NL1025844A1 - Benzopyranverbindingen voor gebruik bij de behandeling en preventie van ontstekingsgerelateerde aandoeningen. - Google Patents

Benzopyranverbindingen voor gebruik bij de behandeling en preventie van ontstekingsgerelateerde aandoeningen.

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Publication number
NL1025844A1
NL1025844A1 NL1025844A NL1025844A NL1025844A1 NL 1025844 A1 NL1025844 A1 NL 1025844A1 NL 1025844 A NL1025844 A NL 1025844A NL 1025844 A NL1025844 A NL 1025844A NL 1025844 A1 NL1025844 A1 NL 1025844A1
Authority
NL
Netherlands
Prior art keywords
prevention
treatment
inflammatory diseases
benzopyran compounds
benzopyran
Prior art date
Application number
NL1025844A
Other languages
English (en)
Other versions
NL1025844C2 (nl
Inventor
Karl William Aston
David Louis Brown
Jeffrey Steven Carter
Angela M Deprow
Theresa R Fletcher
E Ann Hallinan
Bruce Cameron Hamper
Renee M Huff
James Richard Kiefer Jr
Francis Koszyk
Steven W Kramer
Subo Liao
David Christopher Limburg
John Robert Springer
Sofya Tsymbalov
Lijuan Jane Wang
Li Xing
Yi Yu
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of NL1025844A1 publication Critical patent/NL1025844A1/nl
Application granted granted Critical
Publication of NL1025844C2 publication Critical patent/NL1025844C2/nl

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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NL1025844A 2003-03-31 2004-03-29 Benzopyranverbindingen voor gebruik bij de behandeling en preventie van ontstekingsgerelateerde aandoeningen. NL1025844C2 (nl)

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US45921403P 2003-03-31 2003-03-31
US45921403 2003-03-31

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NL1025844A1 true NL1025844A1 (nl) 2004-10-01
NL1025844C2 NL1025844C2 (nl) 2005-03-01

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US6034256A (en) * 1997-04-21 2000-03-07 G.D. Searle & Co. Substituted benzopyran derivatives for the treatment of inflammation
WO2006011052A1 (en) * 2004-07-23 2006-02-02 Pharmacia & Upjohn Company Llc Method for the racemization of 2-trifluoro-2h-chromene-3-carboxylic acids
WO2006011045A1 (en) * 2004-07-23 2006-02-02 Warner-Lambert Company Llc Photoracemization of 2-trifluoromethyl-2h-chromene-3-carboxylic acid derivatives
BRPI0512251A (pt) * 2004-07-23 2008-02-19 Pharmacia & Upjohn Co Llc método enantioseletivo para separação de derivados do ácido 2-trifluormetil-2h-cromeno-3-carboxìlico substituìdo
WO2006040676A1 (en) * 2004-10-12 2006-04-20 Pharmacia & Upjohn Company Llc Nitrosated benzopyran compounds as novel cyclooxygenase-2 selective inhibitors
GB0608825D0 (en) * 2006-05-04 2006-06-14 Glaxo Group Ltd Compounds
CN102757417B (zh) 2012-06-18 2014-09-24 中国科学院广州生物医药与健康研究院 氘代苯并吡喃类化合物及其应用
JP6061373B2 (ja) * 2012-07-24 2017-01-18 国立研究開発法人産業技術総合研究所 2−ヒドロキシベンズアルデヒド化合物、これを含有するコラーゲン細胞外分泌阻害剤及び医薬品組成物
CN103012350B (zh) * 2012-12-07 2015-02-04 中国科学院广州生物医药与健康研究院 苯并吡喃类手性化合物的合成方法
EP3094333B1 (en) * 2014-01-14 2020-10-14 Euclises Pharmaceuticals, Inc. No-releasing nitrooxy-chromene conjugates
EP3126451B1 (en) 2014-04-01 2020-09-09 Howard Hughes Medical Institute Azetidine-substituted fluorescent compounds
EP3310822B1 (en) * 2015-06-19 2023-10-11 SABIC Global Technologies B.V. Procatalyst for polymerization of olefins comprising an aminobenzoate internal donor and a 1,3-diether internal donor in a specific ratio
GB2543550A (en) 2015-10-21 2017-04-26 Hox Therapeutics Ltd Peptides
WO2020120528A1 (en) * 2018-12-14 2020-06-18 F. Hoffmann-La Roche Ag N-containing chromen-4-one derivatives for the treatment and prophylaxis of hepatitis b virus infection

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US6034256A (en) * 1997-04-21 2000-03-07 G.D. Searle & Co. Substituted benzopyran derivatives for the treatment of inflammation

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UY28247A1 (es) 2004-11-08
CL2004000664A1 (es) 2005-02-04
CA2519291A1 (en) 2004-10-14
US20050148627A1 (en) 2005-07-07
TW200504045A (en) 2005-02-01
AR043951A1 (es) 2005-08-17
NL1025844C2 (nl) 2005-03-01
PE20050393A1 (es) 2005-05-30
BRPI0408389A (pt) 2006-03-01
JP2006522091A (ja) 2006-09-28
EP1631562A1 (en) 2006-03-08
WO2004087687A1 (en) 2004-10-14
PA8599301A1 (es) 2004-12-16
MXPA05010423A (es) 2006-04-24

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