MA53098A - Médicament pour prévenir ou traiter une maladie ophtalmique associée à une néovascularisation intraoculaire et/ou à une perméabilité vasculaire intraoculaire accrues - Google Patents

Médicament pour prévenir ou traiter une maladie ophtalmique associée à une néovascularisation intraoculaire et/ou à une perméabilité vasculaire intraoculaire accrues

Info

Publication number
MA53098A
MA53098A MA053098A MA53098A MA53098A MA 53098 A MA53098 A MA 53098A MA 053098 A MA053098 A MA 053098A MA 53098 A MA53098 A MA 53098A MA 53098 A MA53098 A MA 53098A
Authority
MA
Morocco
Prior art keywords
medicine
preventing
disease associated
vascular permeability
ophthalmic disease
Prior art date
Application number
MA053098A
Other languages
English (en)
Inventor
Tomohiro Aoki
Ichiro Aramori
Hideaki Hara
Shuh Narumiya
Rie Yamamoto
Original Assignee
Astellas Pharma Inc
Univ Kyoto
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astellas Pharma Inc, Univ Kyoto filed Critical Astellas Pharma Inc
Publication of MA53098A publication Critical patent/MA53098A/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41841,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/453Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with oxygen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
MA053098A 2018-02-02 2019-02-01 Médicament pour prévenir ou traiter une maladie ophtalmique associée à une néovascularisation intraoculaire et/ou à une perméabilité vasculaire intraoculaire accrues MA53098A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2018016911 2018-02-02

Publications (1)

Publication Number Publication Date
MA53098A true MA53098A (fr) 2021-05-12

Family

ID=67479734

Family Applications (1)

Application Number Title Priority Date Filing Date
MA053098A MA53098A (fr) 2018-02-02 2019-02-01 Médicament pour prévenir ou traiter une maladie ophtalmique associée à une néovascularisation intraoculaire et/ou à une perméabilité vasculaire intraoculaire accrues

Country Status (17)

Country Link
US (1) US20210113529A1 (fr)
EP (1) EP3747471A4 (fr)
JP (1) JPWO2019151470A1 (fr)
KR (1) KR20200116953A (fr)
CN (1) CN111683682A (fr)
AU (1) AU2019214265A1 (fr)
BR (1) BR112020015567A2 (fr)
CA (1) CA3089952A1 (fr)
IL (1) IL275603A (fr)
JO (1) JOP20200186A1 (fr)
MA (1) MA53098A (fr)
MX (1) MX2020007948A (fr)
PH (1) PH12020551015A1 (fr)
RU (1) RU2020128700A (fr)
SG (1) SG11202006255UA (fr)
WO (1) WO2019151470A1 (fr)
ZA (1) ZA202004327B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021148439A1 (fr) * 2020-01-21 2021-07-29 INSERM (Institut National de la Santé et de la Recherche Médicale) Procédés de stimulation de la fonction cérébrovasculaire
WO2021163355A1 (fr) * 2020-02-11 2021-08-19 Arena Pharmaceuticals, Inc. Formulations et méthodes de traitement d'affections liées au récepteur s1p1
CN113082031A (zh) * 2021-03-09 2021-07-09 温州医科大学附属眼视光医院 一种多巴胺d1和d2受体非选择性激动剂在作为制备治疗眼部病理性血管新生药物的应用

Family Cites Families (27)

* Cited by examiner, † Cited by third party
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CN100431534C (zh) 2003-06-24 2008-11-12 康涅狄格大学 血管内皮鞘氨醇-1-磷酸受体拮抗剂在制备药物中的应用
US7794713B2 (en) 2004-04-07 2010-09-14 Lpath, Inc. Compositions and methods for the treatment and prevention of hyperproliferative diseases
EP1798226A4 (fr) 2004-08-04 2009-06-17 Taisho Pharmaceutical Co Ltd Derive de traizol
GB0504544D0 (en) * 2005-03-04 2005-04-13 Novartis Ag Organic compounds
WO2007089018A1 (fr) 2006-02-03 2007-08-09 Taisho Pharmaceutical Co., Ltd. Dérivé de triazole
CN101415687B (zh) 2006-02-06 2012-02-08 大正制药株式会社 鞘氨醇-1-磷酸结合抑制物质
BRPI0709866B8 (pt) * 2006-04-03 2021-05-25 Astellas Pharma Inc compostos héteros e composição farmacêutica compreendendo ditos compostos
WO2008055072A2 (fr) 2006-10-27 2008-05-08 Lpath, Inc. Compositions et procédés pour traiter des maladies et des troubles oculaires
CA2666709A1 (fr) 2006-11-10 2008-05-29 Genentech, Inc. Procede pour traiter une degenerescence maculaire liee a l'age
EP2014653A1 (fr) 2007-06-15 2009-01-14 Bioprojet Nouveaux dérivés d'acide dicarboxylique comme agonistes du recepteur S1P1
DK2177512T3 (da) 2007-08-01 2012-06-18 Taisho Pharmaceutical Co Ltd S1P1-bindingshæmmer
KR101589332B1 (ko) 2008-12-05 2016-01-27 아스텔라스세이야쿠 가부시키가이샤 2h-크로멘 화합물 및 그의 유도체
JP2013508385A (ja) 2009-10-23 2013-03-07 アラーガン インコーポレイテッド 治療上有用な、受容体修飾薬としてのクマリン化合物
CA2780987C (fr) 2009-11-24 2018-03-06 Allergan, Inc. Nouveaux composes servant de modulateurs de recepteurs presentant une utilite therapeutique
WO2011087066A1 (fr) 2010-01-14 2011-07-21 株式会社三和化学研究所 Produit pharmaceutique destiné au traitement prophylactique ou thérapeutique de troubles accompagnés d'une angiogenèse oculaire et/ou d'une perméabilité vasculaire oculaire supérieure à la normale
US8273776B2 (en) 2010-04-16 2012-09-25 Allergan, Inc Biphenyl oxadiazole derivatives as sphingosine-1-phosphate receptors modulators
US8530462B2 (en) 2010-11-24 2013-09-10 Allergan, Inc. Indole modulators of S1P receptors
EP2643303A1 (fr) 2010-11-24 2013-10-02 Allergan, Inc. Modulateurs de récepteurs de la s1p
BR112013013633A2 (pt) 2010-12-03 2016-11-08 Allergan Inc derivados de alquina e alceno como moduladores do receptor de esfingosina 1-fosfato-1
WO2012105610A1 (fr) 2011-02-02 2012-08-09 公立大学法人名古屋市立大学 Agent médicinal pour la prévention ou le traitement de maladies associées à une néovascularisation intraoculaire et/ou une hyperperméabilité vasculaire intraoculaire
CA2833305A1 (fr) 2011-04-14 2012-10-18 Allergan, Inc. Derives de methylazetidines bicycliques phenyliques en tant que modulateurs des recepteurs de sphingosine-1 phosphate
WO2012145236A1 (fr) 2011-04-18 2012-10-26 Allergan, Inc. Dérivés de méthylamines bicycliques substitués à titre de modulateurs des récepteurs de sphingosine-1 phosphate
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JP2018016911A (ja) 2016-07-28 2018-02-01 村田機械株式会社 解析装置

Also Published As

Publication number Publication date
CA3089952A1 (fr) 2019-08-08
BR112020015567A2 (pt) 2021-02-02
EP3747471A1 (fr) 2020-12-09
SG11202006255UA (en) 2020-07-29
PH12020551015A1 (en) 2021-09-06
US20210113529A1 (en) 2021-04-22
ZA202004327B (en) 2022-01-26
RU2020128700A (ru) 2022-03-02
RU2020128700A3 (fr) 2022-03-02
JPWO2019151470A1 (ja) 2021-02-25
WO2019151470A1 (fr) 2019-08-08
MX2020007948A (es) 2020-12-10
AU2019214265A1 (en) 2020-07-23
JOP20200186A1 (ar) 2020-07-29
CN111683682A (zh) 2020-09-18
EP3747471A4 (fr) 2021-10-27
IL275603A (en) 2020-08-31
KR20200116953A (ko) 2020-10-13

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