MX9703288A - Oxazolil- y tiazolilimidazo-benzo- y tienodiacepinas y su uso como medicamentos. - Google Patents

Oxazolil- y tiazolilimidazo-benzo- y tienodiacepinas y su uso como medicamentos.

Info

Publication number
MX9703288A
MX9703288A MX9703288A MX9703288A MX9703288A MX 9703288 A MX9703288 A MX 9703288A MX 9703288 A MX9703288 A MX 9703288A MX 9703288 A MX9703288 A MX 9703288A MX 9703288 A MX9703288 A MX 9703288A
Authority
MX
Mexico
Prior art keywords
thiazolylimidazo
thienodiazepines
oxazolyl
medicaments
benzo
Prior art date
Application number
MX9703288A
Other languages
English (en)
Other versions
MXPA97003288A (es
Inventor
Bernd Buttelmann
Thierry Godel
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MXPA97003288A publication Critical patent/MXPA97003288A/es
Publication of MX9703288A publication Critical patent/MX9703288A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La invencion se relaciona con imidazoidacepinas sustituidas básicamente de formula general (I). Esos compuestos pueden usarse como anxiolíticos y/o antoconvulsionantes y/o relajantes musculares y/o sustancias activas sedantes-hipnoticas.
MX9703288A 1994-11-11 1995-11-08 Oxazolil- y tiazolilimidazo-benzo- y tienodiacepinas y su uso como medicamentos. MX9703288A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
CH338694 1994-11-11
CH2261/95 1995-08-04
CH3386/94 1995-08-04
CH226195 1995-08-04
PCT/EP1995/004393 WO1996015129A1 (en) 1994-11-11 1995-11-08 Oxazolyl- and thiazolylimidazo-benzo- and thienodiazepines and their use as medicaments

Publications (2)

Publication Number Publication Date
MXPA97003288A MXPA97003288A (es) 1997-08-01
MX9703288A true MX9703288A (es) 1997-08-30

Family

ID=25689945

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9703288A MX9703288A (es) 1994-11-11 1995-11-08 Oxazolil- y tiazolilimidazo-benzo- y tienodiacepinas y su uso como medicamentos.

Country Status (12)

Country Link
US (2) US5885986A (es)
EP (1) EP0790999A1 (es)
JP (1) JP2989013B2 (es)
CN (1) CN1046519C (es)
AU (1) AU3982695A (es)
BR (1) BR9509711A (es)
FI (1) FI971990A0 (es)
IL (1) IL115882A (es)
MA (1) MA23716A1 (es)
MX (1) MX9703288A (es)
TW (1) TW349100B (es)
WO (1) WO1996015129A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2534639C (en) * 2003-07-31 2013-07-30 Immunomedics, Inc. Anti-cd19 antibodies
WO2009024325A2 (en) * 2007-08-20 2009-02-26 Evotec Neurosciences Gmbh Treatment of sleep disorders
US20090054412A1 (en) * 2007-08-20 2009-02-26 John Alan Kemp Treatment of Sleep Disorders
JP7013446B2 (ja) * 2016-08-16 2022-02-15 ユーダブリューエム・リサーチ・ファウンデーション，インコーポレーテッド Ｇａｂａ（ａ）受容体モジュレーター、及び、喘息における気道過敏及び炎症を抑制するための方法
CN111285878B (zh) * 2020-04-03 2022-05-13 杭州新博思生物医药有限公司 二氮杂卓类化合物及制法与其药用盐、前药和用途

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1143728A (en) * 1979-10-04 1983-03-29 Max Gerecke Imidazodiazepine derivatives
IL74070A (en) * 1984-01-19 1988-12-30 Hoffmann La Roche Imidazodiazepine derivatives,their manufacture and pharmaceutical compositions containing them
AU587802B2 (en) * 1985-03-08 1989-08-31 Ferrosan A/S Novel oxadiazolyl imidazobenzodiazepine derivatives and methods of preparing such compounds
US4771051A (en) * 1985-05-17 1988-09-13 A/S Ferrosan 3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments
TW201311B (es) * 1991-06-17 1993-03-01 Hoffmann La Roche
CA2143246C (en) * 1994-03-16 2000-08-22 Thierry Godel Imidazodiazepines

Also Published As

Publication number Publication date
IL115882A (en) 1998-10-30
WO1996015129A1 (en) 1996-05-23
CN1167487A (zh) 1997-12-10
IL115882A0 (en) 1996-01-31
BR9509711A (pt) 1997-09-30
EP0790999A1 (en) 1997-08-27
US5885986A (en) 1999-03-23
JP2989013B2 (ja) 1999-12-13
AU3982695A (en) 1996-06-06
TW349100B (en) 1999-01-01
FI971990A (fi) 1997-05-09
FI971990A0 (fi) 1997-05-09
CN1046519C (zh) 1999-11-17
US5962450A (en) 1999-10-05
JPH10505098A (ja) 1998-05-19
MA23716A1 (fr) 1996-07-01

Similar Documents

Publication Publication Date Title
GR3036867T3 (en) Hydroxymethylimidazodiazepines and their esters
ZA981936B (en) Novel benzimidazole inhibitors of fructose 1,6-bisphosphatase.
ATE182892T1 (de) Mercaptoacetylamide von pyridazo(1,2-a>(1,2>- diazepin -derivaten als eukephalinase und ace- inhibitoren
GB9514473D0 (en) Chemical compounds
IL119462A0 (en) Pyrrolopyrimidines
TR200000151T2 (tr) Yeni bileşimler.
TR200000197T2 (tr) Yeni bileşimler
MX9700557A (es) Dihidrobenzofuranos.
IT1285770B1 (it) Composti corticoidei
ES2157992T3 (es) Alcoxi-alquil-carbamatos de imidazo(1,2-a)piridinas.
IL129337A0 (en) Bicyclic aryl carboxamides and their therapeutic use
GB2380939B (en) Treatment or prevention of auto-immune diseases
HU9601646D0 (en) 4-benzoylisoxazoles and their use as herbicides
IS4367A (is) CCK eða gastrín temprandi 5-heterósýklísk-1,5-bensódíazepín
MX9703288A (es) Oxazolil- y tiazolilimidazo-benzo- y tienodiacepinas y su uso como medicamentos.
DE3688807D1 (de) Isolierung von castanospermin und dessen verwendung als antidiabetisches heilmittel.
UA22175A (uk) Протиаритмічний та протисудорожний засіб
IT1276751B1 (it) Composti ad attivita' antitumorale
ES2151820A1 (es) Herbicidas a base de derivados de 1,3-oxazin-4-ona, composiciones que los contienen y procedimiento para su preparacion.
MX9706424A (es) Uso de la moxonidina para el tratamiento de la aterosclerosis.

Legal Events

Date Code Title Description
FA Abandonment or withdrawal