MX9304970A - ACIDOS ß-AMINOALQUIL- Y ß-N-PEPTIDILAMINOALQUIL-BORONICOS. - Google Patents

ACIDOS ß-AMINOALQUIL- Y ß-N-PEPTIDILAMINOALQUIL-BORONICOS.

Info

Publication number
MX9304970A
MX9304970A MX9304970A MX9304970A MX9304970A MX 9304970 A MX9304970 A MX 9304970A MX 9304970 A MX9304970 A MX 9304970A MX 9304970 A MX9304970 A MX 9304970A MX 9304970 A MX9304970 A MX 9304970A
Authority
MX
Mexico
Prior art keywords
peptidylaminoalkyl
aminoalkyl
boronic acids
alkyl
aryl
Prior art date
Application number
MX9304970A
Other languages
English (en)
Inventor
David William Bjorkquist
Rajan Keshav Panandiker
Original Assignee
Procter & Gamble
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Procter & Gamble filed Critical Procter & Gamble
Publication of MX9304970A publication Critical patent/MX9304970A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C11—ANIMAL OR VEGETABLE OILS, FATS, FATTY SUBSTANCES OR WAXES; FATTY ACIDS THEREFROM; DETERGENTS; CANDLES
    • C11D—DETERGENT COMPOSITIONS; USE OF SINGLE SUBSTANCES AS DETERGENTS; SOAP OR SOAP-MAKING; RESIN SOAPS; RECOVERY OF GLYCEROL
    • C11D3/00—Other compounding ingredients of detergent compositions covered in group C11D1/00
    • C11D3/16—Organic compounds
    • C11D3/38—Products with no well-defined composition, e.g. natural products
    • C11D3/386—Preparations containing enzymes, e.g. protease or amylase
    • C11D3/38663—Stabilised liquid enzyme compositions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Wood Science & Technology (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Detergent Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Un compuesto que tiene la fórmula: en donde R1, R2 y R3 son independientemente hidrógeno o alquilo de 1 a 4 átomos de carbono; n es de 2 a 4; X es arilo, arilo sustituido o alquilo de 1 a 6 átomos de carbono; Y se selecciona del grupo que consiste de hidrógeno, aminoácido, dipéptido o tripéptido enlazado por medio de un ácido carboxílico C-terminal, y está presente el grupo protector de amina.
MX9304970A 1992-08-14 1993-08-16 ACIDOS ß-AMINOALQUIL- Y ß-N-PEPTIDILAMINOALQUIL-BORONICOS. MX9304970A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/931,809 US5442100A (en) 1992-08-14 1992-08-14 β-aminoalkyl and β-N-peptidylaminoalkyl boronic acids

Publications (1)

Publication Number Publication Date
MX9304970A true MX9304970A (es) 1994-05-31

Family

ID=25461390

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9304970A MX9304970A (es) 1992-08-14 1993-08-16 ACIDOS ß-AMINOALQUIL- Y ß-N-PEPTIDILAMINOALQUIL-BORONICOS.

Country Status (10)

Country Link
US (2) US5442100A (es)
EP (1) EP0655067B1 (es)
JP (1) JPH08500113A (es)
CN (1) CN1047596C (es)
AT (1) ATE159945T1 (es)
AU (1) AU4799793A (es)
DE (1) DE69315079T2 (es)
MX (1) MX9304970A (es)
TW (1) TW251274B (es)
WO (1) WO1994004542A1 (es)

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US9241947B2 (en) 2013-01-04 2016-01-26 Rempex Pharmaceuticals, Inc. Boronic acid derivatives and therapeutic uses thereof
KR20150103269A (ko) 2013-01-04 2015-09-09 렘펙스 파머수티클스 인코퍼레이티드 보론산 유도체 및 그의 치료적 용도
EP2970830B1 (en) 2013-03-14 2017-12-13 Novozymes A/S Enzyme and inhibitor contained in water-soluble films
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Also Published As

Publication number Publication date
WO1994004542A1 (en) 1994-03-03
AU4799793A (en) 1994-03-15
CN1047596C (zh) 1999-12-22
TW251274B (es) 1995-07-11
EP0655067B1 (en) 1997-11-05
US5488157A (en) 1996-01-30
EP0655067A1 (en) 1995-05-31
ATE159945T1 (de) 1997-11-15
JPH08500113A (ja) 1996-01-09
CN1090850A (zh) 1994-08-17
US5442100A (en) 1995-08-15
DE69315079D1 (de) 1997-12-11
DE69315079T2 (de) 1998-06-04

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