KR20150127246A - 류코트라이엔 a4 가수분해효소의 저해제 - Google Patents

류코트라이엔 a4 가수분해효소의 저해제 Download PDF

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KR20150127246A
KR20150127246A KR1020157028772A KR20157028772A KR20150127246A KR 20150127246 A KR20150127246 A KR 20150127246A KR 1020157028772 A KR1020157028772 A KR 1020157028772A KR 20157028772 A KR20157028772 A KR 20157028772A KR 20150127246 A KR20150127246 A KR 20150127246A
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윌리엄 길퍼드
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켈탁시스, 인코퍼레이티드
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Neurosurgery (AREA)
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  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
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  • Communicable Diseases (AREA)
  • Transplantation (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Otolaryngology (AREA)
KR1020157028772A 2013-03-14 2014-03-14 류코트라이엔 a4 가수분해효소의 저해제 Ceased KR20150127246A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361781193P 2013-03-14 2013-03-14
US61/781,193 2013-03-14
PCT/US2014/027428 WO2014152518A2 (en) 2013-03-14 2014-03-14 Inhibitors of leukotriene a4 hydrolase

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KR20150127246A true KR20150127246A (ko) 2015-11-16

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US (2) US9777006B2 (enExample)
EP (1) EP2970309A4 (enExample)
JP (1) JP6534650B2 (enExample)
KR (1) KR20150127246A (enExample)
AU (1) AU2014239567B2 (enExample)
BR (1) BR112015022864A8 (enExample)
CA (1) CA2906084A1 (enExample)
MX (1) MX2015011678A (enExample)
RU (1) RU2678196C2 (enExample)
WO (1) WO2014152518A2 (enExample)

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