KR860008965A - 1,3-프로판디온 유도체를 제조하는 방법 - Google Patents

1,3-프로판디온 유도체를 제조하는 방법 Download PDF

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KR860008965A
KR860008965A KR1019860003922A KR860003922A KR860008965A KR 860008965 A KR860008965 A KR 860008965A KR 1019860003922 A KR1019860003922 A KR 1019860003922A KR 860003922 A KR860003922 A KR 860003922A KR 860008965 A KR860008965 A KR 860008965A
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formula
compound
prepared
propanedione
sodium salt
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KR900001022B1 (ko
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죠셉 보이스베뉴 루돌프
딘 크루스 개리
에드워드 크래머 케네드
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일라이 릴리 앤드 캄파니
메리 앤 터커
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/42—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms with nitro or nitroso radicals directly attached to ring carbon atoms
    • C07D333/44—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms with nitro or nitroso radicals directly attached to ring carbon atoms attached in position 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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    • C07C49/04—Saturated compounds containing keto groups bound to acyclic carbon atoms
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
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    • A01N35/04—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having two bonds to hetero atoms with at the most one bond to halogen, e.g. aldehyde radical containing aldehyde or keto groups, or thio analogues thereof, directly attached to an aromatic ring system, e.g. acetophenone; Derivatives thereof, e.g. acetals
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
    • A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
    • A01N43/06—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings
    • A01N43/10—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom five-membered rings with sulfur as the ring hetero atom
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    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/673—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by change of size of the carbon skeleton
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    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
    • C07C49/813—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen polycyclic
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
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    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/82—Ketones containing a keto group bound to a six-membered aromatic ring containing hydroxy groups
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/42—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms with nitro or nitroso radicals directly attached to ring carbon atoms

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
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Abstract

내용 없음

Description

1,3-프로판디온 유도체를 제조하는 방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (7)

  1. 일반식(Ⅱ)의 화합물을 일반식(Ⅱ)의 화합물의 음이온을 생성하기에 충분히 강한 염기의 존재하에 일반식(Ⅲ)의 산의 활성화된 형태로 아실화하거나; R-가 C1-C4퍼플루오로-알킬이고, R1이 C3-C6퍼플루오로-사이클로알킬인 일반식(Ⅳ)의 화합물을 가수 분해하여, R1이 C3-C6퍼플루오로사이클로알킬인 일반식(Ⅰ)의 화합물을 생성함을 특징으로하여 일반식(Ⅰ)의 화합물, 또는 이의 나트륨염, 칼륨염 또는 리툼염(단, R이 5-브로모-또는 5-클로로-티엔-2-일이고, R1이 C3-퍼플루오로알킬인 경우, 일반식 (Ⅰ)의 화합물은 나트륨염, 칼륨염 또는 리튬염 형태로서 존재하여야 한다)을 제조하는 방법.
    상기 식에서, R은 할로겐, 트리플루오로메틸, 니트로, 클로로에테닐 또는 브로모에테닐로 치환된 페닐 또는 티에닐이고; R1은 C3-C6퍼플루오로알킬 또는 퍼플루오로사이클로알킬이다.
  2. 제1항에 있어서, R 그룹이 1 또는 2개의 치환체로 치환된 화합물을 제조하는 방법.
  3. 제1항 또는 제2항에 있어서, R이 치환된 페닐이고, R1이 C2퍼플루오로알킬인 일반식(I)의 화합물을 제조하는 방법.
  4. 제2항에 있어서, 1-퍼플루오로프로필-3-(3-트리플루오로메틸페닐)-1,3-프로판디온 또는 이의 나트륨염을 제조하는 방법.
  5. 제2항에 있어서, 1-퍼플루오로프로필-3-(4-트리플루오로메틸페닐)-1,3-프로판디온 또는 이의 나트륨염을 제조하는 방법.
  6. 제2항에 있어서, 1-퍼플루오로프로필-3-(2,4-디플루오로페닐)-1,3-프로판디온 또는 이의 나트륨염을 제조하는 방법.
  7. 제2항에 있어서, 1-퍼플루오로프로필-3-[3,5-비스(트리플루오로메틸)페닐]-1,3-프로판디온 또는 이의 나트륨염을 제조하는 방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019860003922A 1985-05-20 1986-05-20 1, 3-프로판디온 유도체 KR900001022B1 (ko)

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US73617785A 1985-05-20 1985-05-20
US736177 1985-05-20

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KR860008965A true KR860008965A (ko) 1986-12-19
KR900001022B1 KR900001022B1 (ko) 1990-02-24

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KR1019860003922A KR900001022B1 (ko) 1985-05-20 1986-05-20 1, 3-프로판디온 유도체

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EP (1) EP0202903A3 (ko)
JP (1) JPS61271244A (ko)
KR (1) KR900001022B1 (ko)
AU (1) AU5753786A (ko)
DK (1) DK233386A (ko)
ES (1) ES8707706A1 (ko)
GR (1) GR861301B (ko)
HU (1) HU202469B (ko)
NZ (1) NZ216225A (ko)
PT (1) PT82611B (ko)
SU (1) SU1535381A3 (ko)
ZA (1) ZA863712B (ko)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5618547A (en) * 1985-05-20 1997-04-08 British Technology Group Limited Control of ectoparasites
US4870109A (en) * 1985-05-20 1989-09-26 Eli Lilly And Company Control of ectoparasites
US5281571A (en) * 1990-10-18 1994-01-25 Monsanto Company Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3362935A (en) * 1965-09-03 1968-01-09 Dow Chemical Co Vinylphenyl-perfluoroalkyl-propane-diones and polymers derived therefrom
US3636214A (en) * 1969-07-03 1972-01-18 Grace W R & Co Certain substituted 1 3 diketones as soil fungicides
ZA714221B (en) * 1970-07-10 1972-03-29 Astra Ab Insecticides
US3700416A (en) * 1970-09-04 1972-10-24 Kerr Mc Gee Chem Corp Extraction of vanadium and copper with fluorinated beta-diketones
US3647712A (en) * 1970-09-04 1972-03-07 Kerr Mc Gee Chem Corp Mixture of alcohols and fluorinated beta-diketones useful as extractant in recovery of vanadium

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AU5753786A (en) 1986-11-27
HUT45959A (en) 1988-09-28
PT82611B (en) 1988-04-22
GR861301B (en) 1986-09-16
HU202469B (en) 1991-03-28
NZ216225A (en) 1989-08-29
ZA863712B (en) 1987-12-30
EP0202903A2 (en) 1986-11-26
DK233386D0 (da) 1986-05-20
ES555109A0 (es) 1987-08-16
DK233386A (da) 1986-11-21
ES8707706A1 (es) 1987-08-16
KR900001022B1 (ko) 1990-02-24
JPS61271244A (ja) 1986-12-01
SU1535381A3 (ru) 1990-01-07
PT82611A (en) 1986-06-01
EP0202903A3 (en) 1987-07-01

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