MX2010006926A - 4-imidazolidinonas como inhibidores del canal de potasio kv1.5. - Google Patents

4-imidazolidinonas como inhibidores del canal de potasio kv1.5.

Info

Publication number
MX2010006926A
MX2010006926A MX2010006926A MX2010006926A MX2010006926A MX 2010006926 A MX2010006926 A MX 2010006926A MX 2010006926 A MX2010006926 A MX 2010006926A MX 2010006926 A MX2010006926 A MX 2010006926A MX 2010006926 A MX2010006926 A MX 2010006926A
Authority
MX
Mexico
Prior art keywords
imidazolidinones
potassium channel
channel inhibitors
present teachings
selective
Prior art date
Application number
MX2010006926A
Other languages
English (en)
Spanish (es)
Inventor
Shengde Wu
Benjamin E Blass
John M Janusz
James M Ii Ridgeway
Original Assignee
Wyeth Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Llc filed Critical Wyeth Llc
Publication of MX2010006926A publication Critical patent/MX2010006926A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MX2010006926A 2007-12-19 2008-12-18 4-imidazolidinonas como inhibidores del canal de potasio kv1.5. MX2010006926A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1493707P 2007-12-19 2007-12-19
PCT/US2008/087459 WO2009079630A1 (fr) 2007-12-19 2008-12-18 4-imidazolidinones comme inhibiteurs du canal potassique kv1.5

Publications (1)

Publication Number Publication Date
MX2010006926A true MX2010006926A (es) 2010-08-02

Family

ID=40379648

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2010006926A MX2010006926A (es) 2007-12-19 2008-12-18 4-imidazolidinonas como inhibidores del canal de potasio kv1.5.

Country Status (8)

Country Link
EP (1) EP2234983A1 (fr)
JP (1) JP2011507887A (fr)
AU (1) AU2008338374A1 (fr)
BR (1) BRPI0821394A2 (fr)
CA (1) CA2709187A1 (fr)
MX (1) MX2010006926A (fr)
WO (1) WO2009079630A1 (fr)
ZA (1) ZA201005086B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO3175985T3 (fr) 2011-07-01 2018-04-28
JP2015504923A (ja) 2012-01-27 2015-02-16 ギリアード サイエンシーズ, インコーポレイテッド 後期ナトリウムイオンチャネル遮断剤およびカリウムイオンチャネル遮断剤を使用する併用療法
WO2014134419A1 (fr) 2013-03-01 2014-09-04 Gilead Sciences, Inc. Utilisation de bloqueurs ikach pour le traitement de maladies cardiaques

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY125533A (en) * 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
PE20080207A1 (es) * 2006-06-20 2008-05-08 Wyeth Corp DERIVADOS DE 1-N-AMINO-2-IMIDAZOLIDINONAS COMO INHIBIDORES DEL CANAL DE POTASIO Kv1.5

Also Published As

Publication number Publication date
EP2234983A1 (fr) 2010-10-06
WO2009079630A1 (fr) 2009-06-25
ZA201005086B (en) 2011-03-30
AU2008338374A1 (en) 2009-06-25
BRPI0821394A2 (pt) 2015-06-16
CA2709187A1 (fr) 2009-06-25
JP2011507887A (ja) 2011-03-10

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Legal Events

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