MA54223A - Dérivés de 2,3-dihydro-1h-pyrrolo[3,4-c]pyridin-1-one servant d'inhibiteurs de hpk1 pour le traitement du cancer - Google Patents
Dérivés de 2,3-dihydro-1h-pyrrolo[3,4-c]pyridin-1-one servant d'inhibiteurs de hpk1 pour le traitement du cancerInfo
- Publication number
- MA54223A MA54223A MA054223A MA54223A MA54223A MA 54223 A MA54223 A MA 54223A MA 054223 A MA054223 A MA 054223A MA 54223 A MA54223 A MA 54223A MA 54223 A MA54223 A MA 54223A
- Authority
- MA
- Morocco
- Prior art keywords
- pyrrolo
- pyridin
- dihydro
- cancer
- treatment
- Prior art date
Links
- QDSJMVZVUSYEMY-UHFFFAOYSA-N 2,3-dihydropyrrolo[3,4-c]pyridin-1-one Chemical class N1=CC=C2C(=O)NCC2=C1 QDSJMVZVUSYEMY-UHFFFAOYSA-N 0.000 title 1
- 101001059991 Homo sapiens Mitogen-activated protein kinase kinase kinase kinase 1 Proteins 0.000 title 1
- 102100028199 Mitogen-activated protein kinase kinase kinase kinase 1 Human genes 0.000 title 1
- 206010028980 Neoplasm Diseases 0.000 title 1
- 201000011510 cancer Diseases 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862767602P | 2018-11-15 | 2018-11-15 | |
PCT/IB2019/059702 WO2020100027A1 (fr) | 2018-11-15 | 2019-11-12 | Dérivés de 2,3-dihydro-1h-pyrrolo[3,4-c]pyridin-1-one servant d'inhibiteurs de hpk1 pour le traitement du cancer |
Publications (2)
Publication Number | Publication Date |
---|---|
MA54223A true MA54223A (fr) | 2022-02-23 |
MA54223B1 MA54223B1 (fr) | 2023-10-31 |
Family
ID=77369712
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA54223A MA54223B1 (fr) | 2018-11-15 | 2019-11-12 | Dérivés de 2,3-dihydro-1h-pyrrolo[3,4-c]pyridin-1-one en tant qu'inhibiteurs de hpk1 pour le traitement du cancer |
Country Status (2)
Country | Link |
---|---|
AR (1) | AR117073A1 (fr) |
MA (1) | MA54223B1 (fr) |
-
2019
- 2019-11-12 MA MA54223A patent/MA54223B1/fr unknown
- 2019-11-14 AR ARP190103343A patent/AR117073A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
MA54223B1 (fr) | 2023-10-31 |
AR117073A1 (es) | 2021-07-07 |
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