MA45902A - Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine - Google Patents

Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine

Info

Publication number
MA45902A
MA45902A MA045902A MA45902A MA45902A MA 45902 A MA45902 A MA 45902A MA 045902 A MA045902 A MA 045902A MA 45902 A MA45902 A MA 45902A MA 45902 A MA45902 A MA 45902A
Authority
MA
Morocco
Prior art keywords
bruprenorphine
procedures
preparation
acetate salt
acetate
Prior art date
Application number
MA045902A
Other languages
English (en)
Inventor
C Frederick M Huntley
Erik Wayne Kataisto
Helge Alfred Reisch
Archana Sharma
Jake Larry Stymiest
Original Assignee
Rhodes Tech
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhodes Tech filed Critical Rhodes Tech
Publication of MA45902A publication Critical patent/MA45902A/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
    • C07D489/09—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems
    • C07D489/10—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14
    • C07D489/12—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: containing 4aH-8, 9 c-Iminoethano- phenanthro [4, 5-b, c, d] furan ring systems condensed with carbocyclic rings or ring systems with a bridge between positions 6 and 14 the bridge containing only two carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
MA045902A 2015-03-10 2016-03-09 Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine MA45902A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562131114P 2015-03-10 2015-03-10

Publications (1)

Publication Number Publication Date
MA45902A true MA45902A (fr) 2019-06-19

Family

ID=55524412

Family Applications (1)

Application Number Title Priority Date Filing Date
MA045902A MA45902A (fr) 2015-03-10 2016-03-09 Sel d'acã‰tate de bruprã‰norphine et procã‰dã‰s pour la prã‰paration de bruprã‰norphine

Country Status (19)

Country Link
US (6) US10406152B2 (fr)
EP (1) EP3283490A1 (fr)
JP (2) JP6660399B2 (fr)
KR (2) KR20200045010A (fr)
CN (1) CN107660207B (fr)
AR (1) AR103902A1 (fr)
AU (2) AU2016230750B2 (fr)
BR (1) BR112017019357A2 (fr)
CA (2) CA3104099A1 (fr)
CO (1) CO2017009130A2 (fr)
EA (1) EA201792014A1 (fr)
IL (1) IL254384A0 (fr)
MA (1) MA45902A (fr)
MX (1) MX2017011606A (fr)
NZ (1) NZ735736A (fr)
PH (1) PH12017501641A1 (fr)
SG (1) SG11201707350TA (fr)
TW (2) TW202037597A (fr)
WO (1) WO2016142877A1 (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2970999A2 (fr) 2013-03-15 2016-01-20 The Board Of Trustees Of The University Of the Leland Stanford Junior University Microbes produisant des alcaloïdes de benzylisiquinoline (bia) et leurs procédés de fabrication et d'utilisation
US11124814B2 (en) 2013-11-04 2021-09-21 The Board Of Trustees Of The Leland Stanford Junior University Benzylisoquinoline alkaloid (BIA) precursor producing microbes, and methods of making and using the same
CA3104099A1 (fr) 2015-03-10 2016-09-15 Rhodes Technologies Sel d'acetate de bruprenorphine et procedes pour la preparation de bruprenorphine
CA2983419A1 (fr) 2015-05-04 2016-11-10 The Board Of Trustees Of The Leland Stanford Junior University Precuseur d'alcaloide de benzylisoquinoline (bia) produisant des microbes, et ses procedes de fabrication et d'utilisation
CN107960102A (zh) 2015-05-08 2018-04-24 小利兰·斯坦福大学托管委员会 产生差向异构酶和苄基异喹啉生物碱的方法
CA3043591A1 (fr) 2016-10-18 2018-04-26 Antheia, Inc. Procedes de production d'alcaloides de benzylisoquinoline nor-opioides et nal-opioides
WO2019028390A1 (fr) 2017-08-03 2019-02-07 Antheia, Inc. Alcaloïde benzylisoquinoléine épimérases génétiquement modifiées et procédés de production des alcaloïdes benzylisoquinoléine
CA3089256C (fr) * 2018-05-11 2023-10-10 Alar Pharmaceuticals Inc. Formulations injectables a action prolongee et formes cristallines de derives de buprenorphine
CA3132968A1 (fr) 2019-03-08 2020-09-17 The Board Of Trustees Of The Leland Stanford Junior Unversity Cellules hotes non vegetales produisant des alcaloides tropaniques (at) et procedes de production et d'utilisation associes
CA3260542A1 (fr) * 2022-06-24 2023-12-28 Alar Pharmaceuticals Inc. Composition pharmaceutique stable de buprénorphine et son procédé de préparation et son utilisation

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Also Published As

Publication number Publication date
JP2020033359A (ja) 2020-03-05
CA2977732A1 (fr) 2016-09-15
AU2016230750B2 (en) 2019-05-30
US20180235955A1 (en) 2018-08-23
US20190314364A1 (en) 2019-10-17
CA2977732C (fr) 2021-02-23
AR103902A1 (es) 2017-06-14
MX2017011606A (es) 2017-10-26
JP2018507882A (ja) 2018-03-22
NZ735736A (en) 2019-02-22
KR20200045010A (ko) 2020-04-29
PH12017501641A1 (en) 2018-02-12
SG11201707350TA (en) 2017-10-30
US10835528B2 (en) 2020-11-17
TWI699367B (zh) 2020-07-21
US9926329B2 (en) 2018-03-27
CO2017009130A2 (es) 2017-11-21
JP6660399B2 (ja) 2020-03-11
CN107660207B (zh) 2020-09-29
AU2016230750A1 (en) 2017-10-12
CN107660207A (zh) 2018-02-02
US10874662B2 (en) 2020-12-29
US20210046066A1 (en) 2021-02-18
WO2016142877A1 (fr) 2016-09-15
US20190298713A1 (en) 2019-10-03
US10406152B2 (en) 2019-09-10
BR112017019357A2 (pt) 2018-06-05
IL254384A0 (en) 2017-11-30
EP3283490A1 (fr) 2018-02-21
KR20170137738A (ko) 2017-12-13
AU2019203308A1 (en) 2019-05-30
EA201792014A1 (ru) 2018-01-31
CA3104099A1 (fr) 2016-09-15
US10278967B2 (en) 2019-05-07
US20180162866A1 (en) 2018-06-14
TW201639856A (zh) 2016-11-16
TW202037597A (zh) 2020-10-16
US20170197975A1 (en) 2017-07-13

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