KR20180107121A - 팬 인테그린 길항제로서의 메타-아자사이클릭 아미노 벤조산 유도체 - Google Patents

팬 인테그린 길항제로서의 메타-아자사이클릭 아미노 벤조산 유도체 Download PDF

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KR20180107121A
KR20180107121A KR1020187021837A KR20187021837A KR20180107121A KR 20180107121 A KR20180107121 A KR 20180107121A KR 1020187021837 A KR1020187021837 A KR 1020187021837A KR 20187021837 A KR20187021837 A KR 20187021837A KR 20180107121 A KR20180107121 A KR 20180107121A
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disease
amino
disorder
compound
hydroxy
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피터 지. 루민스키
데이빗 더블유. 그릭스
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세인트 루이스 유니버시티
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KR1020187021837A 2015-12-30 2016-12-30 팬 인테그린 길항제로서의 메타-아자사이클릭 아미노 벤조산 유도체 Withdrawn KR20180107121A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562273246P 2015-12-30 2015-12-30
US62/273,246 2015-12-30
PCT/US2016/069511 WO2017117538A1 (en) 2015-12-30 2016-12-30 Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists

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KR20180107121A true KR20180107121A (ko) 2018-10-01

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US (3) US10035778B2 (https=)
EP (2) EP3738953A1 (https=)
JP (1) JP2019500355A (https=)
KR (1) KR20180107121A (https=)
CN (1) CN108779077A (https=)
AU (1) AU2016381336A1 (https=)
BR (1) BR112018012981A2 (https=)
CA (1) CA3008023A1 (https=)
CO (1) CO2018007278A2 (https=)
ES (1) ES2806276T3 (https=)
HK (1) HK1244806A1 (https=)
IL (1) IL259951A (https=)
PH (1) PH12018501362A1 (https=)
RU (1) RU2729518C2 (https=)
SG (1) SG11201805387RA (https=)
WO (1) WO2017117538A1 (https=)

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SG11201805387RA (en) * 2015-12-30 2018-07-30 Univ Saint Louis Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists
MX394210B (es) 2017-02-28 2025-03-04 Morphic Therapeutic Inc INHIBIDORES DE INTEGRINA AVß6.
MA52117A (fr) 2017-02-28 2022-04-06 Morphic Therapeutic Inc Inhibiteurs de l'intégrine (alpha-v) (bêta-6)
US11739326B2 (en) * 2017-11-14 2023-08-29 Massachusetts Eye And Ear Infirmary RUNX1 inhibition for treatment of proliferative vitreoretinopathy and conditions associated with epithelial to mesenchymal transition
SI3844162T1 (sl) 2018-08-29 2025-06-30 Morphic Therapeutic, Inc. Zaviralci integrina alfa v beta6
WO2020047239A1 (en) 2018-08-29 2020-03-05 Morphic Therapeutic, Inc. INHIBITING αV β6 INTEGRIN
WO2020047208A1 (en) 2018-08-29 2020-03-05 Morphic Therapeutic, Inc. Inhibitors of (alpha-v)(beta-6) integrin
EP4034236A1 (en) 2019-09-26 2022-08-03 Abionyx Pharma SA Compounds useful for treating liver diseases
US20230060422A1 (en) * 2019-12-20 2023-03-02 Novartis Ag Combination treatment of liver diseases using integrin inhibitors
KR20230011967A (ko) 2020-05-14 2023-01-25 유비이 가부시키가이샤 1,4,5,6-테트라하이드로피리미딘-2-아민 유도체
WO2022189856A1 (en) 2021-03-08 2022-09-15 Abionyx Pharma Sa Compounds useful for treating liver diseases
WO2023085396A1 (ja) 2021-11-12 2023-05-19 Ｕｂｅ株式会社 アルポート症候群を治療または予防するための医薬組成物
EP4733297A1 (en) * 2023-06-22 2026-04-29 Antibody Therapeutics, Inc. Integrin-inhibiting small molecule compound

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US20200199079A1 (en) 2020-06-25
AU2016381336A1 (en) 2018-06-28
US10577330B2 (en) 2020-03-03
CA3008023A1 (en) 2017-07-06
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US20180072684A1 (en) 2018-03-15
US10035778B2 (en) 2018-07-31
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