MX9601953A - Nuevo compesto derivados de 5h-tiazolo [3,2-a] pirimidin-5-ona. - Google Patents

Nuevo compesto derivados de 5h-tiazolo [3,2-a] pirimidin-5-ona.

Info

Publication number
MX9601953A
MX9601953A MX9601953A MX9601953A MX9601953A MX 9601953 A MX9601953 A MX 9601953A MX 9601953 A MX9601953 A MX 9601953A MX 9601953 A MX9601953 A MX 9601953A MX 9601953 A MX9601953 A MX 9601953A
Authority
MX
Mexico
Prior art keywords
tiazol
pyrimidin
new compounds
compounds derived
carbon atoms
Prior art date
Application number
MX9601953A
Other languages
English (en)
Other versions
MXPA96001953A (es
Inventor
Rafael Foguet
Lluis Anglada
Aureli Sacristan
Josep M Castello
Jose A Ortiz
Original Assignee
Ferrer Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrer Int filed Critical Ferrer Int
Publication of MXPA96001953A publication Critical patent/MXPA96001953A/es
Publication of MX9601953A publication Critical patent/MX9601953A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Abstract

La presente invencion se refiere a nuevos compuestos derivados de 5H-tiazolo[3,2-a]pirimidin-5-ona, de formula general (I): donde Ar es un resto fenil opcionalmente sustituído por uno o dos grupos elegidos entre halogeno, alquil cuyo numero de átomos de carbono está comprendido entre 1 y 4, metilendioxi, alcoxi cuyo numero de átomos de carbono está comprendido entre 1 y 4, y trifluorometil; y R es un resto elegido entre (a) o (b): así como sus sales de adicion farmacéuticamente aceptables. La presente invencion también describe procedimientos e intermedios para su obtencion y composiciones farmacéuticas que los contienen.
MX9601953A 1995-05-26 1996-05-23 Nuevo compesto derivados de 5h-tiazolo [3,2-a] pirimidin-5-ona. MX9601953A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES09501029A ES2097093B1 (es) 1995-05-26 1995-05-26 Nuevos compuestos derivados de 5h-tiazolo (3,2-a) pirimidin-5-ona.
ES9501029 1995-05-26
ESES9501029 1995-05-26

Publications (2)

Publication Number Publication Date
MXPA96001953A MXPA96001953A (es) 1997-08-01
MX9601953A true MX9601953A (es) 1997-08-30

Family

ID=8290506

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9601953A MX9601953A (es) 1995-05-26 1996-05-23 Nuevo compesto derivados de 5h-tiazolo [3,2-a] pirimidin-5-ona.

Country Status (17)

Country Link
US (1) US5798361A (es)
EP (1) EP0773947B1 (es)
JP (1) JPH10503782A (es)
AT (1) ATE196633T1 (es)
AU (1) AU698455B2 (es)
CA (1) CA2195578A1 (es)
DE (1) DE69610477T2 (es)
DK (1) DK0773947T3 (es)
ES (1) ES2097093B1 (es)
IL (1) IL118280A (es)
MX (1) MX9601953A (es)
NO (1) NO308304B1 (es)
NZ (1) NZ308533A (es)
PT (1) PT773947E (es)
TW (1) TW430666B (es)
WO (1) WO1996037498A1 (es)
ZA (1) ZA964091B (es)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4443451A (en) * 1981-07-15 1984-04-17 Janssen Pharmaceutica N.V. Bicyclic pyrimidin-5-one derivatives
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
NZ254113A (en) * 1992-07-13 1995-08-28 Janssen Pharmaceutica Nv Fused piperidine derivatives and medicaments

Also Published As

Publication number Publication date
ES2097093A1 (es) 1997-03-16
WO1996037498A1 (en) 1996-11-28
IL118280A0 (en) 1996-09-12
ZA964091B (en) 1997-01-21
TW430666B (en) 2001-04-21
EP0773947A1 (en) 1997-05-21
ATE196633T1 (de) 2000-10-15
PT773947E (pt) 2001-01-31
IL118280A (en) 1999-10-28
AU5820396A (en) 1996-12-11
NO970327D0 (no) 1997-01-24
EP0773947B1 (en) 2000-09-27
CA2195578A1 (en) 1996-11-28
NO308304B1 (no) 2000-08-28
DE69610477T2 (de) 2001-05-10
DE69610477D1 (de) 2000-11-02
NO970327L (no) 1997-01-24
NZ308533A (en) 1997-11-24
US5798361A (en) 1998-08-25
AU698455B2 (en) 1998-10-29
JPH10503782A (ja) 1998-04-07
DK0773947T3 (da) 2000-10-16
ES2097093B1 (es) 1998-01-16

Similar Documents

Publication Publication Date Title
JO1351B1 (en) Chemical compounds
AU3461697A (en) Heterocyclic compounds, their production and use
EP0999834A4 (en) ANTITHROMOSIS
MXPA02004448A (es) Derivados de imidazopiridina como inhibidores de la fosfodiesterasa vii.
AU2267495A (en) Benzamide derivatives as vasopressin antagonists
BE2014C034I2 (en) Derivatives of 3-(2-oxo- 1,3']bipyrrolidinyl-3-ylidenemethyl)-cephems
NZ503912A (en) Piperidinylaminomethyl trifluoromethyl cyclic ether compounds and their use as substance P antagonists
PL309874A1 (en) Novel derivatives of pyrrolocarbasol, method of obtaining them and pharmaceutical composition containing such derivatives
AU1507888A (en) New bicyclic compounds, processes for preparation thereof and pharmaceutical composition comprising the same
HRP20000027B1 (en) Process for the preparation of alkoxyfuranoneamine derivatives, compounds obtained by this process, and the use of these compounds
MX9601953A (es) Nuevo compesto derivados de 5h-tiazolo [3,2-a] pirimidin-5-ona.
IE901104L (en) New bronchospasmolytic compounds and process for their¹preparation
MXPA04002838A (es) Derivados de alquilaminopiridazinona sustituidos, procedimiento para la preparacion de los mismos y composiciones farmaceuticas que los contienen.
IE781467L (en) 4"-ureido-oleandomycin derivatives
ES8707951A1 (es) Derivados de tetrazol
ES8801656A1 (es) Un procedimiento para la preparacion de un compuesto de quinazolinona.

Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees