KR20210074318A - 이미다졸 유도체의 제조 방법 - Google Patents
이미다졸 유도체의 제조 방법 Download PDFInfo
- Publication number
- KR20210074318A KR20210074318A KR1020217013665A KR20217013665A KR20210074318A KR 20210074318 A KR20210074318 A KR 20210074318A KR 1020217013665 A KR1020217013665 A KR 1020217013665A KR 20217013665 A KR20217013665 A KR 20217013665A KR 20210074318 A KR20210074318 A KR 20210074318A
- Authority
- KR
- South Korea
- Prior art keywords
- alkyl
- cycloalkyl
- alkylamino
- alkoxy
- methyl
- Prior art date
Links
- GZZWUFNRZMEUKY-BRJRFNKRSA-N CC(CN)[C@@H](C)F Chemical compound CC(CN)[C@@H](C)F GZZWUFNRZMEUKY-BRJRFNKRSA-N 0.000 description 1
- PBVRXCCSTPVIML-UHFFFAOYSA-N CCSc([n](C)c(Br)n1)c1I Chemical compound CCSc([n](C)c(Br)n1)c1I PBVRXCCSTPVIML-UHFFFAOYSA-N 0.000 description 1
- 0 CCSc1c(C(N(C)C(C)NN)=NF)nc(*)[n]1C Chemical compound CCSc1c(C(N(C)C(C)NN)=NF)nc(*)[n]1C 0.000 description 1
- VJDLYTOOOXOWBD-UHFFFAOYSA-M C[n]1c([Zn]Cl)nc2c1NNC(C(C(F)(F)F)(F)F)=C2 Chemical compound C[n]1c([Zn]Cl)nc2c1NNC(C(C(F)(F)F)(F)F)=C2 VJDLYTOOOXOWBD-UHFFFAOYSA-M 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP18199885.7 | 2018-10-11 | ||
| EP18199885 | 2018-10-11 | ||
| PCT/EP2019/077304 WO2020074558A1 (fr) | 2018-10-11 | 2019-10-09 | Procédé de préparation de dérivés imidazolés |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20210074318A true KR20210074318A (ko) | 2021-06-21 |
Family
ID=63833924
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020217013665A KR20210074318A (ko) | 2018-10-11 | 2019-10-09 | 이미다졸 유도체의 제조 방법 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20220009930A1 (fr) |
| EP (1) | EP3864015B1 (fr) |
| JP (1) | JP2022512640A (fr) |
| KR (1) | KR20210074318A (fr) |
| CN (1) | CN112867713B (fr) |
| BR (1) | BR112021005723A2 (fr) |
| DK (1) | DK3864015T3 (fr) |
| ES (1) | ES2951539T3 (fr) |
| FI (1) | FI3864015T3 (fr) |
| IL (1) | IL282036B2 (fr) |
| MX (1) | MX2021004081A (fr) |
| TW (1) | TWI820232B (fr) |
| WO (1) | WO2020074558A1 (fr) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2023532548A (ja) | 2020-07-02 | 2023-07-28 | バイエル・アクチエンゲゼルシヤフト | 有害生物防除剤としてのヘテロサイクレン誘導体 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0212048D0 (en) | 2002-05-24 | 2002-07-03 | Merck Sharp & Dohme | Therapeutic agents |
| EP1940829A2 (fr) | 2005-10-14 | 2008-07-09 | NeuroSearch A/S | Derives d'imidazole utilises pour moduler le complexe du recepteur gabaa |
| WO2010083145A1 (fr) | 2009-01-16 | 2010-07-22 | Merck Sharp & Dohme Corp. | Imidazo[1,2-a]pyridines et imidazo[1,2-b]pyridazines utilisés en tant qu'inhibiteurs de la kinase mark |
| WO2013066729A1 (fr) | 2011-10-31 | 2013-05-10 | Merck Sharp & Dohme Corp. | Aminopyrimidinones en tant qu'inhibiteurs de kinases associées au récepteur de l'interleukine |
| CA2895504A1 (fr) | 2012-12-20 | 2014-06-26 | Merck Sharp & Dohme Corp. | Imidazopyridines substituees en tant qu'inhibiteurs de hdm2 |
| US9376441B2 (en) | 2013-07-31 | 2016-06-28 | Gilead Sciences, Inc. | Substituted pyrrolidines as SYK inhibitors |
| KR102420235B1 (ko) * | 2016-08-16 | 2022-07-12 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 3H-이미다졸[4,5-c]피리딘 유도체와 유기금속 아연-아민 염기의 반응에 의한 2-(3,6-디할로피리딘-2-일)-3H-이미다졸[4,5-c]피리딘 유도체 및 관련 화합물의 제조 방법 |
| GB201614314D0 (en) | 2016-08-22 | 2016-10-05 | Discuva Ltd | Antibiotic compounds |
| US11083199B2 (en) | 2017-01-10 | 2021-08-10 | Bayer Aktiengesellschaft | Heterocycle derivatives as pesticides |
| WO2018130437A1 (fr) * | 2017-01-10 | 2018-07-19 | Bayer Aktiengesellschaft | Dérivés hétérocycliques utilisés comme pesticides |
-
2019
- 2019-10-09 FI FIEP19780272.1T patent/FI3864015T3/fi active
- 2019-10-09 JP JP2021519568A patent/JP2022512640A/ja active Pending
- 2019-10-09 KR KR1020217013665A patent/KR20210074318A/ko unknown
- 2019-10-09 EP EP19780272.1A patent/EP3864015B1/fr active Active
- 2019-10-09 DK DK19780272.1T patent/DK3864015T3/da active
- 2019-10-09 BR BR112021005723-4A patent/BR112021005723A2/pt unknown
- 2019-10-09 CN CN201980066392.2A patent/CN112867713B/zh active Active
- 2019-10-09 ES ES19780272T patent/ES2951539T3/es active Active
- 2019-10-09 US US17/283,661 patent/US20220009930A1/en active Pending
- 2019-10-09 IL IL282036A patent/IL282036B2/en unknown
- 2019-10-09 WO PCT/EP2019/077304 patent/WO2020074558A1/fr unknown
- 2019-10-09 MX MX2021004081A patent/MX2021004081A/es unknown
- 2019-10-09 TW TW108136617A patent/TWI820232B/zh active
Also Published As
| Publication number | Publication date |
|---|---|
| DK3864015T3 (da) | 2023-07-31 |
| EP3864015B1 (fr) | 2023-05-10 |
| US20220009930A1 (en) | 2022-01-13 |
| JP2022512640A (ja) | 2022-02-07 |
| BR112021005723A2 (pt) | 2021-06-22 |
| WO2020074558A1 (fr) | 2020-04-16 |
| CN112867713A (zh) | 2021-05-28 |
| TW202028201A (zh) | 2020-08-01 |
| FI3864015T3 (fi) | 2023-07-26 |
| TWI820232B (zh) | 2023-11-01 |
| ES2951539T3 (es) | 2023-10-23 |
| IL282036A (en) | 2021-05-31 |
| EP3864015A1 (fr) | 2021-08-18 |
| MX2021004081A (es) | 2021-06-04 |
| IL282036B1 (en) | 2023-11-01 |
| IL282036B2 (en) | 2024-03-01 |
| CN112867713B (zh) | 2023-05-05 |
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