MA28548B1 - Composes macrocycliques inhibiteurs de replication virale - Google Patents

Composes macrocycliques inhibiteurs de replication virale

Info

Publication number
MA28548B1
MA28548B1 MA29407A MA29407A MA28548B1 MA 28548 B1 MA28548 B1 MA 28548B1 MA 29407 A MA29407 A MA 29407A MA 29407 A MA29407 A MA 29407A MA 28548 B1 MA28548 B1 MA 28548B1
Authority
MA
Morocco
Prior art keywords
viral replication
macrocyclic compounds
replication inhibitors
inhibitors
macrocyclic
Prior art date
Application number
MA29407A
Other languages
English (en)
Inventor
Lawrence M Blatt
Steven M Wenglowsky
Steven W Andrews
Yutong Jiang
April L Kennedy
Kevin R Condroski
John A Josey
Peter J Stengel
Machender R Madduru
George A Doherty
Benjamin T Woodard
Original Assignee
Intermune Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Intermune Inc filed Critical Intermune Inc
Publication of MA28548B1 publication Critical patent/MA28548B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
MA29407A 2004-03-30 2006-10-20 Composes macrocycliques inhibiteurs de replication virale MA28548B1 (fr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US55816104P 2004-03-30 2004-03-30
US56241804P 2004-04-14 2004-04-14
US61246004P 2004-09-22 2004-09-22
US61238104P 2004-09-22 2004-09-22

Publications (1)

Publication Number Publication Date
MA28548B1 true MA28548B1 (fr) 2007-04-03

Family

ID=35005653

Family Applications (1)

Application Number Title Priority Date Filing Date
MA29407A MA28548B1 (fr) 2004-03-30 2006-10-20 Composes macrocycliques inhibiteurs de replication virale

Country Status (16)

Country Link
EP (1) EP1749007A2 (fr)
JP (1) JP4950026B2 (fr)
AP (1) AP2006003763A0 (fr)
AR (1) AR050321A1 (fr)
AU (1) AU2005228894B9 (fr)
BR (1) BRPI0509467A (fr)
CA (1) CA2560897C (fr)
CU (1) CU23787B7 (fr)
EA (1) EA012389B1 (fr)
EC (1) ECSP066959A (fr)
GE (1) GEP20104926B (fr)
IL (1) IL177917A0 (fr)
MA (1) MA28548B1 (fr)
NO (1) NO20064933L (fr)
NZ (1) NZ549697A (fr)
WO (1) WO2005095403A2 (fr)

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Also Published As

Publication number Publication date
GEP20104926B (en) 2010-03-25
ECSP066959A (es) 2006-12-20
AU2005228894B2 (en) 2011-08-25
CA2560897A1 (fr) 2005-10-13
EP1749007A2 (fr) 2007-02-07
AU2005228894A1 (en) 2005-10-13
WO2005095403A3 (fr) 2005-12-01
JP2007531749A (ja) 2007-11-08
IL177917A0 (en) 2006-12-31
JP4950026B2 (ja) 2012-06-13
AP2006003763A0 (en) 2006-10-31
NO20064933L (no) 2006-12-15
CA2560897C (fr) 2012-06-12
CU23787B7 (es) 2012-03-15
AU2005228894B9 (en) 2011-10-13
BRPI0509467A (pt) 2007-09-11
AR050321A1 (es) 2006-10-18
EA200601467A1 (ru) 2007-06-29
WO2005095403A2 (fr) 2005-10-13
CU20090209A7 (es) 2011-04-26
NZ549697A (en) 2009-12-24
EA012389B1 (ru) 2009-10-30

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