MXPA01008911A - Benzoil-indoles n-sustituidos utiles como agentes estrogenicos.. - Google Patents

Benzoil-indoles n-sustituidos utiles como agentes estrogenicos..

Info

Publication number
MXPA01008911A
MXPA01008911A MXPA01008911A MXPA01008911A MXPA01008911A MX PA01008911 A MXPA01008911 A MX PA01008911A MX PA01008911 A MXPA01008911 A MX PA01008911A MX PA01008911 A MXPA01008911 A MX PA01008911A MX PA01008911 A MXPA01008911 A MX PA01008911A
Authority
MX
Mexico
Prior art keywords
formula
compound
alkyl
pharmaceutically acceptable
compound according
Prior art date
Application number
MXPA01008911A
Other languages
English (en)
Spanish (es)
Inventor
Marci Catherine Koko
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of MXPA01008911A publication Critical patent/MXPA01008911A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
MXPA01008911A 1999-03-04 2000-02-22 Benzoil-indoles n-sustituidos utiles como agentes estrogenicos.. MXPA01008911A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26241399A 1999-03-04 1999-03-04
PCT/US2000/004386 WO2000051983A1 (fr) 1999-03-04 2000-02-22 Indols benzoyles n-substitues comme agents oestrogenes

Publications (1)

Publication Number Publication Date
MXPA01008911A true MXPA01008911A (es) 2002-10-23

Family

ID=22997395

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA01008911A MXPA01008911A (es) 1999-03-04 2000-02-22 Benzoil-indoles n-sustituidos utiles como agentes estrogenicos..

Country Status (8)

Country Link
EP (1) EP1159268A1 (fr)
JP (1) JP2002538141A (fr)
CN (1) CN1342144A (fr)
AR (1) AR022797A1 (fr)
AU (1) AU3859400A (fr)
CA (1) CA2364914A1 (fr)
MX (1) MXPA01008911A (fr)
WO (1) WO2000051983A1 (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5998402A (en) 1996-04-19 1999-12-07 American Home Products Corporation 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
US7632955B2 (en) 2001-12-13 2009-12-15 National Health Research Institutes Indole compounds
TWI317634B (en) 2001-12-13 2009-12-01 Nat Health Research Institutes Aroyl indoles compounds
US7528165B2 (en) 2001-12-13 2009-05-05 National Health Research Institutes Indole compounds
AU2003263402A1 (en) 2002-09-20 2004-04-08 Pfizer Products Inc. Amide and sulfonamide ligands for the estrogen receptor
CN100506795C (zh) * 2003-06-18 2009-07-01 中国科学院上海药物研究所 茚酮并吲哚类化合物、制备方法及它的医学用途
US7250440B2 (en) * 2003-08-12 2007-07-31 Wyeth (Hydroxyphenyl)-1H-indole-3-carbaldehyde oxime derivatives as estrogenic agents
US7456289B2 (en) 2004-12-31 2008-11-25 National Health Research Institutes Anti-tumor compounds
PL2276732T3 (pl) 2008-04-16 2015-11-30 Karobio Ab Nowe ligandy receptora estrogenowego

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1993023374A1 (fr) * 1992-05-08 1993-11-25 Otsuka Pharmaceutical Factory, Inc. Derive d'indole
EP0802183B1 (fr) * 1996-04-19 2001-10-10 American Home Products Corporation Composés oestrogènes

Also Published As

Publication number Publication date
CA2364914A1 (fr) 2000-09-08
WO2000051983A1 (fr) 2000-09-08
JP2002538141A (ja) 2002-11-12
AU3859400A (en) 2000-09-21
EP1159268A1 (fr) 2001-12-05
CN1342144A (zh) 2002-03-27
AR022797A1 (es) 2002-09-04

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