KR850002261A - 디페닐-메틸렌-에틸아민 유도체의 제조방법 - Google Patents

디페닐-메틸렌-에틸아민 유도체의 제조방법 Download PDF

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KR850002261A
KR850002261A KR1019840004560A KR840004560A KR850002261A KR 850002261 A KR850002261 A KR 850002261A KR 1019840004560 A KR1019840004560 A KR 1019840004560A KR 840004560 A KR840004560 A KR 840004560A KR 850002261 A KR850002261 A KR 850002261A
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pyridinemethyl
formula
carbon atoms
methylene
pyridyl
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KR1019840004560A
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KR900007198B1 (ko
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디. 시레라 자비에르
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로메오 알. 안드 레올리
소시에다드 에스파놀라드 에스페시아리다데스 파마코-테라퓨티카스, 에스. 에이
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Abstract

내용 없음

Description

디페닐－메틸렌－에틸아민 유도체의 제조방법
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (1)

  1. 하익 일반식(Ⅱ)의 아민과 하기 일반식(Ⅲ)의 할로겐 유도체와 반응시킴을 특징으로 하는 하기 구조식(Ⅰ)의 디페닐－메틸렌－에틸아민에서 유도된 신규의 화합물과 이들의 약리학적 염의 제조방법.
    식중에서, R1:H－ 또는 F－R2:H－;CH3－;CH2COCH2COOH;CH2NHCONH2
    R3:N－또는 CH3－ R4:H－;C6H5－;HO－C8H4－X:－H H－;－CH2－CH2－;－CH＝CH－ Y:＝H2
    R6:CH3－;CH3CH2－ 또는 4 탄소 원자까지의 알킬기 R7:CH3－;CH3－CH＝C(★스캔) 또는 4 탄소원자까지의 알칼기 R2Z(피페라진 고리형성) ::수소, 4 탄소원자까지의 알킬기, 알릴, 2－히드록시메틸, 카르브에톡시메틸, 카르복시메틸, 3－카르보메톡시알릴, N－피롤리디노카르보닐메틸, 1－아다만틸, 2－피리딜, 4－피리딜, 젠질, 신나밀, 펜아실, 3－벤조일알릴, 2－큼로로벤질, 피페로닐, 2－피리딘메틸, 3－피리딘메틸, 4－피리딘메틸, 2－푸르푸릴, 2－테닐, 2－(N－메틸피롤릴)메틸, 3－피페리딘메틸, 3－카르보메톡시－4－히드록시벤질, N－모노폴리노메틸 우레아카르보닐메틸.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019840004560A 1983-08-02 1984-07-31 디페닐-메틸렌-에틸아민 유도체의 제조방법 KR900007198B1 (ko)

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ES524680A ES8502099A1 (es) 1983-08-02 1983-08-02 Procedimiento de obtencion de nuevos compuestos derivados de la difenil-metilen-etilamina.
ES524680 1983-08-02
ES524.680 1983-08-02

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US4882351A (en) * 1987-10-14 1989-11-21 Roussel Uclaf Tricyclic compounds
IT1222986B (it) * 1987-10-23 1990-09-12 Texcontor Ets Derivati dell'efedrina esterificata aventi attivita' antiulcera prolungata nel tempo
EP0581767B1 (en) * 1990-05-18 1997-09-03 Merrell Pharmaceuticals Inc. 5H-DIBENZO(a,d)CYCLOHEPTENES AS MUSCARINIC RECEPTOR ANTAGONISTS
US5508280A (en) * 1990-05-18 1996-04-16 Merrell Pharmaceuticals, Inc. 5H-Dibenzo (A,D) cycloheptenes as muscarinic receptor antagonists
JP2574733Y2 (ja) * 1991-09-04 1998-06-18 松下電器産業株式会社 車両用ハーネス案内装置
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US6613905B1 (en) * 1998-01-21 2003-09-02 Millennium Pharmaceuticals, Inc. Chemokine receptor antagonists and methods of use therefor
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GB202205895D0 (en) 2022-04-22 2022-06-08 Atrogi Ab New medical uses

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EP0132764A2 (en) 1985-02-13
US5112826A (en) 1992-05-12
JPH0625091B2 (ja) 1994-04-06
US4835156A (en) 1989-05-30
JPS60126265A (ja) 1985-07-05
ZA845940B (en) 1986-08-27
EP0132764B1 (en) 1991-01-02
KR900007198B1 (ko) 1990-10-05
EP0357956A2 (en) 1990-03-14
EP0132764A3 (en) 1985-12-04
AU580963B2 (en) 1989-02-09
AU3131684A (en) 1985-02-07
EP0357956A3 (en) 1990-08-29
ES524680A0 (es) 1984-12-16
US4835179A (en) 1989-05-30
NZ208691A (en) 1989-06-28
DE3483798D1 (de) 1991-02-07
ES8502099A1 (es) 1984-12-16
CA1243018A (en) 1988-10-11

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