NO142260C - ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIENOTRIAZOLODIAZEPINE DERIVATIVES - Google Patents

ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIENOTRIAZOLODIAZEPINE DERIVATIVES

Info

Publication number
NO142260C
NO142260C NO740405A NO740405A NO142260C NO 142260 C NO142260 C NO 142260C NO 740405 A NO740405 A NO 740405A NO 740405 A NO740405 A NO 740405A NO 142260 C NO142260 C NO 142260C
Authority
NO
Norway
Prior art keywords
tienotriazolodiazepine
derivatives
preparation
therapeutically active
analogy procedure
Prior art date
Application number
NO740405A
Other languages
Norwegian (no)
Other versions
NO142260B (en
NO740405L (en
Inventor
Joseph Hellerbach
Paul Zeller
Dieter Binder
Otto Hromatka
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO740405L publication Critical patent/NO740405L/en
Publication of NO142260B publication Critical patent/NO142260B/en
Publication of NO142260C publication Critical patent/NO142260C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
NO740405A 1973-02-08 1974-02-07 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIENOTRIAZOLODIAZEPINE DERIVATIVES NO142260C (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH179973A CH584223A5 (en) 1973-02-08 1973-02-08

Publications (3)

Publication Number Publication Date
NO740405L NO740405L (en) 1974-08-09
NO142260B NO142260B (en) 1980-04-14
NO142260C true NO142260C (en) 1980-07-23

Family

ID=4218866

Family Applications (1)

Application Number Title Priority Date Filing Date
NO740405A NO142260C (en) 1973-02-08 1974-02-07 ANALOGY PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIENOTRIAZOLODIAZEPINE DERIVATIVES

Country Status (24)

Country Link
JP (1) JPS5833234B2 (en)
AR (2) AR203188A1 (en)
AT (1) AT343118B (en)
BE (1) BE810705A (en)
CA (1) CA1049009A (en)
CH (1) CH584223A5 (en)
DD (1) DD112454A5 (en)
DE (1) DE2405682C3 (en)
DK (1) DK137679B (en)
FI (1) FI58129C (en)
FR (1) FR2217007B1 (en)
GB (2) GB1456162A (en)
HU (2) HU170423B (en)
IE (1) IE38883B1 (en)
IL (1) IL44095A (en)
LU (1) LU69338A1 (en)
NL (1) NL174045C (en)
NO (1) NO142260C (en)
PH (1) PH12303A (en)
PL (3) PL96107B1 (en)
SE (1) SE416399B (en)
SU (3) SU715028A3 (en)
YU (1) YU39716B (en)
ZA (1) ZA74472B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT338799B (en) * 1974-03-02 1977-09-12 Boehringer Sohn Ingelheim PROCESS FOR PREPARING NEW SUBSTITUTED 6-ARYL-4H-S-TRIAZOLO- (3,4C) -THIENO- (2,3E) -1,4-DIAZEPINE AND THEIR SALTS
DE2533924C3 (en) * 1975-07-30 1979-05-03 C.H. Boehringer Sohn, 6507 Ingelheim Process for the preparation of 6-aryl-4H-striazolo [3,4-c] thieno [2,3-e] 1,4-diazepines
DE2531678C3 (en) * 1975-07-16 1979-06-28 C.H. Boehringer Sohn, 6507 Ingelheim Thieno [2,3e] triazole [3,4c] 5,6-dihydro-1,4-diazepines and processes for their preparation
DE2708121A1 (en) * 1977-02-25 1978-09-07 Boehringer Sohn Ingelheim TRIAZOLO-THIENO-DIAZEPIN-L-ONE, METHOD FOR THEIR PRODUCTION AND MEDICINAL PRODUCTS
FI63033C (en) * 1977-07-21 1983-04-11 Boehringer Sohn Ingelheim FREQUENCY REQUIREMENT FOR ANXIOLYTIC TRANSQUILLATION OF SEED / ELLER NEUROLEPTIC SUBSTITUTES 1-PIPERAZINYL-4H-S-TRIAZOLO (3,4-C) THIENO (2,3-E) -1,4-DIAZEPERE
DE3502392A1 (en) * 1985-01-25 1986-07-31 Boehringer Ingelheim KG, 6507 Ingelheim NEW THIENO-TRIAZOLO-1,4-DIAZEPINO-2-CARBONIC ACID AMIDES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS
DE3778559D1 (en) * 1986-01-21 1992-06-04 Boehringer Ingelheim Kg THIENO-1,4-DIAZEPINE.
JP2582225B2 (en) * 1994-04-15 1997-02-19 ナショナル住宅産業株式会社 Fittings
WO1995032963A1 (en) * 1994-06-01 1995-12-07 Yoshitomi Pharmaceutical Industries, Ltd. Thienylazole compound and thienotriazolodiazepine compound
WO1997009048A1 (en) * 1995-09-09 1997-03-13 F. Hoffmann-La Roche Ag Use of a thienotriazolodiazepine to increase apolipoprotein a-i levels

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904641A (en) * 1971-06-18 1975-09-09 Yoshitomi Pharmaceutical Triazolothienodiazepine compounds

Also Published As

Publication number Publication date
DE2405682A1 (en) 1974-08-15
PL97275B1 (en) 1978-02-28
JPS49102698A (en) 1974-09-27
SU747429A4 (en) 1980-07-23
IL44095A (en) 1979-03-12
NL174045C (en) 1984-04-16
NO142260B (en) 1980-04-14
ATA96474A (en) 1977-09-15
PL96107B1 (en) 1977-12-31
FI58129C (en) 1980-12-10
AT343118B (en) 1978-05-10
BE810705A (en) 1974-08-07
CH584223A5 (en) 1977-01-31
AR203188A1 (en) 1975-08-22
NL174045B (en) 1983-11-16
SU1060115A3 (en) 1983-12-07
FR2217007A1 (en) 1974-09-06
ZA74472B (en) 1974-11-27
NO740405L (en) 1974-08-09
IE38883L (en) 1974-08-08
DE2405682C3 (en) 1981-03-12
FI58129B (en) 1980-08-29
NL7401117A (en) 1974-08-12
CA1049009A (en) 1979-02-20
HU170423B (en) 1977-06-28
DK137679C (en) 1978-09-25
SU715028A3 (en) 1980-02-05
GB1456162A (en) 1976-11-17
GB1456161A (en) 1976-11-17
JPS5833234B2 (en) 1983-07-18
IE38883B1 (en) 1978-06-21
HU173741B (en) 1979-08-28
YU22874A (en) 1982-06-30
PH12303A (en) 1979-01-16
SE416399B (en) 1980-12-22
FR2217007B1 (en) 1978-02-03
PL97304B1 (en) 1978-02-28
AR217034A1 (en) 1980-02-29
YU39716B (en) 1985-04-30
DD112454A5 (en) 1975-04-12
DK137679B (en) 1978-04-17
DE2405682B2 (en) 1980-07-17
AU6485574A (en) 1975-07-24
IL44095A0 (en) 1974-05-16
LU69338A1 (en) 1975-12-09

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