MX2010008518A - Ciertas entidades quimicas, composiciones y metodos. - Google Patents

Ciertas entidades quimicas, composiciones y metodos.

Info

Publication number
MX2010008518A
MX2010008518A MX2010008518A MX2010008518A MX2010008518A MX 2010008518 A MX2010008518 A MX 2010008518A MX 2010008518 A MX2010008518 A MX 2010008518A MX 2010008518 A MX2010008518 A MX 2010008518A MX 2010008518 A MX2010008518 A MX 2010008518A
Authority
MX
Mexico
Prior art keywords
skeletal
methods
muscle
chemical entities
certain chemical
Prior art date
Application number
MX2010008518A
Other languages
English (en)
Spanish (es)
Inventor
Gustave Bergnes
Luke W Ashcraft
Jianchao Wang
Bradley P Morgan
Alex Muci
Zhe Yang
Scott Collibee
Jeff Gardina
Brian Stoltz
Original Assignee
Cytokinetics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cytokinetics Inc filed Critical Cytokinetics Inc
Publication of MX2010008518A publication Critical patent/MX2010008518A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
MX2010008518A 2008-02-04 2009-02-02 Ciertas entidades quimicas, composiciones y metodos. MX2010008518A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2606708P 2008-02-04 2008-02-04
PCT/US2009/000686 WO2009099594A1 (en) 2008-02-04 2009-02-02 Certain chemical entities, compositions and methods

Publications (1)

Publication Number Publication Date
MX2010008518A true MX2010008518A (es) 2010-11-10

Family

ID=40952391

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010008518A MX2010008518A (es) 2008-02-04 2009-02-02 Ciertas entidades quimicas, composiciones y metodos.

Country Status (18)

Country Link
US (2) US7989469B2 (OSRAM)
EP (1) EP2244711A4 (OSRAM)
JP (1) JP2011510985A (OSRAM)
KR (1) KR20100119773A (OSRAM)
CN (1) CN101983061A (OSRAM)
AR (1) AR072242A1 (OSRAM)
AU (1) AU2009210787A1 (OSRAM)
BR (1) BRPI0907502A2 (OSRAM)
CA (1) CA2713864A1 (OSRAM)
CL (1) CL2009000246A1 (OSRAM)
CO (1) CO6290673A2 (OSRAM)
EA (1) EA201001224A1 (OSRAM)
EC (2) ECSP10010430A (OSRAM)
IL (1) IL207367A0 (OSRAM)
MX (1) MX2010008518A (OSRAM)
TW (1) TW200946524A (OSRAM)
WO (1) WO2009099594A1 (OSRAM)
ZA (1) ZA201005780B (OSRAM)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8299248B2 (en) 2006-08-02 2012-10-30 Cytokinetics, Incorporated Certain 1H-imidazo[4,5-b]pyrazin-2(3H)-ones and 1H-imidazo[4,5-b]pyrazin-2-ols and methods for their use
EA201001224A1 (ru) * 2008-02-04 2011-08-30 Цитокинетикс, Инкорпорейтед Химические соединения, композиции и способы их использования
CN102127070A (zh) * 2010-01-15 2011-07-20 山东轩竹医药科技有限公司 吡啶并环衍生物
ES2547687T3 (es) * 2011-07-09 2015-10-08 Xuanzhu Pharma Co., Ltd. Forma cristalina I de sal de un inhibidor de dipeptidil-peptidasa IV y procedimiento de preparación y uso de la misma
KR101951220B1 (ko) 2011-07-13 2019-02-22 싸이토키네틱스, 인코포레이티드 조합 als 치료법
JP6352244B2 (ja) * 2012-04-11 2018-07-04 サイトキネティックス, インコーポレイテッド 骨格筋疲労に対する耐性を向上させるための方法
RS63018B1 (sr) 2014-04-29 2022-04-29 Cytokinetics Inc Metode za smanjenje opadanja vitalnog kapaciteta
TW201927738A (zh) * 2017-12-14 2019-07-16 丹麥商Nmd藥品公司 用於治療神經肌肉病症的化合物
TWI794369B (zh) * 2017-12-14 2023-03-01 丹麥商Nmd藥品公司 用於治療神經肌肉病症的化合物
AU2020284742A1 (en) * 2019-05-28 2022-02-03 Mankind Pharma Ltd. Novel compounds for inhibition of Janus Kinase 1
EP4333982A1 (en) * 2021-05-06 2024-03-13 Exscientia Al Limited Pkc-theta modulators
CN118702622A (zh) * 2024-08-30 2024-09-27 阜新达得利化工股份有限公司 一种3-溴-2-氰基吡啶的制备方法

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0206860D0 (en) * 2002-03-22 2002-05-01 Glaxo Group Ltd Compounds
GB0212048D0 (en) * 2002-05-24 2002-07-03 Merck Sharp & Dohme Therapeutic agents
WO2004043913A2 (en) 2002-11-08 2004-05-27 Trimeris, Inc. Hetero-substituted benzimidazole compounds and antiviral uses thereof
AU2004253543B2 (en) 2003-07-01 2009-02-19 Merck & Co., Inc. Ophthalmic compositions for treating ocular hypertension
CA2550091A1 (en) 2003-12-19 2005-07-07 Elixir Pharmaceuticals, Inc. Methods of treating a disorder
WO2005072412A2 (en) 2004-01-29 2005-08-11 Elixir Pharmaceuticals, Inc. Anti-viral therapeutics
WO2005108374A1 (en) 2004-04-29 2005-11-17 Fmc Corporation Insecticidal diazole and triazole derivatives
GB0420719D0 (en) 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
WO2007078815A2 (en) * 2005-12-16 2007-07-12 Cytokinetics, Inc. Certain chemical entities, compositions, and methods
US8227603B2 (en) 2006-08-01 2012-07-24 Cytokinetics, Inc. Modulating skeletal muscle
EA017925B1 (ru) 2006-08-02 2013-04-30 Цитокинетикс, Инкорпорэйтед ПРОИЗВОДНЫЕ 1Н-ИМИДАЗО[4,5-b]ПИРАЗИНА
KR101504669B1 (ko) 2006-10-19 2015-03-20 시그날 파마소티칼 엘엘씨 헤테로아릴 화합물, 이들의 조성물 그리고 단백질 키나아제 억제제로서의 이들의 용도
CL2007002994A1 (es) 2006-10-19 2008-02-08 Wyeth Corp Compuestos derivados heterociclicos que contienen sulfamoilo, inhibidores de hsp90; composicion farmaceutica; y uso para el tratamiento del cancer, tal como cancer de mama, de colon y prostata, entre otros.
WO2008075007A1 (en) * 2006-12-21 2008-06-26 Cancer Research Technology Limited Morpholino-substituted bicycloheteroaryl compounds and their use as anti cancer agents
WO2008121333A1 (en) * 2007-03-30 2008-10-09 Cytokinetics, Incorporated Certain chemical entities, compositions and methods
US7998976B2 (en) 2008-02-04 2011-08-16 Cytokinetics, Inc. Certain chemical entities, compositions and methods
EA201001224A1 (ru) * 2008-02-04 2011-08-30 Цитокинетикс, Инкорпорейтед Химические соединения, композиции и способы их использования
AU2009324894B2 (en) 2008-11-25 2015-04-09 University Of Rochester MLK inhibitors and methods of use

Also Published As

Publication number Publication date
US7989469B2 (en) 2011-08-02
EP2244711A1 (en) 2010-11-03
EA201001224A1 (ru) 2011-08-30
CL2009000246A1 (es) 2009-06-26
CA2713864A1 (en) 2009-08-13
ECSP10010432A (es) 2011-01-31
CO6290673A2 (es) 2011-06-20
AR072242A1 (es) 2010-08-18
US20110312975A1 (en) 2011-12-22
US20090253737A1 (en) 2009-10-08
ECSP10010430A (es) 2011-02-28
JP2011510985A (ja) 2011-04-07
TW200946524A (en) 2009-11-16
KR20100119773A (ko) 2010-11-10
ZA201005780B (en) 2011-04-28
CN101983061A (zh) 2011-03-02
BRPI0907502A2 (pt) 2019-01-15
WO2009099594A1 (en) 2009-08-13
EP2244711A4 (en) 2011-08-24
IL207367A0 (en) 2010-12-30
AU2009210787A1 (en) 2009-08-13

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