NO148416C - ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLIDINE, MORPHOLINE AND TIAZAN DERIVATIVES - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLIDINE, MORPHOLINE AND TIAZAN DERIVATIVES

Info

Publication number
NO148416C
NO148416C NO774126A NO774126A NO148416C NO 148416 C NO148416 C NO 148416C NO 774126 A NO774126 A NO 774126A NO 774126 A NO774126 A NO 774126A NO 148416 C NO148416 C NO 148416C
Authority
NO
Norway
Prior art keywords
tiazan
tiazolidine
morpholine
derivatives
preparation
Prior art date
Application number
NO774126A
Other languages
Norwegian (no)
Other versions
NO774126L (en
NO148416B (en
Inventor
Miguel Angel Ondetti
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of NO774126L publication Critical patent/NO774126L/en
Publication of NO148416B publication Critical patent/NO148416B/en
Publication of NO148416C publication Critical patent/NO148416C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D277/06Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/041,3-Thiazines; Hydrogenated 1,3-thiazines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/101,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/121,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO774126A 1976-12-03 1977-12-02 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLIDINE, MORPHOLINE AND TIAZAN DERIVATIVES NO148416C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US74728176A 1976-12-03 1976-12-03
US83610777A 1977-09-23 1977-09-23

Publications (3)

Publication Number Publication Date
NO774126L NO774126L (en) 1978-06-06
NO148416B NO148416B (en) 1983-06-27
NO148416C true NO148416C (en) 1983-10-12

Family

ID=27114718

Family Applications (1)

Application Number Title Priority Date Filing Date
NO774126A NO148416C (en) 1976-12-03 1977-12-02 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLIDINE, MORPHOLINE AND TIAZAN DERIVATIVES

Country Status (28)

Country Link
JP (1) JPS5382778A (en)
AR (1) AR220689A1 (en)
AT (1) AT363467B (en)
AU (1) AU518147B2 (en)
BG (1) BG32269A3 (en)
CA (1) CA1146940A (en)
CH (1) CH634062A5 (en)
DD (1) DD133798A5 (en)
DE (1) DE2752719C2 (en)
DK (1) DK152494C (en)
EG (1) EG13037A (en)
ES (1) ES464555A1 (en)
FI (1) FI67378C (en)
FR (1) FR2372817A1 (en)
GB (1) GB1578940A (en)
GR (1) GR72453B (en)
HK (1) HK55881A (en)
IE (1) IE46169B1 (en)
IL (1) IL53352A0 (en)
IN (1) IN146945B (en)
IT (1) IT1092179B (en)
NL (3) NL171055C (en)
NO (1) NO148416C (en)
NZ (1) NZ185800A (en)
PT (1) PT67352B (en)
RO (2) RO78013A (en)
SE (1) SE441267B (en)
YU (1) YU41823B (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2395998A1 (en) * 1977-06-29 1979-01-26 Yoshitomi Pharmaceutical NEW THIAZOLIDINE DERIVATIVES AND THEIR APPLICATION IN THE TREATMENT OF HYPERTENSION
JPS5455565A (en) * 1977-10-06 1979-05-02 Santen Pharmaceut Co Ltd Novel thiazolidine derivative
US4430344A (en) * 1978-04-08 1984-02-07 Santen Pharmaceutical Co., Ltd. Antihypertensive 4-thiazolidinecarboxylic acids
JPS557255A (en) * 1978-07-03 1980-01-19 Santen Pharmaceut Co Ltd Thiazolidine derivative
JPS5531022A (en) * 1978-08-24 1980-03-05 Yoshitomi Pharmaceut Ind Ltd Hydroxamic acid derivative and its preparation
GR73585B (en) * 1978-09-11 1984-03-26 Univ Miami
JPS5540622A (en) * 1978-09-14 1980-03-22 Santen Pharmaceut Co Ltd Hypotensive agent
JPS5829950B2 (en) * 1978-10-05 1983-06-25 ウェルファイド株式会社 Cyclic iminocarboxylic acid derivatives and their salts
US4483861A (en) * 1978-10-31 1984-11-20 Santen Pharmaceutical Co., Ltd. Antihypertensive sulfur-containing compounds
JPS5562060A (en) * 1978-10-31 1980-05-10 Santen Pharmaceut Co Ltd Sulfur-containing compound
US4347371A (en) * 1978-12-30 1982-08-31 Santen Pharmaceutical Co., Ltd. Disulfide compounds
JPS55124757A (en) * 1979-03-17 1980-09-26 Santen Pharmaceut Co Ltd Sulfur-containing compound
JPS565415A (en) * 1979-06-26 1981-01-20 Santen Pharmaceut Co Ltd Ester-type hypotensor
JPS5683483A (en) * 1979-12-13 1981-07-08 Santen Pharmaceut Co Ltd Thiazolidine compound
JPS56139455A (en) * 1980-04-02 1981-10-30 Santen Pharmaceut Co Ltd Sulfur-containing acylaminoacid
DE3152643A1 (en) * 1980-12-29 1982-12-16 Santen Pharmaceutical Co Ltd HETEROCYCLIC 5-MEMBERED RING COMPOUNDS
JPH0662529B2 (en) * 1984-07-13 1994-08-17 三共株式会社 Amino acid derivative
EP0190685B1 (en) * 1985-02-04 1992-07-01 G.D. Searle & Co. Heterocyclic amides

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2446100C3 (en) * 1974-09-26 1982-01-14 Ludwig Merckle Kg Chem. Pharm. Fabrik, 7902 Blaubeuren Phenoxyalkanecarboxamides of thiazolidinecarboxylic acids, process for their preparation and pharmaceuticals
AU509899B2 (en) * 1976-02-13 1980-05-29 E.R. Squibb & Sons, Inc. Proline derivatives and related compounds

Also Published As

Publication number Publication date
NL8201146A (en) 1982-07-01
CA1146940A (en) 1983-05-24
EG13037A (en) 1980-12-31
JPS618834B2 (en) 1986-03-18
RO78013A (en) 1981-12-25
HK55881A (en) 1981-11-20
AT363467B (en) 1981-08-10
DE2752719C2 (en) 1982-03-25
PT67352A (en) 1978-01-01
IL53352A0 (en) 1978-01-31
JPS5382778A (en) 1978-07-21
NZ185800A (en) 1980-04-28
IE46169L (en) 1978-06-03
FI67378B (en) 1984-11-30
FI773640A (en) 1978-06-04
FR2372817B1 (en) 1981-06-19
GB1578940A (en) 1980-11-12
FR2372817A1 (en) 1978-06-30
FI67378C (en) 1985-03-11
NO774126L (en) 1978-06-06
AU3037977A (en) 1979-05-17
IT1092179B (en) 1985-07-06
NL171055C (en) 1983-02-01
NL7713274A (en) 1978-06-06
RO72596A (en) 1983-08-03
DK152494C (en) 1988-07-25
AU518147B2 (en) 1981-09-17
AR220689A1 (en) 1980-11-28
IE46169B1 (en) 1983-03-09
DK152494B (en) 1988-03-07
GR72453B (en) 1983-11-09
SE441267B (en) 1985-09-23
NO148416B (en) 1983-06-27
PT67352B (en) 1979-05-15
YU283777A (en) 1983-01-21
DK538277A (en) 1978-06-04
ES464555A1 (en) 1978-09-01
IN146945B (en) 1979-10-20
DE2752719A1 (en) 1978-06-08
YU41823B (en) 1988-02-29
NL8201145A (en) 1982-07-01
CH634062A5 (en) 1983-01-14
RO72596B (en) 1983-07-30
DD133798A5 (en) 1979-01-24
BG32269A3 (en) 1982-06-15
SE7713722L (en) 1978-06-04
ATA857677A (en) 1981-01-15

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