NO141717C - Analogifremgangsmaate til fremstilling av farmakologisk aktive triazolopyridaziner - Google Patents

Analogifremgangsmaate til fremstilling av farmakologisk aktive triazolopyridaziner

Info

Publication number
NO141717C
NO141717C NO743140A NO743140A NO141717C NO 141717 C NO141717 C NO 141717C NO 743140 A NO743140 A NO 743140A NO 743140 A NO743140 A NO 743140A NO 141717 C NO141717 C NO 141717C
Authority
NO
Norway
Prior art keywords
triazolopyridazines
preparation
pharmacologically active
analogue procedure
analogue
Prior art date
Application number
NO743140A
Other languages
English (en)
Norwegian (no)
Other versions
NO743140L (xx
NO141717B (no
Inventor
Elvio Bellasio
Ambrogio Campi
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Publication of NO743140L publication Critical patent/NO743140L/no
Publication of NO141717B publication Critical patent/NO141717B/no
Publication of NO141717C publication Critical patent/NO141717C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO743140A 1973-09-21 1974-09-02 Analogifremgangsmaate til fremstilling av farmakologisk aktive triazolopyridaziner NO141717C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US399661A US3915968A (en) 1973-09-21 1973-09-21 Triazolopyridazines

Publications (3)

Publication Number Publication Date
NO743140L NO743140L (xx) 1975-04-14
NO141717B NO141717B (no) 1980-01-21
NO141717C true NO141717C (no) 1980-04-30

Family

ID=23580450

Family Applications (1)

Application Number Title Priority Date Filing Date
NO743140A NO141717C (no) 1973-09-21 1974-09-02 Analogifremgangsmaate til fremstilling av farmakologisk aktive triazolopyridaziner

Country Status (25)

Country Link
US (1) US3915968A (xx)
JP (1) JPS537439B2 (xx)
AR (2) AR206514A1 (xx)
AT (1) AT336604B (xx)
BE (1) BE820163A (xx)
CA (1) CA1034948A (xx)
CH (2) CH595382A5 (xx)
DD (1) DD113543A5 (xx)
DE (1) DE2444322C3 (xx)
DK (1) DK138692B (xx)
ES (2) ES430277A1 (xx)
FI (1) FI56013C (xx)
FR (1) FR2244519B1 (xx)
GB (1) GB1480621A (xx)
HU (1) HU171789B (xx)
IE (1) IE40651B1 (xx)
IL (1) IL45654A (xx)
LU (1) LU70949A1 (xx)
NL (1) NL7411849A (xx)
NO (1) NO141717C (xx)
PL (1) PL91748B1 (xx)
RO (1) RO64487A (xx)
SE (1) SE419990B (xx)
SU (2) SU576940A3 (xx)
ZA (1) ZA745482B (xx)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3994898A (en) * 1975-10-16 1976-11-30 E. R. Squibb & Sons, Inc. 1,2,4-Triazolo (4,3-b) pyridazin-3-ones
GR70309B (xx) * 1979-10-29 1982-09-08 Dow Chemical Co
US4526890A (en) * 1979-10-29 1985-07-02 The Dow Chemical Company 3,6,7,8-Substituted-s-triazolo[4,3-b]pyridazines as bronchodilators
US4260756A (en) * 1979-11-15 1981-04-07 American Cyanamid Company 6- And 8-heteroaryl-1,2,4-triazolo[4,3-b]pyridazines
US4293554A (en) * 1980-02-21 1981-10-06 American Cyanamid Company Method of treating asthma
US4487930A (en) * 1982-09-07 1984-12-11 The Dow Chemical Company 6-[(Cyclic amino)alkylamino]-tetrahydrotriazolo[3,4-a]phthalazines
DE3311753A1 (de) * 1983-03-31 1984-10-04 Hoechst Ag, 6230 Frankfurt Substituierte 6-aryl-1,2,4-triazolo(4,3-b)pyridazine - ihre herstellung und verwendung -
US4578464A (en) * 1983-11-22 1986-03-25 Merrell Dow Pharmaceuticals Inc. 6-Hydroxyalkylamino-8-methyl-1,2,4-triazolo-[4,3-b]pyridazine and related compounds
ZA873934B (en) * 1986-06-05 1987-12-02 Merrell Dow Pharmaceuticals Inc. 2,3-dihydro-1-(8-methyl-1,2,4-triazolo(4,3-b)pyridazin-6-yl)-4(1h)-pyridinone
US5011835A (en) * 1990-02-07 1991-04-30 Merrell Dow Pharmaceuticals Inc. Substituted triazolopyridazines, pharmaceutical compositions and use
FR2668151A1 (fr) * 1990-10-23 1992-04-24 Rhone Poulenc Agrochimie Composes a groupe triazolopyridazine leurs preparations et compositions herbicides les contenant.
LT3200B (en) 1992-03-18 1995-03-27 Takeda Chemical Industries Ltd Triazolopyridazine methodfor production thereof and use
CA2120997A1 (en) * 1993-04-12 1994-10-13 Akio Miyake Triazolopyridazine derivatives, their production and use
WO2003074525A1 (fr) 2002-03-01 2003-09-12 Yamanouchi Pharmaceutical Co., Ltd. Compose heterocyclique azote
CA2498237A1 (en) * 2002-09-13 2004-03-25 Merck & Co., Inc. Fused heterobicyclo substituted phenyl metabotropic glutamate-5 modulators
US9422290B2 (en) 2012-11-13 2016-08-23 Boehringer Ingelheim International Gmbh Triazolopyridazine
US9266891B2 (en) 2012-11-16 2016-02-23 Boehringer Ingelheim International Gmbh Substituted [1,2,4]triazolo[4,3-A]pyrazines that are BRD4 inhibitors
GB201321745D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
CN112142744A (zh) * 2019-06-28 2020-12-29 上海瑛派药业有限公司 取代的稠合杂芳双环化合物作为激酶抑制剂及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1248409A (fr) * 1957-06-13 1960-12-16 Bellon Labor Sa Roger Perfectionnements aux procédés de préparation de dérivés de la triazolo [4-3,b]pyridazine
DE2161586A1 (de) * 1971-12-11 1973-06-14 Boehringer Mannheim Gmbh Nitrofuryl-triazolo eckige klammer auf 4,3-b eckige klammer zu pyridazin-derivate

Also Published As

Publication number Publication date
SU576940A3 (ru) 1977-10-15
CH595382A5 (xx) 1978-02-15
IL45654A (en) 1977-07-31
FI56013C (fi) 1979-11-12
DK138692B (da) 1978-10-16
DE2444322A1 (de) 1975-03-27
NO743140L (xx) 1975-04-14
DE2444322C3 (de) 1981-03-19
DD113543A5 (xx) 1975-06-12
DK138692C (xx) 1979-03-19
DK496374A (xx) 1975-05-20
LU70949A1 (xx) 1975-03-06
NO141717B (no) 1980-01-21
HU171789B (hu) 1978-03-28
IL45654A0 (en) 1974-11-29
DE2444322B2 (de) 1980-08-07
GB1480621A (en) 1977-07-20
SE7411888L (xx) 1975-03-24
IE40651B1 (en) 1979-07-18
FI56013B (fi) 1979-07-31
AU7305374A (en) 1976-03-11
FR2244519A1 (xx) 1975-04-18
RO64487A (fr) 1979-06-15
SE419990B (sv) 1981-09-07
PL91748B1 (xx) 1977-03-31
CA1034948A (en) 1978-07-18
JPS5058092A (xx) 1975-05-20
CH599212A5 (xx) 1978-05-12
ES432243A1 (es) 1977-04-16
FR2244519B1 (xx) 1978-07-21
US3915968A (en) 1975-10-28
ZA745482B (en) 1975-09-24
FI265674A (xx) 1975-03-22
NL7411849A (nl) 1975-03-25
ES430277A1 (es) 1976-12-16
ATA755074A (de) 1976-09-15
IE40651L (en) 1975-03-21
AR206514A1 (es) 1976-07-30
BE820163A (fr) 1975-01-16
AT336604B (de) 1977-05-10
JPS537439B2 (xx) 1978-03-17
SU545261A3 (ru) 1977-01-30
AR206643A1 (es) 1976-08-06

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