NL8003141A - Biologisch aktieve tricyclische aminen. - Google Patents

Biologisch aktieve tricyclische aminen. Download PDF

Info

Publication number
NL8003141A
NL8003141A NL8003141A NL8003141A NL8003141A NL 8003141 A NL8003141 A NL 8003141A NL 8003141 A NL8003141 A NL 8003141A NL 8003141 A NL8003141 A NL 8003141A NL 8003141 A NL8003141 A NL 8003141A
Authority
NL
Netherlands
Prior art keywords
hexahydro
hcl
phenalen
compounds
cis
Prior art date
Application number
NL8003141A
Other languages
English (en)
Dutch (nl)
Original Assignee
Akzo Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nv filed Critical Akzo Nv
Priority to NL8003141A priority Critical patent/NL8003141A/nl
Priority to AU71730/81A priority patent/AU546950B2/en
Priority to JP56501692A priority patent/JPS57500734A/ja
Priority to PCT/EP1981/000055 priority patent/WO1981003490A1/de
Priority to AT81200545T priority patent/ATE6635T1/de
Priority to EP81200545A priority patent/EP0041293B1/en
Priority to DE8181200545T priority patent/DE3162608D1/de
Priority to IE1144/81A priority patent/IE51611B1/en
Priority to ZA00813498A priority patent/ZA813498B/xx
Priority to PT73081A priority patent/PT73081B/pt
Priority to GR65098A priority patent/GR74556B/el
Priority to ES502629A priority patent/ES8207500A1/es
Priority to CA000378600A priority patent/CA1157472A/en
Priority to HU811801A priority patent/HU183490B/hu
Priority to DK452681A priority patent/DK152284C/da
Priority to FI813437A priority patent/FI67535C/fi
Publication of NL8003141A publication Critical patent/NL8003141A/nl
Priority to US06/460,259 priority patent/US4564698A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NL8003141A 1980-05-30 1980-05-30 Biologisch aktieve tricyclische aminen. NL8003141A (nl)

Priority Applications (17)

Application Number Priority Date Filing Date Title
NL8003141A NL8003141A (nl) 1980-05-30 1980-05-30 Biologisch aktieve tricyclische aminen.
AU71730/81A AU546950B2 (en) 1980-05-30 1981-05-21 Biologically-active tricyclic amines,methods for their preparation and pharmaceutical compositions containing same
JP56501692A JPS57500734A (fi) 1980-05-30 1981-05-21
PCT/EP1981/000055 WO1981003490A1 (en) 1980-05-30 1981-05-21 Biologically-active tricyclic amines,methods for their preparation and pharmaceutical compositions containing same
AT81200545T ATE6635T1 (de) 1980-05-30 1981-05-21 Biologisch aktive trizyklische amine, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate.
EP81200545A EP0041293B1 (en) 1980-05-30 1981-05-21 Biologically-active tricyclic amines, methods for their preparation and pharmaceutical compositions containing same
DE8181200545T DE3162608D1 (en) 1980-05-30 1981-05-21 Biologically-active tricyclic amines, methods for their preparation and pharmaceutical compositions containing same
IE1144/81A IE51611B1 (en) 1980-05-30 1981-05-22 Biologically-active tricyclic amines,methods for their preparation and pharmaceutical compositions containing same
ZA00813498A ZA813498B (en) 1980-05-30 1981-05-25 Biologically-active tricyclic amines,methods for their preparation and pharmaceutical compositions containing same
PT73081A PT73081B (en) 1980-05-30 1981-05-25 Biologically-active tricyclic amines methods for their preparation and pharmaceutical compositions containing same
GR65098A GR74556B (fi) 1980-05-30 1981-05-28
ES502629A ES8207500A1 (es) 1980-05-30 1981-05-29 Un procedimiento para la preparacion de nuevos compuestos triciclicos.
CA000378600A CA1157472A (en) 1980-05-30 1981-05-29 Biologically-active tricyclic amines, methods for their preparation and pharmaceutical compositions containing same
HU811801A HU183490B (en) 1980-05-30 1981-09-21 Process for producing biologically active tricyclic amines
DK452681A DK152284C (da) 1980-05-30 1981-10-13 Analogifremgangsmaade til fremstilling af tricykliske aminer
FI813437A FI67535C (fi) 1980-05-30 1981-11-02 Foerfarande foer framstaellning av nya biologiskt aktiva tricykliska aminer
US06/460,259 US4564698A (en) 1980-05-30 1983-01-24 Biologically-active tricyclic amines

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
NL8003141A NL8003141A (nl) 1980-05-30 1980-05-30 Biologisch aktieve tricyclische aminen.
NL8003141 1980-05-30

Publications (1)

Publication Number Publication Date
NL8003141A true NL8003141A (nl) 1982-01-04

Family

ID=19835385

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8003141A NL8003141A (nl) 1980-05-30 1980-05-30 Biologisch aktieve tricyclische aminen.

Country Status (17)

Country Link
US (1) US4564698A (fi)
EP (1) EP0041293B1 (fi)
JP (1) JPS57500734A (fi)
AT (1) ATE6635T1 (fi)
AU (1) AU546950B2 (fi)
CA (1) CA1157472A (fi)
DE (1) DE3162608D1 (fi)
DK (1) DK152284C (fi)
ES (1) ES8207500A1 (fi)
FI (1) FI67535C (fi)
GR (1) GR74556B (fi)
HU (1) HU183490B (fi)
IE (1) IE51611B1 (fi)
NL (1) NL8003141A (fi)
PT (1) PT73081B (fi)
WO (1) WO1981003490A1 (fi)
ZA (1) ZA813498B (fi)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0234113A1 (en) * 1985-12-31 1987-09-02 The Upjohn Company 2,3-Dihydro-1H-phenalene-2-amino compounds as anti-psychotic drugs
AU3563389A (en) * 1988-05-09 1989-11-29 Upjohn Company, The Anxiolytic/anti-depressant 2,3-dihydro-1h-phenalen-2-amines
US5055414A (en) * 1988-07-05 1991-10-08 Eastman Kodak Company Phenalenimine fluorescent dyes and their use in analytical methods
IE892812L (en) * 1988-09-12 1990-03-12 Brendan Coleman Tricyclic aromatase inhibitors
FR2732964B1 (fr) * 1995-04-14 1997-05-16 Adir Nouveaux amides tricycliques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2589934A (en) * 1950-08-24 1952-03-18 Abbott Lab 2-aminomethyl-tetrahydroacenapthones-1 and their preparation
US3198835A (en) * 1960-07-25 1965-08-03 Sterling Drug Inc Pyrenyl methyl tertiary amino amines
US3553093A (en) * 1965-03-19 1971-01-05 Xerox Corp Color photoelectrophoretic imaging process
US3637740A (en) * 1969-04-21 1972-01-25 Pfizer Aminobenzocycloalkane compounds
US3912781A (en) * 1969-06-24 1975-10-14 Ruetgerswerke Ag 1-hydroxymethyl-1,2,3,4-tetrahydrofluoranthene
US3732299A (en) * 1969-11-03 1973-05-08 Squibb & Sons Inc Acenaphthene carboxamides
US3763233A (en) * 1971-08-17 1973-10-02 Sandoz Ag 7-substituted-hexahydro pleiadenes
DE2252945A1 (de) * 1971-11-19 1974-05-09 Basf Ag L-aminomethyl-acenaphthene und verfahren zu ihrer herstellung
NL7306069A (fi) * 1973-05-02 1974-11-05
JPS52133993A (en) * 1976-04-29 1977-11-09 Takeda Chem Ind Ltd 1.2-dihydronaphthalene derivatives and method of preparing the same
GB1590648A (en) * 1976-12-01 1981-06-03 Ciba Geigy Ag N-((naphthothienyl or n-phenanthryl)alkyl) imidazoles their preparation and compositions containing them
DE2862103D1 (en) * 1977-08-19 1982-11-18 Sandoz Ag Propenyl amines, processes for their production and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
DE3162608D1 (en) 1984-04-19
DK152284B (da) 1988-02-15
JPS57500734A (fi) 1982-04-30
EP0041293B1 (en) 1984-03-14
ES502629A0 (es) 1982-10-01
US4564698A (en) 1986-01-14
GR74556B (fi) 1984-06-29
IE811144L (en) 1981-11-30
PT73081A (en) 1981-06-01
ES8207500A1 (es) 1982-10-01
DK452681A (da) 1981-12-10
WO1981003490A1 (en) 1981-12-10
AU546950B2 (en) 1985-09-26
HU183490B (en) 1984-05-28
CA1157472A (en) 1983-11-22
ATE6635T1 (de) 1984-03-15
AU7173081A (en) 1981-12-21
FI67535C (fi) 1985-04-10
EP0041293A1 (en) 1981-12-09
FI67535B (fi) 1984-12-31
DK152284C (da) 1988-08-08
ZA813498B (en) 1982-06-30
PT73081B (en) 1984-10-22
IE51611B1 (en) 1987-01-21
FI813437L (fi) 1981-11-02

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BV The patent application has lapsed