KR20160095035A - 알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법 - Google Patents

알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법 Download PDF

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KR20160095035A
KR20160095035A KR1020167017707A KR20167017707A KR20160095035A KR 20160095035 A KR20160095035 A KR 20160095035A KR 1020167017707 A KR1020167017707 A KR 1020167017707A KR 20167017707 A KR20167017707 A KR 20167017707A KR 20160095035 A KR20160095035 A KR 20160095035A
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compound
pharmaceutically acceptable
acceptable salt
administered
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Korean (ko)
Inventor
엠마누엘 디 토마소
마리-캐롤린 게르마
크리스티안 마사세시
크리스틴 프리치
크리스티안 렌 슈넬
란자나 타보라스
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노파르티스 아게
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Application filed by 노파르티스 아게 filed Critical 노파르티스 아게
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/427—Thiazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

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  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020167017707A 2013-12-06 2014-12-03 알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법 Ceased KR20160095035A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13306679 2013-12-06
EP13306679.5 2013-12-06
PCT/IB2014/066558 WO2015083101A1 (en) 2013-12-06 2014-12-03 Dosage regimen for an alpha-isoform selective phosphatidylinositol 3-kinase inhibitor

Publications (1)

Publication Number Publication Date
KR20160095035A true KR20160095035A (ko) 2016-08-10

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ID=49876516

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KR1020167017707A Ceased KR20160095035A (ko) 2013-12-06 2014-12-03 알파-이소형 선택성 포스파티딜이노시톨 3-키나제 억제제를 위한 투여 요법

Country Status (22)

Country Link
US (4) US20170000778A1 (enExample)
EP (2) EP3076969B1 (enExample)
JP (1) JP2016539149A (enExample)
KR (1) KR20160095035A (enExample)
CN (1) CN105979947A (enExample)
AU (2) AU2014358773A1 (enExample)
BR (1) BR112016011811A2 (enExample)
CA (1) CA2930359C (enExample)
CL (1) CL2016001361A1 (enExample)
DK (1) DK3076969T3 (enExample)
ES (1) ES2899167T3 (enExample)
HU (1) HUE057092T2 (enExample)
IL (1) IL245709B (enExample)
MX (1) MX378409B (enExample)
PH (1) PH12016501026A1 (enExample)
PL (1) PL3076969T3 (enExample)
PT (1) PT3076969T (enExample)
RU (1) RU2680246C1 (enExample)
SI (1) SI3076969T1 (enExample)
TN (1) TN2016000179A1 (enExample)
TW (1) TWI666019B (enExample)
WO (1) WO2015083101A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20180073674A (ko) * 2015-11-02 2018-07-02 노파르티스 아게 포스파티딜이노시톨 3-키나제 억제제에 대한 투여 요법
WO2018060833A1 (en) * 2016-09-27 2018-04-05 Novartis Ag Dosage regimen for alpha-isoform selective phosphatidylinositol 3-kinase inhibitor alpelisib
GB202010627D0 (en) * 2020-07-10 2020-08-26 Qbd (Qs-Ip) Ltd Blocking method

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Also Published As

Publication number Publication date
IL245709A0 (en) 2016-07-31
SI3076969T1 (sl) 2021-12-31
MX378409B (es) 2025-03-10
JP2016539149A (ja) 2016-12-15
EP3076969A1 (en) 2016-10-12
PL3076969T3 (pl) 2022-01-17
EP3076969B1 (en) 2021-09-01
TN2016000179A1 (en) 2017-10-06
CN105979947A (zh) 2016-09-28
EP4000619A1 (en) 2022-05-25
HK1223549A1 (zh) 2017-08-04
WO2015083101A1 (en) 2015-06-11
US20170000778A1 (en) 2017-01-05
CA2930359C (en) 2022-03-01
CA2930359A1 (en) 2015-06-11
DK3076969T3 (da) 2021-11-22
TWI666019B (zh) 2019-07-21
IL245709B (en) 2021-03-25
CL2016001361A1 (es) 2017-02-10
BR112016011811A2 (pt) 2017-08-08
AU2017245292B2 (en) 2018-09-27
HUE057092T2 (hu) 2022-04-28
US10434092B2 (en) 2019-10-08
US20210196696A1 (en) 2021-07-01
MX2016007376A (es) 2017-05-11
RU2680246C1 (ru) 2019-02-19
AU2014358773A1 (en) 2016-06-02
PT3076969T (pt) 2021-11-23
TW201609096A (zh) 2016-03-16
ES2899167T3 (es) 2022-03-10
AU2017245292A1 (en) 2017-11-02
PH12016501026A1 (en) 2016-07-04
US20200069670A1 (en) 2020-03-05
US20180078540A1 (en) 2018-03-22

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