KR20160083950A - N-(4-클로로-2-하이드록시-3-((3s)-3-피페리디닐설포닐)페닐-n′-(3-플루오로-2-메틸페닐)우레아의 하이드로브로마이드 염 - Google Patents
N-(4-클로로-2-하이드록시-3-((3s)-3-피페리디닐설포닐)페닐-n′-(3-플루오로-2-메틸페닐)우레아의 하이드로브로마이드 염 Download PDFInfo
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- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- A61K31/4462—Non condensed piperidines, e.g. piperocaine only substituted in position 3
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB1320021.7A GB201320021D0 (en) | 2013-11-13 | 2013-11-13 | Novel Compounds |
| GB1320021.7 | 2013-11-13 | ||
| PCT/EP2014/074222 WO2015071235A1 (en) | 2013-11-13 | 2014-11-11 | Hydrobromide salt ofn-(4-chloro-2-hydroxy-3-((3s)-3-piperidinylsulfonyl)phenyl-n'-(3-fluoro-2-methylphenyl)urea |
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| KR20160083950A true KR20160083950A (ko) | 2016-07-12 |
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| US (3) | US9809540B2 (OSRAM) |
| EP (1) | EP3068763B1 (OSRAM) |
| JP (1) | JP6401265B2 (OSRAM) |
| KR (1) | KR20160083950A (OSRAM) |
| CN (1) | CN105683162A (OSRAM) |
| AU (1) | AU2014350334B2 (OSRAM) |
| BR (1) | BR112016010409A8 (OSRAM) |
| CA (1) | CA2929907A1 (OSRAM) |
| CY (1) | CY1121581T1 (OSRAM) |
| DK (1) | DK3068763T3 (OSRAM) |
| ES (1) | ES2714721T3 (OSRAM) |
| GB (1) | GB201320021D0 (OSRAM) |
| HR (1) | HRP20190449T1 (OSRAM) |
| HU (1) | HUE041873T2 (OSRAM) |
| LT (1) | LT3068763T (OSRAM) |
| ME (1) | ME03328B (OSRAM) |
| PL (1) | PL3068763T3 (OSRAM) |
| PT (1) | PT3068763T (OSRAM) |
| RS (1) | RS58382B1 (OSRAM) |
| RU (1) | RU2685408C1 (OSRAM) |
| SI (1) | SI3068763T1 (OSRAM) |
| SM (1) | SMT201900156T1 (OSRAM) |
| TR (1) | TR201902981T4 (OSRAM) |
| WO (1) | WO2015071235A1 (OSRAM) |
Families Citing this family (3)
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| WO2015173701A2 (en) * | 2014-05-12 | 2015-11-19 | Glaxosmithkline Intellectual Property (No. 2) Limited | Pharmaceutical compositions for treating infectious diseases |
| RU2018123711A (ru) | 2015-11-30 | 2020-01-09 | Глэксосмитклайн Интеллекчуал Проперти (Но.2) Лимитед | Композиции для внутривенного введения |
| WO2018073248A1 (en) | 2016-10-17 | 2018-04-26 | Icm (Institut Du Cerveau Et De La Moelle Épinière) | Prognosis of demyelinating diseases patients and treatment thereof |
Family Cites Families (1)
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| AU2007240365B2 (en) | 2006-04-21 | 2011-12-15 | Glaxosmithkline Llc | IL-8 receptor antagonists |
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- 2014-11-11 EP EP14799988.2A patent/EP3068763B1/en active Active
- 2014-11-11 SM SM20190156T patent/SMT201900156T1/it unknown
- 2014-11-11 HU HUE14799988A patent/HUE041873T2/hu unknown
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- 2014-11-11 RU RU2016116955A patent/RU2685408C1/ru not_active IP Right Cessation
- 2014-11-11 RS RS20190230A patent/RS58382B1/sr unknown
- 2014-11-11 CA CA2929907A patent/CA2929907A1/en not_active Abandoned
- 2014-11-11 CN CN201480061455.2A patent/CN105683162A/zh active Pending
- 2014-11-11 TR TR2019/02981T patent/TR201902981T4/tr unknown
- 2014-11-11 PT PT14799988T patent/PT3068763T/pt unknown
- 2014-11-11 LT LTEP14799988.2T patent/LT3068763T/lt unknown
- 2014-11-11 BR BR112016010409A patent/BR112016010409A8/pt not_active IP Right Cessation
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2017
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2018
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2019
- 2019-02-26 CY CY20191100237T patent/CY1121581T1/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP3068763B1 (en) | 2018-12-19 |
| EP3068763A1 (en) | 2016-09-21 |
| SMT201900156T1 (it) | 2019-05-10 |
| PT3068763T (pt) | 2019-03-20 |
| CA2929907A1 (en) | 2015-05-21 |
| CY1121581T1 (el) | 2020-05-29 |
| ME03328B (me) | 2019-10-20 |
| US20160264525A1 (en) | 2016-09-15 |
| DK3068763T3 (en) | 2019-03-18 |
| ES2714721T3 (es) | 2019-05-29 |
| HUE041873T2 (hu) | 2019-05-28 |
| RS58382B1 (sr) | 2019-04-30 |
| AU2014350334A1 (en) | 2016-06-02 |
| AU2014350334B2 (en) | 2017-08-10 |
| GB201320021D0 (en) | 2013-12-25 |
| CN105683162A (zh) | 2016-06-15 |
| RU2016116955A (ru) | 2017-12-19 |
| WO2015071235A1 (en) | 2015-05-21 |
| PL3068763T3 (pl) | 2019-05-31 |
| US20190112269A1 (en) | 2019-04-18 |
| JP2016537344A (ja) | 2016-12-01 |
| TR201902981T4 (tr) | 2019-03-21 |
| US10604485B2 (en) | 2020-03-31 |
| JP6401265B2 (ja) | 2018-10-10 |
| US20180079722A1 (en) | 2018-03-22 |
| HRP20190449T1 (hr) | 2019-04-19 |
| BR112016010409A8 (pt) | 2020-04-22 |
| US9809540B2 (en) | 2017-11-07 |
| RU2685408C1 (ru) | 2019-04-18 |
| LT3068763T (lt) | 2019-03-12 |
| SI3068763T1 (sl) | 2019-04-30 |
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