MA48728B1 - Niraparib, acétate d'abiratérone et prednisone pour le traitement du cancer de la prostate - Google Patents

Niraparib, acétate d'abiratérone et prednisone pour le traitement du cancer de la prostate

Info

Publication number
MA48728B1
MA48728B1 MA48728A MA48728A MA48728B1 MA 48728 B1 MA48728 B1 MA 48728B1 MA 48728 A MA48728 A MA 48728A MA 48728 A MA48728 A MA 48728A MA 48728 B1 MA48728 B1 MA 48728B1
Authority
MA
Morocco
Prior art keywords
niraparib
prednisone
prostate cancer
abiraterone acetate
treatment
Prior art date
Application number
MA48728A
Other languages
English (en)
Other versions
MA48728A (fr
Inventor
Margaret K Yu
Linda Anne Snyder
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=62067858&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA48728(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of MA48728A publication Critical patent/MA48728A/fr
Publication of MA48728B1 publication Critical patent/MA48728B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

L'invention concerne des méthodes et des compositions permettant de traiter le cancer de la prostate par l'administration à un patient qui en a besoin d'une quantité thérapeutiquement efficace d'un inhibiteur de parp, par exemple le niraparib ; d'une quantité thérapeutiquement efficace d'un inhibiteur de cyp17, par exemple, l'acétate d'abiratérone, et d'une quantité thérapeutiquement efficace d'un glucocorticoïde, par exemple la prednisone.
MA48728A 2017-04-13 2018-04-09 Niraparib, acétate d'abiratérone et prednisone pour le traitement du cancer de la prostate MA48728B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762485164P 2017-04-13 2017-04-13
PCT/US2018/026661 WO2018191141A1 (fr) 2017-04-13 2018-04-09 Polythérapie contre le cancer de la prostate

Publications (2)

Publication Number Publication Date
MA48728A MA48728A (fr) 2020-04-08
MA48728B1 true MA48728B1 (fr) 2022-10-31

Family

ID=62067858

Family Applications (1)

Application Number Title Priority Date Filing Date
MA48728A MA48728B1 (fr) 2017-04-13 2018-04-09 Niraparib, acétate d'abiratérone et prednisone pour le traitement du cancer de la prostate

Country Status (30)

Country Link
US (2) US20180296574A1 (fr)
EP (3) EP4176879A1 (fr)
JP (3) JP7141408B2 (fr)
KR (1) KR20190134718A (fr)
CN (1) CN110753545A (fr)
AU (2) AU2018251594A1 (fr)
BR (1) BR112019021466A2 (fr)
CA (1) CA3059562A1 (fr)
CL (1) CL2019002871A1 (fr)
CO (1) CO2019011591A2 (fr)
CR (1) CR20190467A (fr)
DK (1) DK3609497T3 (fr)
DO (1) DOP2019000264A (fr)
EA (1) EA201992430A1 (fr)
ES (1) ES2931052T3 (fr)
HR (1) HRP20221327T1 (fr)
HU (1) HUE060460T2 (fr)
JO (1) JOP20190244A1 (fr)
LT (1) LT3609497T (fr)
MA (1) MA48728B1 (fr)
MD (1) MD3609497T2 (fr)
MX (2) MX2019012296A (fr)
NI (1) NI201900105A (fr)
PE (1) PE20200444A1 (fr)
PH (1) PH12019502317A1 (fr)
PL (1) PL3609497T3 (fr)
PT (1) PT3609497T (fr)
RS (1) RS63832B1 (fr)
SG (1) SG11201909552VA (fr)
WO (1) WO2018191141A1 (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20180028521A1 (en) 2016-07-29 2018-02-01 Janssen Pharmaceutica Nv Methods of Treating Prostate Cancer
WO2020139339A1 (fr) * 2018-12-27 2020-07-02 Constellation Pharmaceuticals, Inc. Inhibiteurs de la signalisation de l'ezh2 et du récepteur des androgènes en tant qu'outils pour le ciblage du cancer de la prostate
CN113546037A (zh) * 2020-04-20 2021-10-26 鲁南制药集团股份有限公司 一种醋酸阿比特龙栓剂及其制备方法
IL297984A (en) * 2020-05-08 2023-01-01 Janssen Pharmaceutica Nv Pharmaceutical formulations of abiraterone acetate and niraparib
CN114306236B (zh) * 2021-12-15 2022-10-21 湖南慧泽生物医药科技有限公司 用于负载醋酸阿比特龙的自微乳体系及组合物和应用
TWI828471B (zh) 2021-12-15 2024-01-01 大陸商湖南慧澤生物醫藥科技有限公司 醋酸阿比特龍的自微乳組合物和應用
WO2023194525A1 (fr) * 2022-04-07 2023-10-12 Astrazeneca Ab Polythérapie pour le traitement du cancer

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20080051380A1 (en) * 2006-08-25 2008-02-28 Auerbach Alan H Methods and compositions for treating cancer
EP2478907B1 (fr) * 2006-08-25 2021-04-14 Janssen Oncology, Inc. Compositions pour le traitement du cancer
JP4611444B2 (ja) 2007-01-10 2011-01-12 イステイチユート・デイ・リチエルケ・デイ・ビオロジア・モレコラーレ・ピ・アンジエレツテイ・エツセ・ピー・アー ポリ(adp−リボース)ポリメラーゼ(parp)阻害剤としてのアミド置換インダゾール
KR101653548B1 (ko) 2008-01-08 2016-09-02 머크 샤프 앤드 돔 리미티드 2-{4-[(3s)-피페리딘-3-일]페닐}-2h-인다졸-7-카복스아미드의 약제학적으로 허용되는 염
WO2012009475A1 (fr) * 2010-07-14 2012-01-19 Oregon Health & Science University Méthodes de traitement du cancer par inhibition de la déméthylase 1 spécifique de la lysine
WO2014089324A1 (fr) * 2012-12-07 2014-06-12 Calitor Sciences, Llc Composés cycliques substitués et leurs procédés d'utilisation

Also Published As

Publication number Publication date
US20220175801A1 (en) 2022-06-09
EP3609497A1 (fr) 2020-02-19
ES2931052T3 (es) 2022-12-23
SG11201909552VA (en) 2019-11-28
CA3059562A1 (fr) 2018-10-18
JP2024023344A (ja) 2024-02-21
JP2022141881A (ja) 2022-09-29
PE20200444A1 (es) 2020-02-28
MA48728A (fr) 2020-04-08
JP7141408B2 (ja) 2022-09-22
EP4176879A1 (fr) 2023-05-10
MD3609497T2 (ro) 2023-03-31
MX2023009569A (es) 2023-08-22
AU2024202346A1 (en) 2024-05-02
PH12019502317A1 (en) 2020-07-06
NI201900105A (es) 2020-03-11
JP7407880B2 (ja) 2024-01-04
US20180296574A1 (en) 2018-10-18
EP4176878A1 (fr) 2023-05-10
HRP20221327T1 (hr) 2023-03-17
JP2020516646A (ja) 2020-06-11
EP3609497B1 (fr) 2022-10-12
DOP2019000264A (es) 2020-07-15
HUE060460T2 (hu) 2023-03-28
BR112019021466A2 (pt) 2020-05-12
PT3609497T (pt) 2023-01-23
MX2019012296A (es) 2019-11-28
RS63832B1 (sr) 2023-01-31
JOP20190244A1 (ar) 2019-10-13
KR20190134718A (ko) 2019-12-04
AU2018251594A1 (en) 2019-10-24
CO2019011591A2 (es) 2020-02-28
PL3609497T3 (pl) 2023-01-23
CN110753545A (zh) 2020-02-04
WO2018191141A1 (fr) 2018-10-18
DK3609497T3 (da) 2022-10-31
CL2019002871A1 (es) 2019-12-27
EA201992430A1 (ru) 2020-02-28
LT3609497T (lt) 2022-12-12
CR20190467A (es) 2020-03-09

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