NO138599C - Analogifremgangsmaate til fremstilling av nye, terapeutisk virksomme tienopyrimidinderivater - Google Patents

Analogifremgangsmaate til fremstilling av nye, terapeutisk virksomme tienopyrimidinderivater

Info

Publication number
NO138599C
NO138599C NO1903/73A NO190373A NO138599C NO 138599 C NO138599 C NO 138599C NO 1903/73 A NO1903/73 A NO 1903/73A NO 190373 A NO190373 A NO 190373A NO 138599 C NO138599 C NO 138599C
Authority
NO
Norway
Prior art keywords
tienopyrimidin
analogical
procedures
derivatives
preparation
Prior art date
Application number
NO1903/73A
Other languages
English (en)
Norwegian (no)
Other versions
NO138599B (no
Inventor
Toshiyuki Hirohashi
Hiromi Sato
Shigeho Inaba
Hisao Yamamoto
Original Assignee
Sumitomo Chemical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP4603872A external-priority patent/JPS495994A/ja
Priority claimed from JP6682872A external-priority patent/JPS4926294A/ja
Priority claimed from JP7542072A external-priority patent/JPS4931695A/ja
Priority claimed from JP12367472A external-priority patent/JPS4980093A/ja
Priority claimed from JP12594672A external-priority patent/JPS4981390A/ja
Application filed by Sumitomo Chemical Co filed Critical Sumitomo Chemical Co
Publication of NO138599B publication Critical patent/NO138599B/no
Publication of NO138599C publication Critical patent/NO138599C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/36Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/66Nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO1903/73A 1972-05-09 1973-05-08 Analogifremgangsmaate til fremstilling av nye, terapeutisk virksomme tienopyrimidinderivater NO138599C (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP4603872A JPS495994A (zh) 1972-05-09 1972-05-09
JP6682872A JPS4926294A (zh) 1972-07-03 1972-07-03
JP7542072A JPS4931695A (zh) 1972-07-26 1972-07-26
JP12367472A JPS4980093A (zh) 1972-12-09 1972-12-09
JP12594672A JPS4981390A (zh) 1972-12-14 1972-12-14

Publications (2)

Publication Number Publication Date
NO138599B NO138599B (no) 1978-06-26
NO138599C true NO138599C (no) 1978-10-04

Family

ID=27522520

Family Applications (1)

Application Number Title Priority Date Filing Date
NO1903/73A NO138599C (no) 1972-05-09 1973-05-08 Analogifremgangsmaate til fremstilling av nye, terapeutisk virksomme tienopyrimidinderivater

Country Status (12)

Country Link
US (1) US3957783A (zh)
AT (1) AT329066B (zh)
CA (1) CA997344A (zh)
CH (1) CH586706A5 (zh)
DE (1) DE2323149C3 (zh)
DK (1) DK132498C (zh)
FI (1) FI54312C (zh)
FR (1) FR2183950B1 (zh)
GB (1) GB1397501A (zh)
HU (1) HU169934B (zh)
NL (1) NL7306403A (zh)
NO (1) NO138599C (zh)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4230707A (en) * 1979-08-27 1980-10-28 Warner-Lambert Company Oxo-pyrido[1,2-a]thienopyrimidine compounds and methods for their production
US4703120A (en) * 1986-04-28 1987-10-27 Ortho Pharmaceutical Corporation Furo(3,4-d)pyrimidine-2,4-dione derivatives and intermediates thereof
US6323214B1 (en) 1997-10-29 2001-11-27 Medco Research, Inc Allosteric adenosine receptor modulators
US5939432A (en) * 1997-10-29 1999-08-17 Medco Research, Inc. Thiophenes useful for modulating the adenosine receptor
US6727258B2 (en) 1997-10-29 2004-04-27 King Pharmaceutical Research & Development, Inc. Allosteric adenosine receptor modulators
US7928111B2 (en) * 2007-06-08 2011-04-19 Senomyx, Inc. Compounds including substituted thienopyrimidinone derivatives as ligands for modulating chemosensory receptors
US9603848B2 (en) 2007-06-08 2017-03-28 Senomyx, Inc. Modulation of chemosensory receptors and ligands associated therewith
US8633186B2 (en) * 2007-06-08 2014-01-21 Senomyx Inc. Modulation of chemosensory receptors and ligands associated therewith
US8609173B2 (en) 2008-07-31 2013-12-17 Senomyx Inc. Compositions comprising sweetness enhancers and methods of making them
MY153622A (en) 2008-07-31 2015-02-27 Senomyx Inc Processes and intermediates for making sweet taste enhancers
RU2576451C2 (ru) 2010-08-12 2016-03-10 Синомикс, Инк. Способ улучшения стабильности усилителей сладкого вкуса и композиция, содержащая стабилизированный усилитель сладкого вкуса
AU2013299859B2 (en) 2012-08-06 2017-06-15 Firmenich Incorporated Sweet flavor modifier
JO3155B1 (ar) 2013-02-19 2017-09-20 Senomyx Inc معدِّل نكهة حلوة
BR112021002261A2 (pt) 2018-08-07 2021-05-04 Firmenich Incorporated 2,2-dióxidos de 4-amino-1h-benzo[c][1,2,6]tiadiazina 5-substituídos e formulações e usos dos mesmos

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2117658A1 (de) * 1971-04-10 1972-10-19 Dr. Karl Thomae GmbH, 7951 Biberach Neue 2-(5-Nitro-2-furyl)-thieno eckige Klammer auf 2,3-d eckige Klammer zu pyrimidine und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
FR2183950A1 (zh) 1973-12-21
NO138599B (no) 1978-06-26
FI54312C (fi) 1978-11-10
DK132498C (da) 1976-05-17
ATA408373A (de) 1975-07-15
DE2323149B2 (de) 1978-06-29
NL7306403A (zh) 1973-11-13
GB1397501A (en) 1975-06-11
FR2183950B1 (zh) 1976-07-02
AT329066B (de) 1976-04-26
CH586706A5 (zh) 1977-04-15
HU169934B (zh) 1977-02-28
DK132498B (da) 1975-12-15
FI54312B (fi) 1978-07-31
US3957783A (en) 1976-05-18
DE2323149A1 (de) 1973-11-22
CA997344A (en) 1976-09-21
DE2323149C3 (de) 1979-02-22

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