MXPA03007624A - Procedimiento para la preparacion de (e)-5-(2-bromovinil)-2-desoxiuridina. - Google Patents

Procedimiento para la preparacion de (e)-5-(2-bromovinil)-2-desoxiuridina.

Info

Publication number
MXPA03007624A
MXPA03007624A MXPA03007624A MXPA03007624A MXPA03007624A MX PA03007624 A MXPA03007624 A MX PA03007624A MX PA03007624 A MXPA03007624 A MX PA03007624A MX PA03007624 A MXPA03007624 A MX PA03007624A MX PA03007624 A MXPA03007624 A MX PA03007624A
Authority
MX
Mexico
Prior art keywords
bromovinyl
deoxyuridine
preparation
Prior art date
Application number
MXPA03007624A
Other languages
English (en)
Inventor
Stefano Manzini
Original Assignee
Menarini Ricerche Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7675814&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MXPA03007624(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Menarini Ricerche Spa filed Critical Menarini Ricerche Spa
Publication of MXPA03007624A publication Critical patent/MXPA03007624A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/20Antivirals for DNA viruses
    • A61P31/22Antivirals for DNA viruses for herpes viruses
MXPA03007624A 2001-02-28 2002-02-21 Procedimiento para la preparacion de (e)-5-(2-bromovinil)-2-desoxiuridina. MXPA03007624A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10109657A DE10109657A1 (de) 2001-02-28 2001-02-28 Verfahren zur Herstellung von (E)-5-(2-Bromvinyl)-2`-desoxyuridin
PCT/EP2002/001833 WO2002068443A1 (en) 2001-02-28 2002-02-21 Process for the preparation of (e)-5-(2-bromovinyl)-2'-deoxyuridine

Publications (1)

Publication Number Publication Date
MXPA03007624A true MXPA03007624A (es) 2003-12-04

Family

ID=7675814

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03007624A MXPA03007624A (es) 2001-02-28 2002-02-21 Procedimiento para la preparacion de (e)-5-(2-bromovinil)-2-desoxiuridina.

Country Status (32)

Country Link
US (1) US6864366B2 (es)
EP (1) EP1363928B1 (es)
JP (1) JP2004521132A (es)
KR (1) KR100853280B1 (es)
CN (1) CN1219789C (es)
AR (1) AR032908A1 (es)
AT (1) ATE294810T1 (es)
BG (1) BG66333B1 (es)
BR (1) BRPI0207566B8 (es)
CA (1) CA2439319C (es)
CZ (1) CZ299318B6 (es)
DE (2) DE10109657A1 (es)
DK (1) DK1363928T3 (es)
EA (1) EA006156B1 (es)
EE (1) EE05249B1 (es)
ES (1) ES2239713T3 (es)
HK (1) HK1060134A1 (es)
HR (1) HRP20030671B1 (es)
HU (1) HU229136B1 (es)
IL (2) IL157573A0 (es)
MA (1) MA26267A1 (es)
MX (1) MXPA03007624A (es)
MY (1) MY133371A (es)
PE (1) PE20020892A1 (es)
PL (1) PL210150B1 (es)
PT (1) PT1363928E (es)
RS (1) RS50761B (es)
SK (1) SK287283B6 (es)
TN (1) TNSN03049A1 (es)
UA (1) UA75110C2 (es)
WO (1) WO2002068443A1 (es)
ZA (1) ZA200306639B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101066987B (zh) * 2007-06-14 2010-05-19 上海交通大学 溴呋啶的制备方法
PL3447061T3 (pl) 2011-03-01 2022-01-31 NuCana plc Farmaceutyczna formulacja zawierająca pochodną fosforoamidynianową 5-fluoro-2'-deoksyurydyny do zastosowania w leczeniu nowotworu
GB201715011D0 (en) 2017-09-18 2017-11-01 Nucana Biomed Ltd Floxuridine synthesis
CN115043894A (zh) * 2022-06-22 2022-09-13 华润双鹤药业股份有限公司 一种溴夫定起始物料异构体单晶及其制备方法和应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB215399A (en) * 1922-11-07 1924-05-07 Frederic Valerius Hetzel Improvements in sprocket-wheels
GB1601020A (en) 1978-04-24 1981-10-21 Stichting Grega Vzw 2'-deoxy-5 (2-halogenovinyl)-uridines
HU187736B (en) * 1982-08-04 1986-02-28 Mta Koezponti Kemiai Kutato Intezet,Hu Process for producing /e/ -5-/2-bromovinyl/-2-comma above-deoxyuridine and o-acyl derivatives
DE59202433D1 (de) * 1991-05-06 1995-07-13 Ciba Geigy Ag Verfahren zur Herstellung von Benzolsulfonamiden.

Also Published As

Publication number Publication date
CA2439319C (en) 2010-10-19
BG108129A (bg) 2004-12-30
HRP20030671B1 (en) 2011-11-30
DE60203998D1 (de) 2005-06-09
EP1363928B1 (en) 2005-05-04
CA2439319A1 (en) 2002-09-06
SK10642003A3 (sk) 2004-01-08
PE20020892A1 (es) 2002-12-26
CZ20032295A3 (cs) 2004-01-14
HK1060134A1 (en) 2004-07-30
US6864366B2 (en) 2005-03-08
EE05249B1 (et) 2009-12-15
EA006156B1 (ru) 2005-10-27
US20040077586A1 (en) 2004-04-22
BR0207566A (pt) 2004-09-14
TNSN03049A1 (en) 2005-12-23
JP2004521132A (ja) 2004-07-15
HU229136B1 (en) 2013-08-28
HUP0303323A3 (en) 2008-12-29
HRP20030671A2 (en) 2005-06-30
KR100853280B1 (ko) 2008-08-20
SK287283B6 (sk) 2010-05-07
CZ299318B6 (cs) 2008-06-18
PL363611A1 (en) 2004-11-29
PT1363928E (pt) 2005-07-29
RS50761B (sr) 2010-08-31
AR032908A1 (es) 2003-12-03
CN1219789C (zh) 2005-09-21
WO2002068443A1 (en) 2002-09-06
PL210150B1 (pl) 2011-12-30
ATE294810T1 (de) 2005-05-15
ES2239713T3 (es) 2005-10-01
CN1494550A (zh) 2004-05-05
MY133371A (en) 2007-11-30
DK1363928T3 (da) 2005-12-12
IL157573A0 (en) 2004-03-28
ZA200306639B (en) 2004-08-26
YU67103A (sh) 2006-05-25
EA200300761A1 (ru) 2004-02-26
MA26267A1 (fr) 2004-09-01
IL157573A (en) 2009-09-22
HUP0303323A2 (hu) 2004-01-28
BG66333B1 (bg) 2013-06-28
UA75110C2 (en) 2006-03-15
KR20030081465A (ko) 2003-10-17
DE60203998T2 (de) 2005-09-22
EE200300402A (et) 2003-12-15
EP1363928A1 (en) 2003-11-26
DE10109657A1 (de) 2002-09-05
BRPI0207566B8 (pt) 2021-05-25
BRPI0207566B1 (pt) 2019-04-24

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