MD4258B1 - Utilizarea compusilor coordinativi ai cuprului(II) cu 4-(metoxifenil)tiosemicarbazonele 2-benzoilpiridinei în calitate de inhibitori ai Candida albicans - Google Patents
Utilizarea compusilor coordinativi ai cuprului(II) cu 4-(metoxifenil)tiosemicarbazonele 2-benzoilpiridinei în calitate de inhibitori ai Candida albicans Download PDFInfo
- Publication number
- MD4258B1 MD4258B1 MD20120045A MD20120045A MD4258B1 MD 4258 B1 MD4258 B1 MD 4258B1 MD 20120045 A MD20120045 A MD 20120045A MD 20120045 A MD20120045 A MD 20120045A MD 4258 B1 MD4258 B1 MD 4258B1
- Authority
- MD
- Moldova
- Prior art keywords
- inhibitors
- copper
- candida albicans
- benzoylpyridine
- thiosemicarbazones
- Prior art date
Links
- 241000222122 Candida albicans Species 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 239000003112 inhibitor Substances 0.000 title abstract 3
- JPVYNHNXODAKFH-UHFFFAOYSA-N Cu2+ Chemical compound [Cu+2] JPVYNHNXODAKFH-UHFFFAOYSA-N 0.000 title abstract 2
- 229940042396 direct acting antivirals thiosemicarbazones Drugs 0.000 title abstract 2
- GCSHUYKULREZSJ-UHFFFAOYSA-N phenyl(pyridin-2-yl)methanone Chemical compound C=1C=CC=NC=1C(=O)C1=CC=CC=C1 GCSHUYKULREZSJ-UHFFFAOYSA-N 0.000 title abstract 2
- 150000003584 thiosemicarbazones Chemical class 0.000 title abstract 2
- 229940095731 candida albicans Drugs 0.000 title 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 3
- RYGMFSIKBFXOCR-UHFFFAOYSA-N Copper Chemical compound [Cu] RYGMFSIKBFXOCR-UHFFFAOYSA-N 0.000 abstract 1
- 229910052802 copper Inorganic materials 0.000 abstract 1
- 239000010949 copper Substances 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 229910052723 transition metal Inorganic materials 0.000 abstract 1
- 150000003624 transition metals Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Inventia se refera la medicina, si anume la utilizarea compusilor coordinativi ai cuprului biologic activi din clasa tiosemicarbazonatilor metalelor de tranzitie în calitate de inhibitori ai fungilor din specia Candida albicans.Esenta inventiei consta în utilizarea în calitate de inhibitori ai fungilor din specia Candida albicans a compusilor coordinativi ai cuprului(II) cu 4-(metoxifenil)tiosemicarbazonele 2-benzoilpiridinei cu formula generala:I-IIII: R1 = OCH3, R2 = R3 = H; II: R1 = R3 = H, R2 = OCH3; III: R1 = R2 = H, R3 = OCH3.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20120045A MD4258C1 (ro) | 2012-05-31 | 2012-05-31 | Utilizarea compuşilor coordinativi ai cuprului(II) cu 4-(metoxifenil)tiosemicarbazonele 2-benzoilpiridinei în calitate de inhibitori ai Candida albicans |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| MDA20120045A MD4258C1 (ro) | 2012-05-31 | 2012-05-31 | Utilizarea compuşilor coordinativi ai cuprului(II) cu 4-(metoxifenil)tiosemicarbazonele 2-benzoilpiridinei în calitate de inhibitori ai Candida albicans |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| MD4258B1 true MD4258B1 (ro) | 2013-11-30 |
| MD4258C1 MD4258C1 (ro) | 2014-06-30 |
Family
ID=49724417
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MDA20120045A MD4258C1 (ro) | 2012-05-31 | 2012-05-31 | Utilizarea compuşilor coordinativi ai cuprului(II) cu 4-(metoxifenil)tiosemicarbazonele 2-benzoilpiridinei în calitate de inhibitori ai Candida albicans |
Country Status (1)
| Country | Link |
|---|---|
| MD (1) | MD4258C1 (ro) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4383C1 (ro) * | 2015-03-06 | 2016-06-30 | Государственный Университет Молд0 | Compusul acetato-(8-formilchinolintiosemicarbazono)cupru(II) care manifestă activitate antibacteriană |
| MD4402C1 (ro) * | 2015-09-04 | 2016-09-30 | Государственный Университет Молд0 | Metil-N'-[(2-hidroxinaftalen-1-il)metiliden]-N-prop-2-en-1-ilhidrazonotioat, care manifestă activitate antimicotică faţă de Candida albicans |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3824276A (en) * | 1963-03-14 | 1974-07-16 | Upjohn Co | Substituted-2-oxobutyraldehyde bis(thiosemicarbazones) |
| US6329378B1 (en) * | 1999-02-10 | 2001-12-11 | Anadys Pharmaceuticals, Inc. | Hydrazone, hydrazine and thiosemicarbazone derivatives as antifungal agents |
| MD1812C2 (ro) * | 2000-12-29 | 2002-06-30 | Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова | Complecşi de cupru ca inhibitori de bacterii şi fungi |
| MD2003C2 (ro) * | 2001-01-10 | 2003-03-31 | Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова | Complecşi interni de cupru (II) cu acţiune antimicrobiană şi antimicotică |
| WO2002085358A2 (en) * | 2001-04-20 | 2002-10-31 | Vion Pharmaceuticals, Inc. | Antiviral agents and methods of treating viral infections |
| MD2325G2 (ro) * | 2002-07-10 | 2004-06-30 | Государственный Медицинский И Фармацевтический Университет "Nicolae Testemitanu" Республики Молдова | Complecşi chelaţi ai cuprului(II) - inhibitori ai creşterii şi multiplicării fungilor levurici şi miceliari |
| MD2861G2 (ro) * | 2004-09-20 | 2006-04-30 | Государственный Университет Молд0 | (µ-Imidazol-N,N?)-bis{4-bromo-2-[2-(oxietilimino)-metil]-fenolato(2-)-cupru}, care manifestă activitate antimicotică |
| MD3484G2 (ro) * | 2007-02-12 | 2008-08-31 | Государственный Университет Молд0 | Di-{µ-[N-(2-hidroxietil)-(5-clorosalicilideniminato(-1))]-(O, N, O, Cl}-bis-(nitrato-imidazolcupru) care manifestă activitate antimicotică |
-
2012
- 2012-05-31 MD MDA20120045A patent/MD4258C1/ro not_active IP Right Cessation
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MD4383C1 (ro) * | 2015-03-06 | 2016-06-30 | Государственный Университет Молд0 | Compusul acetato-(8-formilchinolintiosemicarbazono)cupru(II) care manifestă activitate antibacteriană |
| MD4402C1 (ro) * | 2015-09-04 | 2016-09-30 | Государственный Университет Молд0 | Metil-N'-[(2-hidroxinaftalen-1-il)metiliden]-N-prop-2-en-1-ilhidrazonotioat, care manifestă activitate antimicotică faţă de Candida albicans |
Also Published As
| Publication number | Publication date |
|---|---|
| MD4258C1 (ro) | 2014-06-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG4A | Patent for invention issued | ||
| KA4A | Patent for invention lapsed due to non-payment of fees (with right of restoration) | ||
| MM4A | Patent for invention definitely lapsed due to non-payment of fees |