KR890008122A - 1,5-벤조티아제핀 유도체의 제조방법 - Google Patents
1,5-벤조티아제핀 유도체의 제조방법 Download PDFInfo
- Publication number
- KR890008122A KR890008122A KR1019880014917A KR880014917A KR890008122A KR 890008122 A KR890008122 A KR 890008122A KR 1019880014917 A KR1019880014917 A KR 1019880014917A KR 880014917 A KR880014917 A KR 880014917A KR 890008122 A KR890008122 A KR 890008122A
- Authority
- KR
- South Korea
- Prior art keywords
- lower alkyl
- derivative
- compound
- cyclized
- benzothiazepine derivative
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
- KJFRSZASZNLCDF-UHFFFAOYSA-N 1,5-benzothiazepine Chemical class S1C=CC=NC2=CC=CC=C12 KJFRSZASZNLCDF-UHFFFAOYSA-N 0.000 title claims 4
- -1 II Chemical class 0.000 claims 7
- 239000002253 acid Substances 0.000 claims 5
- XBDQKXXYIPTUBI-UHFFFAOYSA-N dimethylselenoniopropionate Natural products CCC(O)=O XBDQKXXYIPTUBI-UHFFFAOYSA-N 0.000 claims 4
- 125000000217 alkyl group Chemical group 0.000 claims 3
- 125000005907 alkyl ester group Chemical group 0.000 claims 2
- 150000008064 anhydrides Chemical class 0.000 claims 2
- 150000001875 compounds Chemical class 0.000 claims 2
- 150000002148 esters Chemical class 0.000 claims 2
- 150000004820 halides Chemical class 0.000 claims 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 claims 2
- 235000019260 propionic acid Nutrition 0.000 claims 2
- 150000003839 salts Chemical class 0.000 claims 2
- 125000004172 4-methoxyphenyl group Chemical group [H]C1=C([H])C(OC([H])([H])[H])=C([H])C([H])=C1* 0.000 claims 1
- WYWKPNIAGOEYTD-UHFFFAOYSA-N 8-chloro-3,5-dihydro-2h-1,5-benzothiazepin-4-one Chemical compound N1C(=O)CCSC2=CC(Cl)=CC=C21 WYWKPNIAGOEYTD-UHFFFAOYSA-N 0.000 claims 1
- FVGKAJGOHWOXLU-UHFFFAOYSA-N [5-[2-(dimethylamino)ethyl]-8-methyl-2-(4-methylphenyl)-4-oxo-2,3-dihydro-1,5-benzothiazepin-3-yl] acetate Chemical group CC(=O)OC1C(=O)N(CCN(C)C)C2=CC=C(C)C=C2SC1C1=CC=C(C)C=C1 FVGKAJGOHWOXLU-UHFFFAOYSA-N 0.000 claims 1
- 125000002252 acyl group Chemical group 0.000 claims 1
- 125000003545 alkoxy group Chemical group 0.000 claims 1
- 125000002147 dimethylamino group Chemical group [H]C([H])([H])N(*)C([H])([H])[H] 0.000 claims 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 1
- 125000005843 halogen group Chemical group 0.000 claims 1
- 150000005599 propionic acid derivatives Chemical class 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D281/02—Seven-membered rings
- C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
- C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP62-287943 | 1987-11-13 | ||
| JP62287943A JPH01128974A (ja) | 1987-11-13 | 1987-11-13 | １，５−ベンゾチアゼピン誘導体の製法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR890008122A true KR890008122A (ko) | 1989-07-08 |
Family
ID=17723745
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019880014917A Ceased KR890008122A (ko) | 1987-11-13 | 1988-11-12 | 1,5-벤조티아제핀 유도체의 제조방법 |
Country Status (8)
| Country | Link |
|---|---|
| JP (1) | JPH01128974A (enrdf_load_stackoverflow) |
| KR (1) | KR890008122A (enrdf_load_stackoverflow) |
| DK (1) | DK631888A (enrdf_load_stackoverflow) |
| FI (1) | FI92393C (enrdf_load_stackoverflow) |
| FR (1) | FR2623192A1 (enrdf_load_stackoverflow) |
| IE (1) | IE61196B1 (enrdf_load_stackoverflow) |
| IL (1) | IL88296A (enrdf_load_stackoverflow) |
| IT (1) | IT1230633B (enrdf_load_stackoverflow) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5057513A (en) * | 1989-05-25 | 1991-10-15 | Fujisawa Pharmaceutical Co., Ltd. | Spiro-thiazepine derivatives useful as paf antagonists |
| ZA94284B (en) * | 1993-01-27 | 1994-08-17 | Shionogi & Co | Process for preparing benzothiazepine derivatives |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS58201773A (ja) * | 1982-05-17 | 1983-11-24 | Tokawa Tetsuo | ベンゾチアゼピン誘導体の製造法 |
| GB8315364D0 (en) * | 1983-06-03 | 1983-07-06 | Tanabe Seiyaku Co | 8-chloro-1 5-benzothiazepine derivatives |
| JPS60109580A (ja) * | 1983-11-16 | 1985-06-15 | Roller Japan Kk | シス−ｄ−２−（４’−メトキシフェニル）−３−アセトキシ−５−（２−ジメチルアミノエチル）−２，３−ジヒドロ−１，５−ベンゾチアゼピン−４（５Ｈ）−オンまたはその塩の製法 |
| JPS60146884A (ja) * | 1984-01-09 | 1985-08-02 | Nippon Chem:Kk | １，５ベンゾチアゼピン誘導体の製造法 |
| GB8406318D0 (en) * | 1984-03-10 | 1984-04-11 | Tanabe Seiyaku Co | 1 5-benzothiazepine derivatives |
| JPS61103877A (ja) * | 1984-10-24 | 1986-05-22 | Tanabe Seiyaku Co Ltd | ベンゾチアゼピン誘導体及びその製法 |
| GB2167063A (en) * | 1984-11-17 | 1986-05-21 | Tanabe Seiyaku Co | 6 or 9-chloro-1, 5-benzothiazepine derivatives |
-
1987
- 1987-11-13 JP JP62287943A patent/JPH01128974A/ja active Pending
-
1988
- 1988-11-01 FI FI885033A patent/FI92393C/fi not_active IP Right Cessation
- 1988-11-04 IL IL8829688A patent/IL88296A/en not_active IP Right Cessation
- 1988-11-08 FR FR8814577A patent/FR2623192A1/fr active Granted
- 1988-11-11 DK DK631888A patent/DK631888A/da not_active Application Discontinuation
- 1988-11-11 IT IT8822602A patent/IT1230633B/it active
- 1988-11-11 IE IE338788A patent/IE61196B1/en not_active IP Right Cessation
- 1988-11-12 KR KR1019880014917A patent/KR890008122A/ko not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| JPH01128974A (ja) | 1989-05-22 |
| DK631888D0 (da) | 1988-11-11 |
| FR2623192A1 (fr) | 1989-05-19 |
| IL88296A0 (en) | 1989-06-30 |
| FI92393C (fi) | 1994-11-10 |
| IT1230633B (it) | 1991-10-28 |
| IE883387L (en) | 1989-05-13 |
| FI885033A7 (fi) | 1989-05-14 |
| FR2623192B1 (enrdf_load_stackoverflow) | 1994-07-13 |
| DK631888A (da) | 1989-05-14 |
| FI885033A0 (fi) | 1988-11-01 |
| IE61196B1 (en) | 1994-10-19 |
| FI92393B (fi) | 1994-07-29 |
| IT8822602A0 (it) | 1988-11-11 |
| IL88296A (en) | 1995-03-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0109 | Patent application |
Patent event code: PA01091R01D Comment text: Patent Application Patent event date: 19881112 |
|
| PG1501 | Laying open of application | ||
| A201 | Request for examination | ||
| PA0201 | Request for examination |
Patent event code: PA02012R01D Patent event date: 19911115 Comment text: Request for Examination of Application Patent event code: PA02011R01I Patent event date: 19881112 Comment text: Patent Application |
|
| E902 | Notification of reason for refusal | ||
| PE0902 | Notice of grounds for rejection |
Comment text: Notification of reason for refusal Patent event date: 19940325 Patent event code: PE09021S01D |
|
| E601 | Decision to refuse application | ||
| PE0601 | Decision on rejection of patent |
Patent event date: 19940829 Comment text: Decision to Refuse Application Patent event code: PE06012S01D Patent event date: 19940325 Comment text: Notification of reason for refusal Patent event code: PE06011S01I |