MA45902A - Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine - Google Patents

Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine

Info

Publication number
MA45902A
MA45902A MA045902A MA45902A MA45902A MA 45902 A MA45902 A MA 45902A MA 045902 A MA045902 A MA 045902A MA 45902 A MA45902 A MA 45902A MA 45902 A MA45902 A MA 45902A
Authority
MA
Morocco
Prior art keywords
bruprenorphine
procedures
preparation
acetate salt
acetate
Prior art date
Application number
MA045902A
Other languages
English (en)
Inventor
C Frederick M Huntley
Erik Wayne Kataisto
Helge Alfred Reisch
Archana Sharma
Jake Larry Stymiest
Original Assignee
Rhodes Tech
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhodes Tech filed Critical Rhodes Tech
Publication of MA45902A publication Critical patent/MA45902A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/09—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems
    • C07D489/10—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14
    • C07D489/12—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14 the bridge containing only two carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Steroid Compounds (AREA)
MA045902A 2015-03-10 2016-03-09 Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine MA45902A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562131114P 2015-03-10 2015-03-10

Publications (1)

Publication Number Publication Date
MA45902A true MA45902A (fr) 2019-06-19

Family

ID=55524412

Family Applications (1)

Application Number Title Priority Date Filing Date
MA045902A MA45902A (fr) 2015-03-10 2016-03-09 Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine

Country Status (19)

Country Link
US (6) US10406152B2 (fr)
EP (1) EP3283490A1 (fr)
JP (2) JP6660399B2 (fr)
KR (2) KR20170137738A (fr)
CN (1) CN107660207B (fr)
AR (1) AR103902A1 (fr)
AU (2) AU2016230750B2 (fr)
BR (1) BR112017019357A2 (fr)
CA (2) CA2977732C (fr)
CO (1) CO2017009130A2 (fr)
EA (1) EA201792014A1 (fr)
IL (1) IL254384A0 (fr)
MA (1) MA45902A (fr)
MX (1) MX2017011606A (fr)
NZ (1) NZ735736A (fr)
PH (1) PH12017501641A1 (fr)
SG (1) SG11201707350TA (fr)
TW (2) TWI699367B (fr)
WO (1) WO2016142877A1 (fr)

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DK3553177T3 (da) 2013-03-15 2021-02-15 Univ Leland Stanford Junior Benzylisoquinolinalkaloider (bia) som producerer mikrober, og fremgangsmåder til fremstilling og anvendelse deraf
WO2015066642A1 (fr) 2013-11-04 2015-05-07 The Board Of Trustees Of The Leland Stanford Junior University Microbes produisant des précurseurs d'un alcaloïde, la benzylisoquinoline, et leurs procédés de production et d'utilisation
KR20170137738A (ko) 2015-03-10 2017-12-13 로드스 테크놀로지즈 부프레노르핀의 아세테이트 염 및 부프레노르핀의 제조방법
EP3292203A4 (fr) 2015-05-04 2019-10-09 The Board of Trustees of the Leland Stanford Junior University Précuseur d'alcaloïde de benzylisoquinoline (bia) produisant des microbes, et ses procédés de fabrication et d'utilisation
WO2016183023A1 (fr) 2015-05-08 2016-11-17 The Board Of Trustees Of The Leland Stanford Junior University Procédés de production d'épimérases et d'alcaloïdes benzylisoquinoléine
WO2018075670A1 (fr) 2016-10-18 2018-04-26 Antheia, Inc. Procédés de production d'alcaloïdes de benzylisoquinoline nor-opioïdes et nal-opioïdes
JP7199417B2 (ja) 2017-08-03 2023-01-05 アンテイア インコーポレイテッド 遺伝子操作されたベンジルイソキノリンアルカロイドエピメラーゼおよびベンジルイソキノリンアルカロイドの生成方法
AU2019266795B2 (en) 2018-05-11 2023-02-09 Alar Pharmaceuticals Inc. Long-acting injectable formulations and crystalline forms of buprenorphine derivatives
JP7779737B2 (ja) 2019-03-08 2025-12-03 ザ ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティー トロパンアルカロイド（ｔａ）産生非植物宿主細胞、ならびにその製造方法および使用方法
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Also Published As

Publication number Publication date
US10278967B2 (en) 2019-05-07
CA2977732C (fr) 2021-02-23
EP3283490A1 (fr) 2018-02-21
AU2016230750B2 (en) 2019-05-30
US10874662B2 (en) 2020-12-29
AR103902A1 (es) 2017-06-14
CO2017009130A2 (es) 2017-11-21
WO2016142877A1 (fr) 2016-09-15
KR20200045010A (ko) 2020-04-29
JP6660399B2 (ja) 2020-03-11
AU2016230750A1 (en) 2017-10-12
US20180235955A1 (en) 2018-08-23
CN107660207B (zh) 2020-09-29
TWI699367B (zh) 2020-07-21
IL254384A0 (en) 2017-11-30
TW202037597A (zh) 2020-10-16
JP2018507882A (ja) 2018-03-22
CN107660207A (zh) 2018-02-02
KR20170137738A (ko) 2017-12-13
US10406152B2 (en) 2019-09-10
US9926329B2 (en) 2018-03-27
NZ735736A (en) 2019-02-22
US20190314364A1 (en) 2019-10-17
CA3104099A1 (fr) 2016-09-15
US20170197975A1 (en) 2017-07-13
US20190298713A1 (en) 2019-10-03
JP2020033359A (ja) 2020-03-05
EA201792014A1 (ru) 2018-01-31
AU2019203308A1 (en) 2019-05-30
BR112017019357A2 (pt) 2018-06-05
US20210046066A1 (en) 2021-02-18
SG11201707350TA (en) 2017-10-30
US10835528B2 (en) 2020-11-17
CA2977732A1 (fr) 2016-09-15
TW201639856A (zh) 2016-11-16
PH12017501641A1 (en) 2018-02-12
MX2017011606A (es) 2017-10-26
US20180162866A1 (en) 2018-06-14

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