KR850000555B1 - 벤즈아졸 유도체의 제조방법 - Google Patents

벤즈아졸 유도체의 제조방법 Download PDF

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Publication number
KR850000555B1
KR850000555B1 KR1019810001768A KR810001768A KR850000555B1 KR 850000555 B1 KR850000555 B1 KR 850000555B1 KR 1019810001768 A KR1019810001768 A KR 1019810001768A KR 810001768 A KR810001768 A KR 810001768A KR 850000555 B1 KR850000555 B1 KR 850000555B1
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KR
South Korea
Prior art keywords
butyl
group
acid
tert
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
KR1019810001768A
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English (en)
Korean (ko)
Other versions
KR830006231A (ko
Inventor
작퀴스 갈라이 진
쉬베이저 에른스트
Original Assignee
시비-가이기 에이지
아놀드 자일러, 에른스트 알테르
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Publication date
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Publication of KR830006231A publication Critical patent/KR830006231A/ko
Application granted granted Critical
Publication of KR850000555B1 publication Critical patent/KR850000555B1/ko
Expired legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/08—Radicals containing only hydrogen and carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/10—Radicals substituted by halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
KR1019810001768A 1980-05-22 1981-05-21 벤즈아졸 유도체의 제조방법 Expired KR850000555B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH401680 1980-05-22
CH4016/80-7 1980-05-22

Publications (2)

Publication Number Publication Date
KR830006231A KR830006231A (ko) 1983-09-20
KR850000555B1 true KR850000555B1 (ko) 1985-04-26

Family

ID=4268232

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019810001768A Expired KR850000555B1 (ko) 1980-05-22 1981-05-21 벤즈아졸 유도체의 제조방법

Country Status (28)

Country Link
US (1) US4511567A (cg-RX-API-DMAC7.html)
EP (1) EP0041046B1 (cg-RX-API-DMAC7.html)
JP (1) JPS5718670A (cg-RX-API-DMAC7.html)
KR (1) KR850000555B1 (cg-RX-API-DMAC7.html)
AU (1) AU547922B2 (cg-RX-API-DMAC7.html)
CY (1) CY1339A (cg-RX-API-DMAC7.html)
DD (1) DD159073A5 (cg-RX-API-DMAC7.html)
DE (1) DE3176402D1 (cg-RX-API-DMAC7.html)
DK (1) DK164786C (cg-RX-API-DMAC7.html)
ES (3) ES8300724A1 (cg-RX-API-DMAC7.html)
FI (1) FI75564C (cg-RX-API-DMAC7.html)
GB (1) GB2076399B (cg-RX-API-DMAC7.html)
GR (1) GR75253B (cg-RX-API-DMAC7.html)
HK (1) HK74686A (cg-RX-API-DMAC7.html)
HU (1) HU186770B (cg-RX-API-DMAC7.html)
IE (1) IE52426B1 (cg-RX-API-DMAC7.html)
IL (1) IL62928A (cg-RX-API-DMAC7.html)
IN (1) IN153293B (cg-RX-API-DMAC7.html)
KE (1) KE3645A (cg-RX-API-DMAC7.html)
MA (1) MA19290A1 (cg-RX-API-DMAC7.html)
MW (1) MW2181A1 (cg-RX-API-DMAC7.html)
MY (1) MY8700141A (cg-RX-API-DMAC7.html)
OA (1) OA06816A (cg-RX-API-DMAC7.html)
PH (1) PH16754A (cg-RX-API-DMAC7.html)
PT (1) PT73066B (cg-RX-API-DMAC7.html)
ZA (1) ZA8103409D (cg-RX-API-DMAC7.html)
ZM (1) ZM4481A1 (cg-RX-API-DMAC7.html)
ZW (1) ZW11981A1 (cg-RX-API-DMAC7.html)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8423697D0 (en) * 1984-09-19 1984-10-24 Ciba Geigy Ag Benzazole derivatives
US5246927A (en) * 1988-08-17 1993-09-21 Ciba-Geigy Corporation Benzazole derivatives, processes for their preparation containing such compounds and the use thereof
WO1992012144A1 (en) * 1990-12-28 1992-07-23 Teijin Limited Condensed benzoxa ring compound, production thereof, and pharmaceutical composition containing the same
WO1997047610A1 (en) * 1996-06-07 1997-12-18 Novartis Ag Benzazole derivatives
US6177572B1 (en) * 1997-08-20 2001-01-23 Sepracor, Inc. Solid and liquid-phase synthesis of benzoxazoles and benzothiazoles and their use
EP3235815A1 (de) * 2016-04-19 2017-10-25 Philipps-Universität Marburg Wirkstoffe gegen parasitäre helminthen

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1087561A (en) * 1963-02-16 1967-10-18 Fisons Pest Control Ltd Fluorinated benzimidazoles and compositions containing them
IE31812B1 (en) * 1967-02-03 1973-01-10 Merck & Co Inc Benzimidazole derivatives
US3646049A (en) * 1970-03-05 1972-02-29 Merck & Co Inc Acylaminobenzimidazole derivatives
US3714180A (en) * 1970-08-12 1973-01-30 Squibb & Sons Inc Sulfonyl benzimidazoles
BE792402A (fr) * 1971-12-07 1973-06-07 Ciba Geigy Composes heterocycliques azotes et medicaments anthelminthiqueset antimicrobiens qui en contiennent

Also Published As

Publication number Publication date
AU7091081A (en) 1981-11-26
CY1339A (en) 1987-01-16
ES513169A0 (es) 1984-07-01
ZM4481A1 (en) 1982-01-21
OA06816A (fr) 1982-12-31
MY8700141A (en) 1987-12-31
GB2076399A (en) 1981-12-02
HU186770B (en) 1985-09-30
FI75564C (fi) 1988-07-11
AU547922B2 (en) 1985-11-14
ZW11981A1 (en) 1981-12-16
PH16754A (en) 1984-02-15
JPS5718670A (en) 1982-01-30
IL62928A (en) 1985-03-31
MW2181A1 (en) 1982-10-13
GB2076399B (en) 1983-11-02
DE3176402D1 (en) 1987-10-08
MA19290A1 (fr) 1982-04-01
FI811531L (fi) 1981-11-23
DK164786B (da) 1992-08-17
PT73066B (en) 1983-02-08
DD159073A5 (de) 1983-02-16
KR830006231A (ko) 1983-09-20
KE3645A (en) 1986-07-11
IN153293B (cg-RX-API-DMAC7.html) 1984-06-30
GR75253B (cg-RX-API-DMAC7.html) 1984-07-13
PT73066A (en) 1981-06-01
ES502355A0 (es) 1982-11-01
DK164786C (da) 1993-01-04
ES8300724A1 (es) 1982-11-01
ES8308316A1 (es) 1983-09-01
EP0041046B1 (de) 1987-09-02
JPH0357099B2 (cg-RX-API-DMAC7.html) 1991-08-30
ES8406452A1 (es) 1984-07-01
IL62928A0 (en) 1981-07-31
DK224381A (da) 1981-11-23
IE811127L (en) 1981-11-22
HK74686A (en) 1986-10-10
IE52426B1 (en) 1987-10-28
ZA8103409D (en) 1982-06-30
EP0041046A1 (de) 1981-12-02
FI75564B (fi) 1988-03-31
US4511567A (en) 1985-04-16
ES513170A0 (es) 1983-09-01

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