ATA96474A - PROCESS FOR THE PREPARATION OF NEW THIENOTRIAZOLODIAZEPINE DERIVATIVES AND THEIR SALTS - Google Patents

PROCESS FOR THE PREPARATION OF NEW THIENOTRIAZOLODIAZEPINE DERIVATIVES AND THEIR SALTS

Info

Publication number
ATA96474A
ATA96474A AT96474A AT96474A ATA96474A AT A96474 A ATA96474 A AT A96474A AT 96474 A AT96474 A AT 96474A AT 96474 A AT96474 A AT 96474A AT A96474 A ATA96474 A AT A96474A
Authority
AT
Austria
Prior art keywords
salts
preparation
new
thienotriazolodiazepine derivatives
thienotriazolodiazepine
Prior art date
Application number
AT96474A
Other languages
German (de)
Other versions
AT343118B (en
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Priority to AT882176A priority Critical patent/AT344183B/en
Priority to AT882276A priority patent/AT342605B/en
Priority to AT882076A priority patent/AT342604B/en
Publication of ATA96474A publication Critical patent/ATA96474A/en
Application granted granted Critical
Publication of AT343118B publication Critical patent/AT343118B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
AT96474A 1973-02-08 1974-02-07 METHOD FOR PRODUCING NEW THIENOTRIAZOLODIAZEPINE DERIVATIVES AND THEIR SALTS AT343118B (en)

Priority Applications (3)

Application Number Priority Date Filing Date Title
AT882176A AT344183B (en) 1973-02-08 1976-11-29 PROCESS FOR THE PREPARATION OF NEW THIENOTRIAZOLODIAZEPINE DERIVATIVES AND THEIR ACID ADDITION SALTS
AT882276A AT342605B (en) 1973-02-08 1976-11-29 PROCESS FOR THE PREPARATION OF NEW THIENOTRIAZOLODIAZEPINE DERIVATIVES AND THEIR SALTS
AT882076A AT342604B (en) 1973-02-08 1976-11-29 PROCESS FOR THE PREPARATION OF NEW THIENOTRIAZOLODIAZEPINE DERIVATIVES AND THEIR ACID ADDITION SALTS

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH179973A CH584223A5 (en) 1973-02-08 1973-02-08

Publications (2)

Publication Number Publication Date
ATA96474A true ATA96474A (en) 1977-09-15
AT343118B AT343118B (en) 1978-05-10

Family

ID=4218866

Family Applications (1)

Application Number Title Priority Date Filing Date
AT96474A AT343118B (en) 1973-02-08 1974-02-07 METHOD FOR PRODUCING NEW THIENOTRIAZOLODIAZEPINE DERIVATIVES AND THEIR SALTS

Country Status (24)

Country Link
JP (1) JPS5833234B2 (en)
AR (2) AR203188A1 (en)
AT (1) AT343118B (en)
BE (1) BE810705A (en)
CA (1) CA1049009A (en)
CH (1) CH584223A5 (en)
DD (1) DD112454A5 (en)
DE (1) DE2405682C3 (en)
DK (1) DK137679B (en)
FI (1) FI58129C (en)
FR (1) FR2217007B1 (en)
GB (2) GB1456161A (en)
HU (2) HU170423B (en)
IE (1) IE38883B1 (en)
IL (1) IL44095A (en)
LU (1) LU69338A1 (en)
NL (1) NL174045C (en)
NO (1) NO142260C (en)
PH (1) PH12303A (en)
PL (3) PL97304B1 (en)
SE (1) SE416399B (en)
SU (3) SU715028A3 (en)
YU (1) YU39716B (en)
ZA (1) ZA74472B (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT338799B (en) * 1974-03-02 1977-09-12 Boehringer Sohn Ingelheim PROCESS FOR PREPARING NEW SUBSTITUTED 6-ARYL-4H-S-TRIAZOLO- (3,4C) -THIENO- (2,3E) -1,4-DIAZEPINE AND THEIR SALTS
DE2531678C3 (en) * 1975-07-16 1979-06-28 C.H. Boehringer Sohn, 6507 Ingelheim Thieno [2,3e] triazole [3,4c] 5,6-dihydro-1,4-diazepines and processes for their preparation
DE2533924C3 (en) * 1975-07-30 1979-05-03 C.H. Boehringer Sohn, 6507 Ingelheim Process for the preparation of 6-aryl-4H-striazolo [3,4-c] thieno [2,3-e] 1,4-diazepines
DE2708121A1 (en) * 1977-02-25 1978-09-07 Boehringer Sohn Ingelheim TRIAZOLO-THIENO-DIAZEPIN-L-ONE, METHOD FOR THEIR PRODUCTION AND MEDICINAL PRODUCTS
FI63033C (en) * 1977-07-21 1983-04-11 Boehringer Sohn Ingelheim FREQUENCY REQUIREMENT FOR ANXIOLYTIC TRANSQUILLATION OF SEED / ELLER NEUROLEPTIC SUBSTITUTES 1-PIPERAZINYL-4H-S-TRIAZOLO (3,4-C) THIENO (2,3-E) -1,4-DIAZEPERE
DE3502392A1 (en) * 1985-01-25 1986-07-31 Boehringer Ingelheim KG, 6507 Ingelheim NEW THIENO-TRIAZOLO-1,4-DIAZEPINO-2-CARBONIC ACID AMIDES, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS
EP0230942B1 (en) * 1986-01-21 1992-04-29 Boehringer Ingelheim Kg Thieno-1,4-diazepines
JP2582225B2 (en) * 1994-04-15 1997-02-19 ナショナル住宅産業株式会社 Fittings
WO1995032963A1 (en) * 1994-06-01 1995-12-07 Yoshitomi Pharmaceutical Industries, Ltd. Thienylazole compound and thienotriazolodiazepine compound
ATE230600T1 (en) * 1995-09-09 2003-01-15 Hoffmann La Roche USE OF A THIENOTRIAZOLEDIAZEPINE TO INCREASE APOLOPOPROTEIN A-I LEVELS

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904641A (en) * 1971-06-18 1975-09-09 Yoshitomi Pharmaceutical Triazolothienodiazepine compounds

Also Published As

Publication number Publication date
IE38883B1 (en) 1978-06-21
SU715028A3 (en) 1980-02-05
PL97275B1 (en) 1978-02-28
GB1456161A (en) 1976-11-17
IL44095A (en) 1979-03-12
NO142260C (en) 1980-07-23
DD112454A5 (en) 1975-04-12
DK137679B (en) 1978-04-17
NO142260B (en) 1980-04-14
LU69338A1 (en) 1975-12-09
BE810705A (en) 1974-08-07
CH584223A5 (en) 1977-01-31
CA1049009A (en) 1979-02-20
AR217034A1 (en) 1980-02-29
AU6485574A (en) 1975-07-24
HU170423B (en) 1977-06-28
DE2405682B2 (en) 1980-07-17
AT343118B (en) 1978-05-10
JPS5833234B2 (en) 1983-07-18
FR2217007B1 (en) 1978-02-03
NL7401117A (en) 1974-08-12
FI58129C (en) 1980-12-10
SE416399B (en) 1980-12-22
HU173741B (en) 1979-08-28
NL174045C (en) 1984-04-16
DE2405682C3 (en) 1981-03-12
IE38883L (en) 1974-08-08
AR203188A1 (en) 1975-08-22
DK137679C (en) 1978-09-25
JPS49102698A (en) 1974-09-27
NO740405L (en) 1974-08-09
FR2217007A1 (en) 1974-09-06
GB1456162A (en) 1976-11-17
IL44095A0 (en) 1974-05-16
ZA74472B (en) 1974-11-27
YU22874A (en) 1982-06-30
YU39716B (en) 1985-04-30
PL96107B1 (en) 1977-12-31
DE2405682A1 (en) 1974-08-15
FI58129B (en) 1980-08-29
SU747429A4 (en) 1980-07-23
PL97304B1 (en) 1978-02-28
SU1060115A3 (en) 1983-12-07
PH12303A (en) 1979-01-16
NL174045B (en) 1983-11-16

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Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties
ELA Expired due to lapse of time