KR860001075A - 피리다지닐우레아 화합물의 제조방법 - Google Patents

피리다지닐우레아 화합물의 제조방법 Download PDF

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Publication number
KR860001075A
KR860001075A KR1019850005085A KR850005085A KR860001075A KR 860001075 A KR860001075 A KR 860001075A KR 1019850005085 A KR1019850005085 A KR 1019850005085A KR 850005085 A KR850005085 A KR 850005085A KR 860001075 A KR860001075 A KR 860001075A
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KR
South Korea
Prior art keywords
alkyl
alkoxy
formula
compound
alkenyl
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KR1019850005085A
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English (en)
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파잘 압둘라 리아즈 (외 1)
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메어리 엔 덕커
일라이 릴리 앤드 캄파니
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Publication of KR860001075A publication Critical patent/KR860001075A/ko

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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/36—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< directly attached to at least one heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/22—Nitrogen and oxygen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

내용 없음

Description

피리다지닐우레아 화합물의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (6)

  1. (A) 구조식 :
    의 카바메이트를 구조식 HNR3R4의 아민과 반응시키거나;
    (B) 구조식 :
    의 아미노피리다진을 구조식 R4NCO의 이소시아네이트와 반응시키거나, 또는 구조식 R3R4NCOCl의 카바모일 클로라이드와 반응시키거나;
    (C)구조식 :
    의 화합물을 구조식 NHR3R4의 아민과 반응시켜서 구조식(Ⅱ)의 화합물을 제조하는 방법.
    상기 식에서, R1은 할로, 트리플루오로메틸, C1―C8알킬, C3―C6사이클로 알킬, (C1―C3알킬), C3―C6사이클로알킬, (C1―C3알콕시) C1―C8알킬, 아다만틸, 페녹시,페닐 또는 할로치환 된 페닐이고, R2는 수소, C1―C6알킬 또는 C2―C8알케닐이고, R3및 R4는 독립적으로 C1―C6알킬, C1―C6알콕시, C2―C6알케닐(C1―C6알콕시), C1―C6알킬, 디(C1―C4알콕시) C1―C6알킬, (하이드록시) C1―C6알킬, 페닐, 벤질, (카복시)C1―C6알킬 또는 (C1―C6아실옥시)C1―C6알킬이거나, 또는 R3및 R4가 질소와 함께 결합하여 피페리진, 모르폴린 또는 피롤리딘 기를 형성하며; m은 1―3의 정수이다. 단, R3및 R4중의 적어도 1개는 C1―C6알킬이다.
  2. 제1항에서, R1는 할로 또는 C1―C4알킬이고, R2는 수소이고; R3및 R4는 독립적으로 C1―C3알킬, C1―C3알콕시, C2―C4알케닐, 하이드록시(C1―C4알킬) 또는 (C1―C6아실옥시) C1―C6알킬이고; m은 1 또는 2인 구조식(Ⅱ)의 화합물을 제조하는 방법.
  3. 제1항에서, N´―〔6―클로로―5―(1,1―디메틸에틸)―3―피리다지닐〕―N―메톡시―N―메틸우레아를 제조하는 방법.
  4. 제1항에서, N―〔2―(아세틸옥시)에틸)―N´―〔6―클로로―5―(1,1―디메틸에틸)―3―피리다지닐〕―N―메틸우레아를 제조하는 방법.
  5. 제1항에서, N´―〔6―클로로―5―(1,1―디메틸에틸)―3―피리다지닐〕―N―(2―하이드록시에틸)―N―메틸우레아를 제조하는 방법.
  6. 식물 또는 식물이 자라는 토양을 구조식(Ⅱ) 화합물의 제조유효량으로 처리해서 원하지 않는 식물의 성장을 억제하는 방법.
    상기식에서, R1은 할로, 트리플루오로메틸, C1―C8알킬, C3―C6사이클로알킬, (C1―C3알킬) C3―C6사이클로알킬, (C1―C3알콕시) C1―C8알킬, 아다만틸, 페녹시, 페닐 또는 할로치환된 페닐이고, R2는 수소, C1―C6알킬 또는 C2―C6알케닐이고; R3및 R4는 독립적으로 수소, C1―C6알킬, C1―C6알콕시, C2―C6알케닐, (C1―C6알콕시) C1―C6알킬, 디(C1―C4알콕시) C1―C6알킬, (하이드록시) C1―C6알킬페닐, 벤질, (카복시) C1―C6알킬 또는 (C1―C6아실옥시) C1―C6알킬이거나; 또는 R3및 R4는 질소원자와 함께 5 또는 6개 원자로 구성된 복소환을 형성하며; m은 0―3의 정수이다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019850005085A 1984-07-17 1985-07-16 피리다지닐우레아 화합물의 제조방법 KR860001075A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US631651 1984-07-17
US06/631,651 US4619686A (en) 1984-07-17 1984-07-17 Pyridazinylurea compounds and methods of use as herbicides

Publications (1)

Publication Number Publication Date
KR860001075A true KR860001075A (ko) 1986-02-22

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KR1019850005085A KR860001075A (ko) 1984-07-17 1985-07-16 피리다지닐우레아 화합물의 제조방법

Country Status (6)

Country Link
US (1) US4619686A (ko)
EP (1) EP0169051A3 (ko)
JP (1) JPS6136271A (ko)
KR (1) KR860001075A (ko)
BR (1) BR8503377A (ko)
IL (1) IL75803A0 (ko)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4735650A (en) * 1985-10-10 1988-04-05 Fmc Corporation Pyridazinylurea N-oxide plant regulators
US4728355A (en) * 1985-10-10 1988-03-01 Fmc Corporation Pyridazinylurea plant regulators
WO2000034267A1 (fr) * 1998-12-04 2000-06-15 Takeda Chemical Industries, Ltd. Procede de production d'un compose d'amide cyclique
TWI372050B (en) 2003-07-03 2012-09-11 Astex Therapeutics Ltd (morpholin-4-ylmethyl-1h-benzimidazol-2-yl)-1h-pyrazoles
MX2007008008A (es) 2004-12-30 2007-11-12 Astex Therapeutics Ltd Compuestos de pirazol que modulan la actividad de las cinasas cdk, gsk y aurora.
US7947006B2 (en) 2005-11-30 2011-05-24 Smith & Nephew, Inc. Hip distraction
US8399442B2 (en) 2005-12-30 2013-03-19 Astex Therapeutics Limited Pharmaceutical compounds
EP2049119A2 (en) 2006-06-29 2009-04-22 Astex Therapeutics Limited Pharmaceutical combinations of 1-cyclopropyl-3-[3-(5-morphoolin-4-ylmethyl-1h-benzoimidazol-2-yl)-1h-1-pyrazol-4-yl]-urea

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1122662A (en) * 1965-02-18 1968-08-07 Fisons Pest Control Ltd Preservation of plant materials
US4093444A (en) * 1973-05-22 1978-06-06 Pepro, Societe Pour Le Developpement Et La Vente De Specialites Chimiques Hydantoin derivatives and methods for regulating plant-growth
US3947437A (en) * 1974-01-22 1976-03-30 The Dow Chemical Company Substituted pyridazinyloxy(thio)phenyl ureas and derivatives thereof
US4144338A (en) * 1977-02-17 1979-03-13 Merck & Co., Inc. N-pyrimidinyl-N-dialkylaminoalkyl ureas
JPS55160768A (en) * 1979-05-31 1980-12-13 Toshihiko Okamoto Plant growth regulating substance
EP0052668B1 (en) * 1980-11-25 1984-03-14 Koichi Prof. Dr. Shudo N-(4-pyridazinyl)-n'-phenylureas and -thioureas as well as plant growth regulators containing same
JPS5877866A (ja) * 1981-11-04 1983-05-11 Mitsui Toatsu Chem Inc アミノピリダジン誘導体および除草剤

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Publication number Publication date
EP0169051A3 (en) 1986-12-10
JPS6136271A (ja) 1986-02-20
EP0169051A2 (en) 1986-01-22
BR8503377A (pt) 1986-04-08
IL75803A0 (en) 1985-11-29
US4619686A (en) 1986-10-28

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