KR960700227A - 저콜레스테린혈증제로서 유용한 스피로사이클로알킬 치환된 아제티디논(Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents) - Google Patents

저콜레스테린혈증제로서 유용한 스피로사이클로알킬 치환된 아제티디논(Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents)

Info

Publication number
KR960700227A
KR960700227A KR1019950702988A KR19950702988A KR960700227A KR 960700227 A KR960700227 A KR 960700227A KR 1019950702988 A KR1019950702988 A KR 1019950702988A KR 19950702988 A KR19950702988 A KR 19950702988A KR 960700227 A KR960700227 A KR 960700227A
Authority
KR
South Korea
Prior art keywords
optionally
alkenylene
sum
substituted
image
Prior art date
Application number
KR1019950702988A
Other languages
English (en)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of KR960700227A publication Critical patent/KR960700227A/ko

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10Spiro-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/12Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom condensed with carbocyclic rings or ring systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1019950702988A 1993-01-21 1995-07-21 저콜레스테린혈증제로서 유용한 스피로사이클로알킬 치환된 아제티디논(Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents) KR960700227A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US643993A 1993-01-21 1993-01-21
PCT/US1994/000421 WO1994017038A1 (en) 1993-01-21 1994-01-19 Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents

Publications (1)

Publication Number Publication Date
KR960700227A true KR960700227A (ko) 1996-01-19

Family

ID=21720894

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019950702988A KR960700227A (ko) 1993-01-21 1995-07-21 저콜레스테린혈증제로서 유용한 스피로사이클로알킬 치환된 아제티디논(Spirocycloalkyl-substituted azetidinones useful as hypocholesterolemic agents)

Country Status (26)

Country Link
US (1) US5698548A (ko)
EP (1) EP0681569B1 (ko)
JP (1) JP2719445B2 (ko)
KR (1) KR960700227A (ko)
CN (1) CN1118163A (ko)
AT (1) ATE199899T1 (ko)
AU (1) AU683048B2 (ko)
CA (1) CA2154257C (ko)
CZ (1) CZ180195A3 (ko)
DE (1) DE69426924T2 (ko)
DK (1) DK0681569T3 (ko)
EE (1) EE9400394A (ko)
ES (1) ES2155849T3 (ko)
FI (1) FI953497A0 (ko)
GR (1) GR3035963T3 (ko)
HU (1) HUT72592A (ko)
IL (1) IL108368A0 (ko)
LT (1) LT3595B (ko)
NO (1) NO952884L (ko)
NZ (1) NZ261714A (ko)
PL (1) PL309978A1 (ko)
PT (1) PT681569E (ko)
SI (1) SI9400022A (ko)
SK (1) SK91195A3 (ko)
WO (1) WO1994017038A1 (ko)
ZA (1) ZA94386B (ko)

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JP4589919B2 (ja) 2003-03-07 2010-12-01 シェーリング コーポレイション 高コレステロール血症の処置のための、置換アゼチジノン化合物、これらの処方物および使用
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CN101541805A (zh) * 2006-09-15 2009-09-23 先灵公司 用于治疗疼痛和脂代射紊乱的氮杂环丁烷和氮杂环丁酮衍生物
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Also Published As

Publication number Publication date
LT3595B (en) 1995-12-27
NO952884L (no) 1995-09-20
NZ261714A (en) 1997-02-24
JP2719445B2 (ja) 1998-02-25
CA2154257C (en) 1999-05-25
DE69426924T2 (de) 2001-08-16
CZ180195A3 (en) 1996-01-17
ZA94386B (en) 1994-07-19
NO952884D0 (no) 1995-07-20
GR3035963T3 (en) 2001-08-31
HUT72592A (en) 1996-05-28
SK91195A3 (en) 1995-12-06
JPH08501110A (ja) 1996-02-06
PL309978A1 (en) 1995-11-13
FI953497A (fi) 1995-07-20
WO1994017038A1 (en) 1994-08-04
ATE199899T1 (de) 2001-04-15
AU683048B2 (en) 1997-10-30
CN1118163A (zh) 1996-03-06
CA2154257A1 (en) 1994-08-04
EP0681569B1 (en) 2001-03-21
EP0681569A1 (en) 1995-11-15
PT681569E (pt) 2001-06-29
ES2155849T3 (es) 2001-06-01
SI9400022A (en) 1995-02-28
EE9400394A (et) 1996-06-17
HU9502194D0 (en) 1995-09-28
IL108368A0 (en) 1994-04-12
FI953497A0 (fi) 1995-07-20
US5698548A (en) 1997-12-16
LTIP1764A (en) 1995-02-27
DE69426924D1 (de) 2001-04-26
AU6087294A (en) 1994-08-15
DK0681569T3 (da) 2001-04-23

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