren zu ihrer herstellung
US4136182A (en) * 1976-05-26 1979-01-23 The Dow Chemical Company Triazolopyridazines used to alleviate bronchial spasms
CA1080712A (en) * 1976-09-22 1980-07-01 Jay D. Albright Hypotensive agents

Also Published As

Publication number Publication date
KR850001701B1 (ko) 1985-11-26
KR830004301A (ko) 1983-07-09
ATE16808T1 (de) 1985-12-15
GR70309B (fi) 1982-09-08
AU536351B2 (en) 1984-05-03
EP0029130B1 (en) 1985-12-04
EP0029130A1 (en) 1981-05-27
DK158353C (da) 1990-10-01
NO803218L (no) 1981-04-30
AR227087A1 (es) 1982-09-15
GB2061275B (en) 1983-08-10
IL61316A0 (en) 1980-12-31
ZA806523B (en) 1982-05-26
DK158353B (da) 1990-05-07
JPS5679690A (en) 1981-06-30
ES8202555A1 (es) 1982-02-01
PT71952B (en) 1982-03-31
IL61316A (en) 1984-03-30
NZ195355A (en) 1984-09-28
DE3071278D1 (en) 1986-01-16
FI70413C (fi) 1986-09-19
AR227651A1 (es) 1982-11-30
AU6356180A (en) 1981-05-07
GB2061275A (en) 1981-05-13
ES506946A0 (es) 1982-09-01
FI70413B (fi) 1986-03-27
NO156011B (no) 1987-03-30
PT71952A (en) 1980-11-01
FI803355L (fi) 1981-04-30
JPH0248558B2 (fi) 1990-10-25
DK457480A (da) 1981-04-30
CA1144544A (en) 1983-04-12
ES8207178A1 (es) 1982-09-01
ES496354A0 (es) 1982-02-01

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