MX2007015607A - Esteres de quinolin 3-sulfonato como moduladores del receptor de nk3. - Google Patents
Esteres de quinolin 3-sulfonato como moduladores del receptor de nk3.Info
- Publication number
- MX2007015607A MX2007015607A MX2007015607A MX2007015607A MX2007015607A MX 2007015607 A MX2007015607 A MX 2007015607A MX 2007015607 A MX2007015607 A MX 2007015607A MX 2007015607 A MX2007015607 A MX 2007015607A MX 2007015607 A MX2007015607 A MX 2007015607A
- Authority
- MX
- Mexico
- Prior art keywords
- phenyl
- independently selected
- alkyl
- halogen
- cycloalkyl
- Prior art date
Links
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- 102100029409 Neuromedin-K receptor Human genes 0.000 title claims description 12
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- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Hospice & Palliative Care (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Otolaryngology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Child & Adolescent Psychology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US69328105P | 2005-06-23 | 2005-06-23 | |
| PCT/SE2006/000758 WO2006137789A1 (en) | 2005-06-23 | 2006-06-21 | Quinoline 3 -sulfonate esters as NK3 receptor modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2007015607A true MX2007015607A (es) | 2008-02-25 |
Family
ID=37570727
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2007015607A MX2007015607A (es) | 2005-06-23 | 2006-06-21 | Esteres de quinolin 3-sulfonato como moduladores del receptor de nk3. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20080194622A1 (enExample) |
| EP (1) | EP1896418A1 (enExample) |
| JP (1) | JP2008546767A (enExample) |
| KR (1) | KR20080031871A (enExample) |
| CN (1) | CN101208304A (enExample) |
| AU (1) | AU2006259890A1 (enExample) |
| CA (1) | CA2613001A1 (enExample) |
| IL (1) | IL188034A0 (enExample) |
| MX (1) | MX2007015607A (enExample) |
| NO (1) | NO20080446L (enExample) |
| WO (1) | WO2006137789A1 (enExample) |
| ZA (1) | ZA200710723B (enExample) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR057130A1 (es) | 2005-09-21 | 2007-11-14 | Astrazeneca Ab | Quinolinas de alquilsulfoxido y una composicion farmaceutica |
| TW201018662A (en) | 2005-12-12 | 2010-05-16 | Astrazeneca Ab | Alkylsulphonamide quinolines |
| AR073891A1 (es) * | 2008-10-20 | 2010-12-09 | Lundbeck & Co As H | Derivados de isoquinolinona antagonistas de receptores nk3, composiciones farmaceuticas que los contienen y uso de los mismos en el tratamiento de psicosis, alzheimer y otras enfermedades. |
| PE20141360A1 (es) | 2011-02-07 | 2014-10-13 | Plexxikon Inc | Compuestos y metodos para la modulacion de quinasas e indicaciones para los mismos. |
| BR112015026519A2 (pt) | 2013-04-19 | 2017-07-25 | Astrazeneca Ab | composto antagonista do receptor nk3 (nk3ra) para uso em um método destinado ao tratamento de síndrome do ovário policístico (sop) |
| WO2017072629A1 (en) | 2015-10-29 | 2017-05-04 | Cadila Healthcare Limited | Pharmaceutical combination of nk3 receptor antagonist and biguanides |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69531458T2 (de) * | 1994-05-27 | 2004-08-05 | Glaxosmithkline S.P.A. | Chinolinderivate als tachykinin nk3 rezeptor antagonisten |
| AR004735A1 (es) * | 1995-11-24 | 1999-03-10 | Smithkline Beecham Spa | Quinoleina 4-amido sustituida, un procedimiento para su preparacion, una composicion farmaceutica que los contiene y el uso de los mismos para lapreparacion de un medicamento. |
| GB0027701D0 (en) * | 2000-11-13 | 2000-12-27 | Smithkline Beecham Spa | Novel compounds |
| EP1385839B1 (en) * | 2001-04-11 | 2006-02-22 | GlaxoSmithKline S.p.A. | 3-substituted quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists |
| GB0318727D0 (en) * | 2003-08-08 | 2003-09-10 | Smithkline Beecham Corp | Novel compounds |
-
2006
- 2006-06-21 WO PCT/SE2006/000758 patent/WO2006137789A1/en not_active Ceased
- 2006-06-21 AU AU2006259890A patent/AU2006259890A1/en not_active Abandoned
- 2006-06-21 JP JP2008518080A patent/JP2008546767A/ja not_active Abandoned
- 2006-06-21 CN CNA2006800228098A patent/CN101208304A/zh active Pending
- 2006-06-21 EP EP06747947A patent/EP1896418A1/en not_active Withdrawn
- 2006-06-21 CA CA002613001A patent/CA2613001A1/en not_active Abandoned
- 2006-06-21 US US11/917,820 patent/US20080194622A1/en not_active Abandoned
- 2006-06-21 KR KR1020077029959A patent/KR20080031871A/ko not_active Withdrawn
- 2006-06-21 MX MX2007015607A patent/MX2007015607A/es not_active Application Discontinuation
-
2007
- 2007-12-10 IL IL188034A patent/IL188034A0/en unknown
- 2007-12-10 ZA ZA200710723A patent/ZA200710723B/xx unknown
-
2008
- 2008-01-23 NO NO20080446A patent/NO20080446L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AU2006259890A1 (en) | 2006-12-28 |
| WO2006137789A8 (en) | 2008-01-17 |
| KR20080031871A (ko) | 2008-04-11 |
| CN101208304A (zh) | 2008-06-25 |
| US20080194622A1 (en) | 2008-08-14 |
| CA2613001A1 (en) | 2006-12-28 |
| IL188034A0 (en) | 2008-03-20 |
| JP2008546767A (ja) | 2008-12-25 |
| NO20080446L (no) | 2008-01-23 |
| ZA200710723B (en) | 2008-12-31 |
| WO2006137789A1 (en) | 2006-12-28 |
| EP1896418A1 (en) | 2008-03-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |