KR920005845B1 - 2,4,5-트리할로게노- 및 2,3,4,5-테트라할로게노벤젠 유도체의 제조방법 - Google Patents

2,4,5-트리할로게노- 및 2,3,4,5-테트라할로게노벤젠 유도체의 제조방법 Download PDF

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Publication number
KR920005845B1
KR920005845B1 KR1019850003889A KR850003889A KR920005845B1 KR 920005845 B1 KR920005845 B1 KR 920005845B1 KR 1019850003889 A KR1019850003889 A KR 1019850003889A KR 850003889 A KR850003889 A KR 850003889A KR 920005845 B1 KR920005845 B1 KR 920005845B1
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chloro
acid
chloride
reaction
oxo
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KR1019850003889A
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Korean (ko)
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KR860000240A (ko
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클라우케 에리히
페터슨 우베
그로에 클라우스
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바이엘악티엔게젤샤프트
에리히 데브리쯔, 요아힘 그렘
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C63/00—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/093—Preparation of halogenated hydrocarbons by replacement by halogens
    • C07C17/10—Preparation of halogenated hydrocarbons by replacement by halogens of hydrogen atoms
    • C07C17/14—Preparation of halogenated hydrocarbons by replacement by halogens of hydrogen atoms in the side-chain of aromatic compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/093—Preparation of halogenated hydrocarbons by replacement by halogens
    • C07C17/16—Preparation of halogenated hydrocarbons by replacement by halogens of hydroxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/02—Monocyclic aromatic halogenated hydrocarbons
    • C07C25/13—Monocyclic aromatic halogenated hydrocarbons containing fluorine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40—Halogenated unsaturated alcohols
    • C07C33/46—Halogenated unsaturated alcohols containing only six-membered aromatic rings as cyclic parts
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/27—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/29—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
    • C07C45/292—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups with chromium derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/42—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by hydrolysis
    • C07C45/43—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by hydrolysis of >CX2 groups, X being halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C47/00—Compounds having —CHO groups
    • C07C47/52—Compounds having —CHO groups bound to carbon atoms of six—membered aromatic rings
    • C07C47/55—Compounds having —CHO groups bound to carbon atoms of six—membered aromatic rings containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C63/00—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings
    • C07C63/68—Compounds having carboxyl groups bound to a carbon atoms of six-membered aromatic rings containing halogen
    • C07C63/70—Monocarboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
KR1019850003889A 1984-06-04 1985-06-04 2,4,5-트리할로게노- 및 2,3,4,5-테트라할로게노벤젠 유도체의 제조방법 Expired KR920005845B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19843420796 DE3420796A1 (de) 1984-06-04 1984-06-04 2,4,5-trihalogen- bzw. 2,3,4,5-tetrahalogenbenzolderivate und verfahren zu ihrer herstellung
DEP3420796.1 1984-06-04

Publications (2)

Publication Number Publication Date
KR860000240A KR860000240A (ko) 1986-01-27
KR920005845B1 true KR920005845B1 (ko) 1992-07-23

Family

ID=6237596

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019850003889A Expired KR920005845B1 (ko) 1984-06-04 1985-06-04 2,4,5-트리할로게노- 및 2,3,4,5-테트라할로게노벤젠 유도체의 제조방법

Country Status (8)

Country Link
US (1) US5072038A (cg-RX-API-DMAC7.html)
EP (1) EP0164619B1 (cg-RX-API-DMAC7.html)
JP (1) JPS617220A (cg-RX-API-DMAC7.html)
KR (1) KR920005845B1 (cg-RX-API-DMAC7.html)
AT (1) ATE37866T1 (cg-RX-API-DMAC7.html)
CA (1) CA1242742A (cg-RX-API-DMAC7.html)
DE (2) DE3420796A1 (cg-RX-API-DMAC7.html)
HU (1) HU195176B (cg-RX-API-DMAC7.html)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0174131A3 (en) * 1984-09-01 1989-06-07 FISONS plc Dihydropyridines, processes and intermediates for their production, and pharmaceutical formulations containing them
EP0230946A3 (en) * 1986-01-20 1988-09-07 Kyorin Pharmaceutical Co., Ltd. Process for the preparation of quinolonecarboxylic acid derivatives
US4791225A (en) * 1986-01-20 1988-12-13 Kyorin Pharmaceutical Co., Ltd. Halogenobenzoic acid derivatives and their preparation
US5286754A (en) * 1986-01-21 1994-02-15 Bayer Aktiengesellschaft Pharmaceutical formulations of ciprofloxacin
DE3601566A1 (de) * 1986-01-21 1987-07-23 Bayer Ag Pharmazeutische zubereitungen von ciprofloxacin
JPS62192321A (ja) * 1986-02-19 1987-08-22 Bayer Japan Kk 魚類用抗菌剤
DE3631906A1 (de) * 1986-09-19 1988-03-31 Bayer Ag Verfahren zur herstellung von benzoesaeure-derivaten
DE3637156C2 (de) * 1986-10-31 1995-12-21 Hoechst Ag Verfahren zur Herstellung von Fluorbenzaldehyden
US5227531A (en) * 1986-10-31 1993-07-13 Hoechst Aktiengesellschaft Process for the preparation of fluorobenzaldehydes
US4831190A (en) * 1986-12-04 1989-05-16 Ube Industries, Ltd. Trifluorohydroxyaromatic acid and preparation thereof
ES2074047T3 (es) * 1987-08-14 1995-09-01 Asahi Glass Co Ltd Compuestos de benzoilo fluorados.
JPH072679B2 (ja) * 1988-04-15 1995-01-18 旭硝子株式会社 ２―クロロ―４，５―ジフルオロ安息香酸誘導体
US4996355A (en) * 1989-04-14 1991-02-26 Mallinckrodt, Inc. Novel intermediates for the production of 2,4,5-trifluorobenzoyl fluoride
IE72169B1 (en) * 1989-11-17 1997-03-26 Asahi Glass Co Ltd Processes for producing 5-fluorobenzoic acids and their intermediates
US4935541A (en) * 1989-11-20 1990-06-19 Occidental Chemical Corporation Preparation of 2,4,5-trifluorobenzoic acid by decarboxylation of 3,4,6-trifluorophthalic anhydride
DE4301247A1 (de) * 1993-01-19 1994-07-21 Bayer Ag Verfahren zur Herstellung mehrfach halogenierter Benzotrichloride und Benzoylchloride sowie neue Trihalogenbenzotrichloride und -benzoylchloride
DE4338525A1 (de) * 1993-11-11 1995-05-18 Bayer Ag Verfahren zur Herstellung von 4,5-Difluorbenzaldehyden
DE4409578A1 (de) * 1994-03-21 1995-09-28 Bayer Ag Verfahren zur Herstellung von 2-Halogen-4,5-difluorbenzoylfluoriden
DE4416329A1 (de) * 1994-05-09 1995-11-16 Hoechst Ag Substituierte 2-Chlor-3,4,5-trifluorbenzole und ein Verfahren zu ihrer Herstellung
US5639888A (en) * 1994-10-03 1997-06-17 American Cyanamid Co. Process for the preparation of acid chloride compounds
DE19627411A1 (de) * 1996-07-09 1998-01-15 Bayer Ag Verfahren zur Decarboxylierung halogenierter aromatischer Carbonsäuren
DE19740632A1 (de) * 1997-09-16 1999-03-18 Bayer Ag Verfahren zur Herstellung von 2,3,4,5-Tetrafluorbenzolderivaten
JP2000086583A (ja) * 1998-09-17 2000-03-28 Asahi Glass Co Ltd 含フッ素ベンジル誘導体の製造方法
JP4200704B2 (ja) * 2002-07-24 2008-12-24 昭和電工株式会社 フッ素化ベンゾニトリルの製造方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB977963A (en) * 1960-05-12 1964-12-16 Imp Smelting Corp Ltd Derivatives of carboxylic acids containing the pentafluorophenyl group
US3230268A (en) * 1962-04-09 1966-01-18 Fuso Chemical Co Ltd Preparation of chloro-substituted benzene derivatives
NL129620C (cg-RX-API-DMAC7.html) * 1963-04-01
US3485865A (en) * 1967-04-05 1969-12-23 Velsicol Chemical Corp N-methoxy and n-ethoxy benzamides
US3816526A (en) * 1972-10-03 1974-06-11 Mobil Oil Corp Method for producing halobenzoyl halides
DE3142856A1 (de) * 1981-10-29 1983-05-11 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von 2,4-dichlor-5-fluor-benzoylchlorid
US4582948A (en) * 1982-02-09 1986-04-15 Occidental Chemical Corporation 3-chloro-4-fluoro-5-nitrobenzotrifluoride
JPS58150543A (ja) * 1982-03-04 1983-09-07 Chisso Corp ２，４，５−トリフルオロ安息香酸トランス−４−（トランス−４′−アルキルシクロヘキシル）シクロヘキシルエステル
JPS6072885A (ja) * 1983-09-28 1985-04-24 Dai Ichi Seiyaku Co Ltd トリフルオロベンゾイル化合物類
EP0160284B1 (en) * 1984-04-26 1990-10-24 Abbott Laboratories Quino-benoxazine antibacterial compounds
US4792618A (en) * 1984-05-02 1988-12-20 Occidental Chemical Corporation Fluorinated carbocylic compounds
US4791225A (en) * 1986-01-20 1988-12-13 Kyorin Pharmaceutical Co., Ltd. Halogenobenzoic acid derivatives and their preparation

Also Published As

Publication number Publication date
KR860000240A (ko) 1986-01-27
CA1242742A (en) 1988-10-04
JPS617220A (ja) 1986-01-13
ATE37866T1 (de) 1988-10-15
US5072038A (en) 1991-12-10
JPH0246015B2 (cg-RX-API-DMAC7.html) 1990-10-12
EP0164619A1 (de) 1985-12-18
DE3420796A1 (de) 1985-12-05
HUT38297A (en) 1986-05-28
EP0164619B1 (de) 1988-10-12
DE3565528D1 (en) 1988-11-17
HU195176B (en) 1988-04-28

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