KR20170139046A - 세미카바자이드-민감성 아민 산화효소(ssao) 효소 억제제로서의 결정질 화합물 - Google Patents
세미카바자이드-민감성 아민 산화효소(ssao) 효소 억제제로서의 결정질 화합물 Download PDFInfo
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- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB1507036.0A GB201507036D0 (en) | 2015-04-24 | 2015-04-24 | Crystalline enzyme inhibitor compound |
| GB1507036.0 | 2015-04-24 | ||
| PCT/GB2016/051120 WO2016170352A1 (en) | 2015-04-24 | 2016-04-22 | Crystalline compound as semicarbazide-sensitive amine oxidase (ssao) enzyme inhibitor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20170139046A true KR20170139046A (ko) | 2017-12-18 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020177032023A Withdrawn KR20170139046A (ko) | 2015-04-24 | 2016-04-22 | 세미카바자이드-민감성 아민 산화효소(ssao) 효소 억제제로서의 결정질 화합물 |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US10369139B2 (enExample) |
| EP (1) | EP3286189B1 (enExample) |
| JP (2) | JP2018513139A (enExample) |
| KR (1) | KR20170139046A (enExample) |
| CN (1) | CN107531701A (enExample) |
| AU (1) | AU2016252236A1 (enExample) |
| BR (1) | BR112017020046A2 (enExample) |
| CA (1) | CA2979157A1 (enExample) |
| EA (1) | EA033064B1 (enExample) |
| GB (1) | GB201507036D0 (enExample) |
| HK (1) | HK1249907A1 (enExample) |
| IL (1) | IL254154A0 (enExample) |
| MX (1) | MX2017013048A (enExample) |
| SG (1) | SG11201707868YA (enExample) |
| WO (1) | WO2016170352A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB201507048D0 (en) * | 2015-04-24 | 2015-06-10 | Proximagen Ltd | Treatment of pain |
| GB201507031D0 (en) | 2015-04-24 | 2015-06-10 | Proximagen Ltd | New pharmaceutical salt forms |
| GB201618029D0 (en) | 2016-10-25 | 2016-12-07 | Proximagen Ltd | New process |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4141899A (en) | 1976-01-07 | 1979-02-27 | Societa' Farmaceutici Italia S.P.A. | 4,5,6,7-Tetrahydroimidazo-[4,5-c]-pyridine derivatives |
| IT1098015B (it) | 1978-08-07 | 1985-08-31 | Farmaceutici Italia | Nuovi 4,5,6,7,-tetraidroimidazo-aperta par.quadrata 4,5-c chiusa par.quadrata-piridin-derivati |
| US6908926B1 (en) | 1999-04-16 | 2005-06-21 | Novo Nordisk A/S | Substituted imidazoles, their preparation and use |
| AU2002214505A1 (en) | 2000-11-09 | 2002-05-21 | Biovitrum Ab | New use of 4, 5, 6, 7-tetrahydroimidazo-(4,5-c)pyridine derivatives |
| SE0004101D0 (sv) | 2000-11-09 | 2000-11-09 | Pharmacia Ab | New use |
| US20070066646A1 (en) | 2005-08-02 | 2007-03-22 | Genmedica Therapeutics Sl | Compounds for Inhibiting Copper-Containing Amine Oxidases and Uses Thereof |
| EP3461499A1 (en) | 2006-06-07 | 2019-04-03 | The Board of Trustees of The Leland Stanford Junior University | Anti-leukocyte recruitment therapy for the treatment of recurrence of epileptic seizures |
| MX2011002581A (es) * | 2008-09-16 | 2011-04-07 | Proximagen Ltd | Compuestos nuevos i. |
| CA2915163A1 (en) | 2013-06-12 | 2014-12-18 | Proximagen Limited | New therapeutic uses of enzyme inhibitors |
| HUE042625T2 (hu) | 2014-04-15 | 2019-07-29 | Pecsi Tudomanyegyetem | Szemikarbazid-szenzitiv amin-oxidáz gátlók fájdalomcsillapítóként való alkalmazásra traumás neuropátiában és neurogén gyulladásban |
| GB201507048D0 (en) * | 2015-04-24 | 2015-06-10 | Proximagen Ltd | Treatment of pain |
| GB201507031D0 (en) * | 2015-04-24 | 2015-06-10 | Proximagen Ltd | New pharmaceutical salt forms |
-
2015
- 2015-04-24 GB GBGB1507036.0A patent/GB201507036D0/en not_active Ceased
-
2016
- 2016-04-22 US US15/567,549 patent/US10369139B2/en not_active Expired - Fee Related
- 2016-04-22 MX MX2017013048A patent/MX2017013048A/es unknown
- 2016-04-22 HK HK18109399.8A patent/HK1249907A1/zh unknown
- 2016-04-22 BR BR112017020046A patent/BR112017020046A2/pt not_active Application Discontinuation
- 2016-04-22 KR KR1020177032023A patent/KR20170139046A/ko not_active Withdrawn
- 2016-04-22 JP JP2017550912A patent/JP2018513139A/ja active Pending
- 2016-04-22 EP EP16718883.8A patent/EP3286189B1/en active Active
- 2016-04-22 EA EA201792122A patent/EA033064B1/ru not_active IP Right Cessation
- 2016-04-22 AU AU2016252236A patent/AU2016252236A1/en not_active Abandoned
- 2016-04-22 CN CN201680023291.3A patent/CN107531701A/zh active Pending
- 2016-04-22 SG SG11201707868YA patent/SG11201707868YA/en unknown
- 2016-04-22 WO PCT/GB2016/051120 patent/WO2016170352A1/en not_active Ceased
- 2016-04-22 CA CA2979157A patent/CA2979157A1/en not_active Abandoned
-
2017
- 2017-08-24 IL IL254154A patent/IL254154A0/en unknown
-
2021
- 2021-01-28 JP JP2021012440A patent/JP2021073259A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| EP3286189A1 (en) | 2018-02-28 |
| JP2021073259A (ja) | 2021-05-13 |
| EA033064B1 (ru) | 2019-08-30 |
| IL254154A0 (en) | 2017-10-31 |
| US20180085357A1 (en) | 2018-03-29 |
| WO2016170352A1 (en) | 2016-10-27 |
| HK1249907A1 (zh) | 2018-11-16 |
| SG11201707868YA (en) | 2017-11-29 |
| CN107531701A (zh) | 2018-01-02 |
| AU2016252236A1 (en) | 2017-10-05 |
| EA201792122A1 (ru) | 2018-03-30 |
| MX2017013048A (es) | 2017-12-08 |
| CA2979157A1 (en) | 2016-10-27 |
| JP2018513139A (ja) | 2018-05-24 |
| US10369139B2 (en) | 2019-08-06 |
| BR112017020046A2 (pt) | 2018-06-05 |
| EP3286189B1 (en) | 2021-05-26 |
| GB201507036D0 (en) | 2015-06-10 |
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