KR890000215B1 - 1, 2-벤즈이소티아졸 피페리딘 및 그의 제조방법 - Google Patents

1, 2-벤즈이소티아졸 피페리딘 및 그의 제조방법 Download PDF

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Publication number
KR890000215B1
KR890000215B1 KR1019850002693A KR850002693A KR890000215B1 KR 890000215 B1 KR890000215 B1 KR 890000215B1 KR 1019850002693 A KR1019850002693 A KR 1019850002693A KR 850002693 A KR850002693 A KR 850002693A KR 890000215 B1 KR890000215 B1 KR 890000215B1
Authority
KR
South Korea
Prior art keywords
compound
lower alkyl
formula
acid
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019850002693A
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English (en)
Korean (ko)
Other versions
KR850007262A (ko
Inventor
티.스트루프쩨브스키 죠셉
Original Assignee
훽스트-러셀 파마슈티칼스 인코포레이티드
마크 이.로가르트
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 훽스트-러셀 파마슈티칼스 인코포레이티드, 마크 이.로가르트 filed Critical 훽스트-러셀 파마슈티칼스 인코포레이티드
Publication of KR850007262A publication Critical patent/KR850007262A/ko
Application granted granted Critical
Publication of KR890000215B1 publication Critical patent/KR890000215B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1019850002693A 1984-04-23 1985-04-22 1, 2-벤즈이소티아졸 피페리딘 및 그의 제조방법 Expired KR890000215B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US06/603,264 US4528292A (en) 1984-04-23 1984-04-23 Antihypertensive 1,2-benzisothiazole piperidines
US603264 1984-04-23
US603,264 1984-04-23

Publications (2)

Publication Number Publication Date
KR850007262A KR850007262A (ko) 1985-12-02
KR890000215B1 true KR890000215B1 (ko) 1989-03-10

Family

ID=24414698

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019850002693A Expired KR890000215B1 (ko) 1984-04-23 1985-04-22 1, 2-벤즈이소티아졸 피페리딘 및 그의 제조방법

Country Status (17)

Country Link
US (1) US4528292A (https=)
EP (1) EP0159666B1 (https=)
JP (1) JPS60233073A (https=)
KR (1) KR890000215B1 (https=)
AT (1) ATE44031T1 (https=)
AU (1) AU581217B2 (https=)
DE (1) DE3571031D1 (https=)
DK (1) DK180185A (https=)
ES (2) ES8608515A1 (https=)
FI (1) FI80692C (https=)
GR (1) GR850963B (https=)
IL (1) IL74981A (https=)
NO (1) NO158421C (https=)
NZ (1) NZ211865A (https=)
PH (1) PH23312A (https=)
PT (1) PT80308B (https=)
ZA (1) ZA852984B (https=)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4355037A (en) * 1981-11-12 1982-10-19 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidyl)-1,2-benzisoxales
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4458076A (en) * 1983-05-31 1984-07-03 Hoechst-Roussel Pharmaceuticals 3-(4-Piperidinyl)-1,2-benzisothiazoles

Also Published As

Publication number Publication date
EP0159666B1 (en) 1989-06-14
AU4163385A (en) 1985-10-31
FI80692C (fi) 1990-07-10
PH23312A (en) 1989-06-30
IL74981A0 (en) 1985-08-30
ES542442A0 (es) 1986-06-16
FI851565L (fi) 1985-10-24
ES8608515A1 (es) 1986-06-16
EP0159666A3 (en) 1987-01-14
DK180185A (da) 1985-10-24
US4528292A (en) 1985-07-09
ATE44031T1 (de) 1989-06-15
NO158421B (no) 1988-05-30
GR850963B (https=) 1985-11-25
DK180185D0 (da) 1985-04-22
PT80308B (en) 1987-02-10
DE3571031D1 (en) 1989-07-20
FI80692B (fi) 1990-03-30
ES8704941A1 (es) 1987-04-16
FI851565A0 (fi) 1985-04-19
NO158421C (no) 1988-09-07
EP0159666A2 (en) 1985-10-30
IL74981A (en) 1990-01-18
ES551323A0 (es) 1987-04-16
KR850007262A (ko) 1985-12-02
NO851606L (no) 1985-10-24
JPS60233073A (ja) 1985-11-19
PT80308A (en) 1985-05-01
AU581217B2 (en) 1989-02-16
NZ211865A (en) 1989-01-06
ZA852984B (en) 1986-01-29

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