MX3308E - Procedimiento para la preparacion de derivados de la tieno-piridina - Google Patents
Procedimiento para la preparacion de derivados de la tieno-piridinaInfo
- Publication number
- MX3308E MX3308E MX000231U MX23176U MX3308E MX 3308 E MX3308 E MX 3308E MX 000231 U MX000231 U MX 000231U MX 23176 U MX23176 U MX 23176U MX 3308 E MX3308 E MX 3308E
- Authority
- MX
- Mexico
- Prior art keywords
- formula
- derivatives
- preparation
- alcoholic
- radical
- Prior art date
Links
- 230000001476 alcoholic effect Effects 0.000 abstract 3
- 239000002253 acid Substances 0.000 abstract 1
- 150000007513 acids Chemical class 0.000 abstract 1
- 125000002252 acyl group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 239000012948 isocyanate Substances 0.000 abstract 1
- 150000002513 isocyanates Chemical class 0.000 abstract 1
- 150000003242 quaternary ammonium salts Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- DBDCNCCRPKTRSD-UHFFFAOYSA-N thieno[3,2-b]pyridine Chemical class C1=CC=C2SC=CC2=N1 DBDCNCCRPKTRSD-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7517007A FR2312247A1 (fr) | 1975-05-30 | 1975-05-30 | Derives de la thieno-pyridine, leur procede de preparation et leurs applications |
Publications (1)
Publication Number | Publication Date |
---|---|
MX3308E true MX3308E (es) | 1980-09-09 |
Family
ID=9155902
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX000231U MX3308E (es) | 1975-05-30 | 1976-05-13 | Procedimiento para la preparacion de derivados de la tieno-piridina |
Country Status (27)
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2376860A1 (fr) * | 1977-01-07 | 1978-08-04 | Parcor | Tetrahydro-4,5,6,7 thieno (2,3-c) et (3,2-c) pyridines, leur procede de preparation et leur application therapeutique |
FR2395271A1 (fr) * | 1977-06-21 | 1979-01-19 | Parcor | Procede de preparation de thieno (2,3-c) et thieno (3,2-c) pyridines |
FR2397417A1 (fr) * | 1977-07-12 | 1979-02-09 | Parcor | Procede de preparation de derives de la thienopyridine |
US4321266A (en) * | 1980-10-06 | 1982-03-23 | Sanofi | 5-o-Cyanobenzyl-4,5,6,7-tetrahydrothieno [3,2-C] pyridine |
FR2597102B1 (fr) * | 1986-04-14 | 1988-08-26 | Sanofi Sa | Derives de l'acide a-(hydroxy-7 tetrahydro-4,5,6,7 thieno (3,2-c) pyridyl-5) phenyl acetique, leur procede de preparation, leur application comme medicament et les compositions les renfermant |
US6090797A (en) * | 1998-09-02 | 2000-07-18 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno(2,3-C)pyridine derivatives |
WO2000014090A1 (en) * | 1998-09-02 | 2000-03-16 | Novo Nordisk A/S | 4,5,6,7-tetrahydro-thieno[2,3-c]pyridine derivatives |
AU2002217464B2 (en) | 2000-12-25 | 2004-12-16 | Daiichi Sankyo Company, Limited | Medicinal compositions containing aspirin |
US7838026B2 (en) | 2001-09-28 | 2010-11-23 | Mcneil-Ppc, Inc. | Burst-release polymer composition and dosage forms comprising the same |
US7122143B2 (en) * | 2001-09-28 | 2006-10-17 | Mcneil-Ppc, Inc. | Methods for manufacturing dosage forms |
US7323192B2 (en) * | 2001-09-28 | 2008-01-29 | Mcneil-Ppc, Inc. | Immediate release tablet |
US20040062804A1 (en) * | 2001-09-28 | 2004-04-01 | Der-Yang Lee | Modified release dosage forms |
US7064211B2 (en) * | 2002-03-22 | 2006-06-20 | Eisai Co., Ltd. | Hemiasterlin derivatives and uses thereof |
TWI350168B (en) * | 2004-05-07 | 2011-10-11 | Incyte Corp | Amido compounds and their use as pharmaceuticals |
NZ551603A (en) * | 2004-06-24 | 2010-11-26 | Incyte Corp | N-substituted piperidines and their use as pharmaceuticals |
JP2008504279A (ja) * | 2004-06-24 | 2008-02-14 | インサイト・コーポレイション | アミド化合物およびその医薬としての使用 |
WO2006002349A1 (en) * | 2004-06-24 | 2006-01-05 | Incyte Corporation | Amido compounds and their use as pharmaceuticals |
EP1768954A4 (en) * | 2004-06-24 | 2008-05-28 | Incyte Corp | 2-METHYLPROPANAMIDES AND THEIR USE AS PHARMACEUTICALS |
EP1778229A4 (en) * | 2004-08-10 | 2009-06-17 | Incyte Corp | AMID COMPOUNDS AND THEIR USE AS MEDICAMENTS |
JP2008520700A (ja) * | 2004-11-18 | 2008-06-19 | インサイト・コーポレイション | 11−βヒドロキシルステロイドデヒドロゲナーゼタイプIの阻害剤およびその使用方法 |
US8673352B2 (en) * | 2005-04-15 | 2014-03-18 | Mcneil-Ppc, Inc. | Modified release dosage form |
CA2621255A1 (en) * | 2005-09-21 | 2007-04-05 | Incyte Corporation | Amido compounds and their use as pharmaceuticals |
AU2006322060A1 (en) * | 2005-12-05 | 2007-06-14 | Incyte Corporation | Lactam compounds and methods of using the same |
WO2007084314A2 (en) * | 2006-01-12 | 2007-07-26 | Incyte Corporation | MODULATORS OF 11-ß HYDROXYL STEROID DEHYDROGENASE TYPE 1, PHARMACEUTICAL COMPOSITIONS THEREOF, AND METHODS OF USING THE SAME |
US20070197530A1 (en) * | 2006-01-31 | 2007-08-23 | Yun-Long Li | Amido compounds and their use as pharmaceuticals |
TW200808807A (en) * | 2006-03-02 | 2008-02-16 | Incyte Corp | Modulators of 11-β hydroxyl steroid dehydrogenase type 1, pharmaceutical compositions thereof, and methods of using the same |
US20070208001A1 (en) * | 2006-03-03 | 2007-09-06 | Jincong Zhuo | Modulators of 11- beta hydroxyl steroid dehydrogenase type 1, pharmaceutical compositions thereof, and methods of using the same |
WO2007130898A1 (en) * | 2006-05-01 | 2007-11-15 | Incyte Corporation | TETRASUBSTITUTED UREAS AS MODULATORS OF 11-β HYDROXYL STEROID DEHYDROGENASE TYPE 1 |
EP2018378A2 (en) * | 2006-05-17 | 2009-01-28 | Incyte Corporation | Heterocyclic inhibitors of 11-b hydroxyl steroid dehydrogenase type i and methods of using the same |
JP5206669B2 (ja) * | 2007-03-30 | 2013-06-12 | 日本新薬株式会社 | ヘテロアリール誘導体 |
CN102241690B (zh) | 2010-05-13 | 2015-08-12 | 天津药物研究院 | 一类含腈基的噻吩并吡啶酯类衍生物、其制备方法和用途 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2215948B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) * | 1973-02-01 | 1976-05-14 | Centre Etd Ind Pharma | |
AR205040A1 (es) * | 1974-07-16 | 1976-03-31 | Parcor | Procedimiento de preparacion de derivados de la tetrahidro-4,5,6,7,-tieno(3,2-c)o(2,3-c)piridina |
-
1975
- 1975-05-30 FR FR7517007A patent/FR2312247A1/fr active Granted
-
1976
- 1976-03-19 CH CH345676A patent/CH613969A5/xx not_active IP Right Cessation
- 1976-03-22 LU LU74617A patent/LU74617A1/xx unknown
- 1976-03-23 GR GR50384A patent/GR59797B/el unknown
- 1976-04-05 YU YU856/76A patent/YU39479B/xx unknown
- 1976-04-12 IE IE763/76A patent/IE43224B1/en unknown
- 1976-04-13 IL IL49405A patent/IL49405A/xx unknown
- 1976-04-14 US US05/676,796 patent/US4076819A/en not_active Expired - Lifetime
- 1976-04-14 CA CA250,739A patent/CA1071633A/en not_active Expired
- 1976-04-14 ZA ZA762263A patent/ZA762263B/xx unknown
- 1976-05-04 ES ES447570A patent/ES447570A1/es not_active Expired
- 1976-05-05 AR AR263208A patent/AR211339A1/es active
- 1976-05-07 NL NL7604944A patent/NL7604944A/xx not_active Application Discontinuation
- 1976-05-13 MX MX000231U patent/MX3308E/es unknown
- 1976-05-17 SU SU762356004A patent/SU667138A3/ru active
- 1976-05-22 RO RO7686177A patent/RO68891A/ro unknown
- 1976-05-26 AT AT386576A patent/AT349471B/de not_active IP Right Cessation
- 1976-05-26 DE DE2623567A patent/DE2623567C2/de not_active Expired
- 1976-05-28 HU HU76PA00001248A patent/HU172176B/hu not_active IP Right Cessation
- 1976-05-28 AU AU14417/76A patent/AU498517B2/en not_active Expired
- 1976-05-28 SE SE7606062A patent/SE421623B/xx not_active IP Right Cessation
- 1976-05-28 GB GB22400/76A patent/GB1501797A/en not_active Expired
- 1976-05-28 DD DD193073A patent/DD125214A5/xx unknown
- 1976-05-28 DK DK235876A patent/DK235876A/da unknown
- 1976-05-28 BE BE167404A patent/BE842310A/xx not_active IP Right Cessation
- 1976-05-29 JP JP51062884A patent/JPS51149297A/ja active Pending
- 1976-05-29 PL PL1976189958A patent/PL100792B1/xx unknown
Also Published As
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