NL7509075A - Werkwijze voor de bereiding van nieuwe 17(alpha),21- -diesters van 17(alpha),21-dihydroxysteroiden uit de pregnaanreeks. - Google Patents
Werkwijze voor de bereiding van nieuwe 17(alpha),21- -diesters van 17(alpha),21-dihydroxysteroiden uit de pregnaanreeks.Info
- Publication number
- NL7509075A NL7509075A NL7509075A NL7509075A NL7509075A NL 7509075 A NL7509075 A NL 7509075A NL 7509075 A NL7509075 A NL 7509075A NL 7509075 A NL7509075 A NL 7509075A NL 7509075 A NL7509075 A NL 7509075A
- Authority
- NL
- Netherlands
- Prior art keywords
- alpha
- dihydroxysteroids
- diesters
- preparation
- new
- Prior art date
Links
- 150000005690 diesters Chemical class 0.000 title 1
- JWMFYGXQPXQEEM-WZBAXQLOSA-N pregnane Chemical class C1CC2CCCC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](CC)[C@@]1(C)CC2 JWMFYGXQPXQEEM-WZBAXQLOSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0088—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing unsubstituted amino radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0061—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16
- C07J5/0069—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group
- C07J5/0076—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa substituted in position 16 by a saturated or unsaturated hydrocarbon group by an alkyl group
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB33786/74A GB1516095A (en) | 1974-07-31 | 1974-07-31 | 17,21-diesters of 17alpha,21-dihydroxy-steroids of the pregnane series |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NL7509075A true NL7509075A (nl) | 1976-02-03 |
Family
ID=10357423
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NL7509075A NL7509075A (nl) | 1974-07-31 | 1975-07-30 | Werkwijze voor de bereiding van nieuwe 17(alpha),21- -diesters van 17(alpha),21-dihydroxysteroiden uit de pregnaanreeks. |
Country Status (13)
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4456602A (en) * | 1982-08-23 | 1984-06-26 | The Upjohn Company | Amine containing ester prodrugs of corticosteroids |
| US4443440A (en) * | 1982-08-30 | 1984-04-17 | The Upjohn Company | Amine containing ester prodrugs of corticosteroids |
| FR2600653B1 (fr) * | 1986-06-24 | 1988-12-16 | Pasteur Strasbourg Universite | Composes de synthese associative d'acides amines soufres ou non soufres avec des derives du d-4 pregnene 3,20-dione ou avec des derives du d-1,4 pregnadiene 3,20-dione aux proprietes glucocorticoides et anti-inflammatoires, procedes d'obtention, compositions pharmaceutiques les contenant. proprietes pharmacologiques et applications |
| DE4333920A1 (de) | 1993-10-05 | 1995-04-13 | Hoechst Ag | Corticoid-17,21-dicarbonsäureester sowie Corticosteroid-17-carbonsäureester-21-kohlensäureester, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1044212B (it) * | 1971-03-17 | 1980-03-20 | Sigma Tau Ind Farmaceuti | Esteri del besametazone e betametazone |
| GB1440063A (en) * | 1972-08-11 | 1976-06-23 | Glaxo Lab Ltd | 17alpha-esters of 17alpha,21-dihydroxy-20-oxo-steroids |
-
1974
- 1974-07-31 GB GB33786/74A patent/GB1516095A/en not_active Expired
-
1975
- 1975-07-30 CH CH996575A patent/CH615442A5/de not_active IP Right Cessation
- 1975-07-30 ES ES439852A patent/ES439852A1/es not_active Expired
- 1975-07-30 ZA ZA00754907A patent/ZA754907B/xx unknown
- 1975-07-30 DK DK346975AA patent/DK139303B/da unknown
- 1975-07-30 NL NL7509075A patent/NL7509075A/xx not_active Application Discontinuation
- 1975-07-30 SE SE7508654A patent/SE7508654L/xx unknown
- 1975-07-30 IE IE1708/75A patent/IE42124B1/en unknown
- 1975-07-30 JP JP50092137A patent/JPS51125059A/ja active Pending
- 1975-07-30 CA CA232,579A patent/CA1058610A/en not_active Expired
- 1975-07-30 DE DE19752534051 patent/DE2534051A1/de not_active Withdrawn
- 1975-07-30 BE BE158780A patent/BE831931A/xx unknown
- 1975-07-30 FR FR7523787A patent/FR2280383A1/fr active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| CH615442A5 (en) | 1980-01-31 |
| FR2280383B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1978-10-06 |
| JPS51125059A (en) | 1976-11-01 |
| IE42124B1 (en) | 1980-06-04 |
| ZA754907B (en) | 1976-07-28 |
| DK139303B (da) | 1979-01-29 |
| BE831931A (fr) | 1976-01-30 |
| SE7508654L (sv) | 1976-02-02 |
| CA1058610A (en) | 1979-07-17 |
| AU8353175A (en) | 1977-02-03 |
| DE2534051A1 (de) | 1976-02-19 |
| DK139303C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1979-08-06 |
| FR2280383A1 (fr) | 1976-02-27 |
| IE42124L (en) | 1976-01-31 |
| DK346975A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1976-02-01 |
| ES439852A1 (es) | 1977-03-01 |
| GB1516095A (en) | 1978-06-28 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NL7606042A (nl) | Werkwijze ter bereiding van zeer zuivere stikstof uit lucht. | |
| NL7506806A (nl) | Werkwijze voor de bereiding van nieuwe benzimida- zolen. | |
| NL7414283A (nl) | Werkwijze voor de bereiding van silanen. | |
| NL7508824A (nl) | Werkwijze voor de bereiding van nieuwe chinazoline- derivaten. | |
| NL7504572A (nl) | Werkwijze voor de bereiding van gesubstitueerde formamidinen. | |
| NL7603249A (nl) | Werkwijze voor de bereiding van 17(alpha)-ester-21-ha- logeenpregnanen. | |
| NL7415432A (nl) | Werkwijze voor de bereiding van nieuwe 7(alpha)-me- thoxycefalosporineverbindingen. | |
| NL7606579A (nl) | Werkwijze voor de bereiding van (alpha)-hydroxyisobu- tyramide uit acetoncyaanhydrien. | |
| NL7412230A (nl) | Werkwijze voor de bereiding van organotintri- halogeniden. | |
| NL7509281A (nl) | Werkwijze voor de bereiding van oligomeren uit lineaire (alpha)-alkenen. | |
| NL7509276A (nl) | Werkwijze voor de bereiding van tertiaire alkenen. | |
| NL7509913A (nl) | Werkwijze voor de bereiding van nieuwe benziso- chinolinederivaten. | |
| NL153205B (nl) | Werkwijze voor de bereiding van organotintrihalogeniden. | |
| NL7509280A (nl) | Werkwijze voor de bereiding van oligomeren uit lineaire (alpha)-alkenen. | |
| NL7610513A (nl) | Werkwijze voor de bereiding van nieuwe n-aryl-n-(1-l-4-piperidinyl)arylaceetamiden. | |
| NL7504135A (nl) | Werkwijze voor de bereiding van gesubstitueerde indoleninen. | |
| NL7509160A (nl) | Werkwijze voor de bereiding van 1,4-naftochinon. | |
| NL7509980A (nl) | Werkwijze voor de bereiding van 7(beta)-acylamino- -7(alpha)-alkoxycefalosporinen. | |
| NL7603449A (nl) | Werkwijze voor de bereiding van (alpha)-fenylpropion- zuren. | |
| NL7509075A (nl) | Werkwijze voor de bereiding van nieuwe 17(alpha),21- -diesters van 17(alpha),21-dihydroxysteroiden uit de pregnaanreeks. | |
| NL7509556A (nl) | Werkwijze voor de bereiding van 17(alpha)-hydroxy-1,3, 5(10), 15-oestratetraenen. | |
| NL7514010A (nl) | Werkwijze voor de bereiding van nieuwe 5-nitroimi- dazolen. | |
| NL7505461A (nl) | Werkwijze voor de bereiding van (alpha)-aminoacyl- penicilline-derivaten. | |
| BE824892A (nl) | Werkwijze voor de bereiding van n,n-diallyldichloor aceetamide | |
| NL7408524A (nl) | Werkwijze voor het bereiden van 17-acylesters 7(alpha),21-dihydroxysteroiden van de pregnaan- . |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BV | The patent application has lapsed |