MC1253A1 - Derives amines de sucre utiles notamment comme medicaments - Google Patents

Derives amines de sucre utiles notamment comme medicaments

Info

Publication number
MC1253A1
MC1253A1 MC791365A MC1365A MC1253A1 MC 1253 A1 MC1253 A1 MC 1253A1 MC 791365 A MC791365 A MC 791365A MC 1365 A MC1365 A MC 1365A MC 1253 A1 MC1253 A1 MC 1253A1
Authority
MC
Monaco
Prior art keywords
medicaments
amine derivatives
derivatives useful
sugar amine
sugar
Prior art date
Application number
MC791365A
Other languages
English (en)
French (fr)
Inventor
K Watanabe
K Ogawa
Y Suhara
K Yokose
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MC1253A1 publication Critical patent/MC1253A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12N—MICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N9/00—Enzymes; Proenzymes; Compositions thereof; Processes for preparing, activating, inhibiting, separating or purifying enzymes
    • C12N9/99—Enzyme inactivation by chemical treatment
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P19/00—Preparation of compounds containing saccharide radicals
    • C12P19/26—Preparation of nitrogen-containing carbohydrates

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Microbiology (AREA)
  • General Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
MC791365A 1978-02-14 1979-02-13 Derives amines de sucre utiles notamment comme medicaments MC1253A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB583478 1978-02-14

Publications (1)

Publication Number Publication Date
MC1253A1 true MC1253A1 (fr) 1980-01-14

Family

ID=9803510

Family Applications (1)

Application Number Title Priority Date Filing Date
MC791365A MC1253A1 (fr) 1978-02-14 1979-02-13 Derives amines de sucre utiles notamment comme medicaments

Country Status (26)

Country Link
US (1) US4273765A (cs)
EP (1) EP0003616B1 (cs)
JP (1) JPS54163511A (cs)
AR (1) AR219150A1 (cs)
AT (1) AT367451B (cs)
AU (1) AU527318B2 (cs)
CA (1) CA1121290A (cs)
DE (2) DE2905649A1 (cs)
DK (1) DK149599C (cs)
ES (1) ES477653A1 (cs)
FI (1) FI63062C (cs)
FR (1) FR2416901A1 (cs)
GR (1) GR72817B (cs)
HU (1) HU181442B (cs)
IE (1) IE47916B1 (cs)
IL (1) IL56626A0 (cs)
LU (1) LU80906A1 (cs)
MC (1) MC1253A1 (cs)
NL (1) NL7901182A (cs)
NO (1) NO153011C (cs)
NZ (1) NZ189625A (cs)
PH (1) PH15084A (cs)
PT (1) PT69218A (cs)
SE (1) SE7901276L (cs)
YU (1) YU41437B (cs)
ZA (1) ZA79528B (cs)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0056194B1 (en) * 1981-01-05 1984-09-12 Takeda Chemical Industries, Ltd. N-substituted pseudo-aminosugars, their production and use
JPS57146713A (en) * 1981-03-09 1982-09-10 Akira Endo Hypoglycemic
US4595678A (en) * 1982-03-19 1986-06-17 Takeda Chemical Industries, Ltd. N-substituted pseudo-aminosugars and pharmaceutical compositions containing same
US4762857A (en) * 1986-05-30 1988-08-09 E. I. Du Pont De Nemours And Company Trehalose as stabilizer and tableting excipient
US4678812A (en) * 1986-05-30 1987-07-07 E. I. Du Pont De Nemours And Company Trehalose as stabilizer and tableting excipient
US4885361A (en) * 1987-07-31 1989-12-05 Hoffmann-La Roche Inc. Sulfated oligosaccharides
ATE132269T1 (de) * 1990-11-30 1996-01-15 Monoclonetics Int Verfahren zur diagnose chronischer niedriger rückenschmerzen und nackenschmerzen
TW381025B (en) * 1993-08-05 2000-02-01 Hoffmann La Roche Pharmaceutical composition containing a glucosidase inhibitor and a lipase inhibitor
IL143225A (en) * 2000-05-24 2008-03-20 Pfizer Preparation of drugs containing α-amylase inhibitors to treat hyperacidity of the inner abdomen
US7022684B2 (en) * 2000-05-24 2006-04-04 Pfizer Inc. Treatment of rumen acidosis with α-amylase inhibitors
EP2428516A1 (en) 2003-11-19 2012-03-14 Metabasis Therapeutics, Inc. Novel phosphorus-containing thyromimetics
US7262318B2 (en) * 2004-03-10 2007-08-28 Pfizer, Inc. Substituted heteroaryl- and phenylsulfamoyl compounds
US20050288340A1 (en) * 2004-06-29 2005-12-29 Pfizer Inc Substituted heteroaryl- and phenylsulfamoyl compounds
EP1819681B1 (en) * 2004-11-23 2009-08-12 Warner-Lambert Company LLC 7-(2h-pyrazol-3-yl)-3,5-dihydroxy-heptanoic acid derivatives as hmg co-a reductase inhibitors for the treatment of lipidemia
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7888376B2 (en) 2005-11-23 2011-02-15 Bristol-Myers Squibb Company Heterocyclic CETP inhibitors
US8404896B2 (en) 2006-12-01 2013-03-26 Bristol-Myers Squibb Company N-((3-benzyl)-2,2-(bis-phenyl)-propan-1-amine derivatives as CETP inhibitors for the treatment of atherosclerosis and cardiovascular diseases
AU2008261102B2 (en) 2007-06-04 2013-11-28 Bausch Health Ireland Limited Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
US8969514B2 (en) 2007-06-04 2015-03-03 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
US8034782B2 (en) 2008-07-16 2011-10-11 Synergy Pharmaceuticals, Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
BRPI0911063A2 (pt) * 2008-04-11 2016-11-01 Astellas Pharma Inc composto aminoaçúcar e processo para produção do mesmo
CA2930674A1 (en) 2008-06-04 2009-12-10 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase useful for the treatment of gastrointestinal disorders, inflammation, cancer and other disorders
WO2010093601A1 (en) 2009-02-10 2010-08-19 Metabasis Therapeutics, Inc. Novel sulfonic acid-containing thyromimetics, and methods for their use
US20130072519A1 (en) 2010-05-21 2013-03-21 Edward Lee Conn 2-phenyl benzoylamides
WO2012027331A1 (en) 2010-08-27 2012-03-01 Ironwood Pharmaceuticals, Inc. Compositions and methods for treating or preventing metabolic syndrome and related diseases and disorders
US9616097B2 (en) 2010-09-15 2017-04-11 Synergy Pharmaceuticals, Inc. Formulations of guanylate cyclase C agonists and methods of use
US20130345392A1 (en) 2011-03-04 2013-12-26 Pfizer Inc Edn3-like peptides and uses thereof
MY188344A (en) 2012-03-09 2021-12-01 Biotropics Malaysia Berhad Extract formulations of rhodamnia cinerea and uses thereof
EP2968439A2 (en) 2013-03-15 2016-01-20 Synergy Pharmaceuticals Inc. Compositions useful for the treatment of gastrointestinal disorders
AU2014235215A1 (en) 2013-03-15 2015-10-01 Synergy Pharmaceuticals Inc. Agonists of guanylate cyclase and their uses
RU2618628C1 (ru) 2013-04-17 2017-05-05 Пфайзер Инк. Производные N-пиперидин-3-илбензамида для лечения сердечно-сосудистых заболеваний
CN113388007A (zh) 2013-06-05 2021-09-14 博士医疗爱尔兰有限公司 鸟苷酸环化酶c的超纯激动剂、制备和使用所述激动剂的方法
DK3186242T3 (da) 2014-08-29 2021-12-20 Tes Pharma S R L Alfa-amino-beta-carboxymuconsyre-semialdehyd-decarboxylasehæmmere
WO2016055901A1 (en) 2014-10-08 2016-04-14 Pfizer Inc. Substituted amide compounds
EP3526199B1 (en) 2016-10-14 2022-04-13 Tes Pharma S.r.l. Inhibitors of alpha-amino-beta-carboxymuconic acid semialdehyde decarboxylase
EP3883930A1 (en) 2018-11-20 2021-09-29 Tes Pharma S.r.l. Inhibitors of alpha-amino-beta-carboxymuconic acid semialdehyde decarboxylase
PT3911648T (pt) 2019-01-18 2025-01-10 Astrazeneca Ab 6¿-[[(1s,3s)-3-[[5-(difluorometoxi)-2-pirimidinil]amino]ciclopentil]amino][1(2h),3¿-bipiridina]-2-ona como inibidor de pcsk9 e seus métodos de utilização

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2064092C2 (de) * 1970-12-28 1983-06-01 Bayer Ag, 5090 Leverkusen Inhibitoren für Glykosidhydrolasen aus Actinomyceten
US4062950A (en) * 1973-09-22 1977-12-13 Bayer Aktiengesellschaft Amino sugar derivatives
DE2347782C3 (de) * 1973-09-22 1979-10-11 Bayer Ag, 5090 Leverkusen Aminozuckerderivate, Verfahren zu ihrer Herstellung sowie diese Verbindungen enthaltende Arzneimittel
US4065557A (en) * 1974-03-21 1977-12-27 Bayer Aktiengesellschaft Amino sugars and their use in improving the meat:fat ratio in animals
USRE29903E (en) 1975-03-19 1979-02-06 American Cyanamid Company Antibacterial antibiotics AM31α, AM31β and AM31γ
DE2614393C3 (de) * 1976-04-02 1980-04-03 Bayer Ag, 5090 Leverkusen Aminozucker-Derivate und diese Verbindungen enthaltende Arzneimittel

Also Published As

Publication number Publication date
HU181442B (en) 1983-07-28
NO153011B (no) 1985-09-23
DK149599C (da) 1987-06-01
EP0003616A2 (de) 1979-08-22
YU34879A (en) 1983-01-21
PH15084A (en) 1982-07-02
FR2416901B1 (cs) 1980-10-24
NL7901182A (nl) 1979-08-16
DE2905649A1 (de) 1979-08-16
PT69218A (en) 1979-03-01
DE2962165D1 (en) 1982-03-25
EP0003616B1 (de) 1982-02-24
NO790469L (no) 1979-08-15
AT367451B (de) 1982-07-12
ZA79528B (en) 1980-02-27
YU41437B (en) 1987-06-30
AU527318B2 (en) 1983-02-24
NZ189625A (en) 1981-05-01
DK61179A (da) 1979-08-15
LU80906A1 (de) 1980-09-24
FR2416901A1 (fr) 1979-09-07
JPS643877B2 (cs) 1989-01-23
FI63062C (fi) 1983-04-11
GR72817B (cs) 1983-12-06
ES477653A1 (es) 1980-03-01
AR219150A1 (es) 1980-07-31
IE47916B1 (en) 1984-07-25
IL56626A0 (en) 1979-05-31
FI63062B (fi) 1982-12-31
IE790274L (en) 1979-08-14
AU4402879A (en) 1979-08-23
ATA108879A (de) 1981-11-15
EP0003616A3 (en) 1979-09-05
US4273765A (en) 1981-06-16
SE7901276L (sv) 1979-08-15
FI790486A7 (fi) 1979-08-15
NO153011C (no) 1986-01-02
CA1121290A (en) 1982-04-06
DK149599B (da) 1986-08-04
JPS54163511A (en) 1979-12-26

Similar Documents

Publication Publication Date Title
MC1253A1 (fr) Derives amines de sucre utiles notamment comme medicaments
AR240949A1 (es) Procedimiento para preparar derivados de acido n-(aminoalcanoil)-aza-biciclocarboxilico
BE850401A (fr) Derives de phtalane et procede de preparation
DK343980A (da) 2,4,6-triiod-isophthalsyrederivater
DK343880A (da) 2,4,6-triiod-isophthalsyrederivater
BE867517A (fr) Derives amines spiranniques, leur preparation et leur utilisation comme medicaments
FI802918A7 (fi) Aminohappojohdannaisia ja menetelmä niiden valmistamiseksi.
PT65853A (fr) Procede de preparation des derives d'amino-alcools
IT8048605A0 (it) Enzimaticamente l-triptofano procedimento per preparare
DE2961799D1 (en) Acylated 1-azolyl-2-hydroxy-butane derivatives, process for their preparation and their use as fungicides
BE839787A (fr) Procede de preparation d'isocyanates aliphatiques
NL7900264A (nl) 4-pyridon-3-carbonzuurderivaten alsmede de bereiding ervan.
BR7907902A (pt) Derivados de benzamida,composicao herbicida,e processo herbicida
BR8004977A (pt) Derivados de eter difenilico,processo para preparar os mesmos e composicoes herbicidas contendo os mesmos
PT66819A (fr) Procede de preparation de n-(1'-allyl 2'-pyrrolidylmethyl)2,3-dimethoxy 5-sulfamoyl benzamida et ses derives
BE857131A (fr) Procede de preparation de proteine monocellulaire
IT1120444B (it) Procedimento per la preparazione di n,n-bis(n-ciano-n-alcinil)-metanimmidammidil)-cistammine e prodotto ottenuto
BE879663A (fr) Procede de preparation du p-aminophenol ameliore
BE815971A (fr) Procede de preparation d'amines et d'urees substituees
NZ191699A (en) N-(1-methyl-2-pyrrolidinyl methyl)-2,3-dimethoxy-5-methyl-sulphamoyl benzamide derivatives pharmaceutical compositions
PT67729A (fr) Procede de preparation de nouveaux derives de l'oxadiazole-1,3,4 et de compositions iongicides qui en contiennent
IL57693A (en) Pharmaceutical compositions with increased hypotensive effect comprising two amine derivatives and their preparation
EG13794A (en) N-(o-ethyl-s-n-propyl-(di)thiophosphoryloxy)-naphthal-imides,process for their preparation and their use as pesticides
FI803177A7 (fi) Menetelmä 3-syanopropionihappoamidin valmistamiseksi.
IT1162430B (it) Antibiotico bn-183b,procedimento per produrlo e composizioni farmaceutiche che lo contengono

Legal Events

Date Code Title Description
YP Annual fee paid